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Search Result

Search Results for " neurokinin receptor "

Targets

Neurokinin receptor Endogenous Metabolite Neurokinin receptor

90

Compounds

1

Natural Products

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
TP1087 Substance P Neurokinin P Endogenous Metabolite , Neurokinin receptor
Substance P (Neurokinin P) (SP) is an undecapeptide (a peptide composed of a chain of 11 amino acid residues) member of the tachykinin neuropeptide family.
TP1008 Neurokinin A α-Neurokinin,Substance K,Neuromedin L Neurokinin receptor
Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.
T7633 Senktide Neurokinin receptor
Senktide is an agonist of tachykinin NK3 receptor.
T23316 SB 218795 Neurokinin receptor
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
T16849 SB-222200 Neurokinin receptor
SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
TP1086 Men 10376 TFA(135306-85-3,free) Men 10376 TFA,Neurokinin-2 receptor antagonist TFA Neurokinin receptor
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats.
T7209 Maropitant Neurokinin receptor
Maropitant is a selective neurokinin (NK1) receptor antagonist.
TP1572 GR-73632 Neurokinin receptor
Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).
T38144 Elinzanetant Neurokinin receptor
Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.
T15278 Fezolinetant ESN-364 Neurokinin receptor
Fezolinetant (ESN-364) is an antagonist of the neurokinin 3 receptor (NK3R). It is used for the treatment of menopausal hot flushes.
T7549 Talnetant SB 223412 Neurokinin receptor
Talnetant (SB 223412) is a selective, competitive, brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission
T76429 Neurokinin Receptor (393-407), rat
Neurokinin Receptor (393-407), rat (SPR393–407), a fragment of the rat neurokinin 1 receptor (NK1R), undergoes rapid endocytosis and subsequent recycling to the plasma membrane upon substance P (SP) binding. This compoun...
T8235 L-732138 Neurokinin receptor
L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)
TP1883 [Lys5,MeLeu9,Nle10]-NKA(4-10) Neurokinin receptor
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
T17156 Tradipitant VLY-686,LY686017 Neurokinin receptor
Tradipitant (VLY-686) is an antagonist of neurokinin-1.
T7554 Substance P (7-11) Substance P 7-11(TFA) Others , Neurokinin receptor
Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .
T16038 Men 10376 Neurokinin-2 receptor antagonist CDK
Men 10376 is a selective antagonist of tachykinin NK-2 receptor. It has a Ki of 4.4 μM for rat small intestine NK-2 receptor.
T6905 Netupitant Ro 67-31898/000,CID 6451149 Neurokinin receptor
Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).
T3716 Rolapitant SCH619734 Neurokinin receptor
Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. ...
T7559 Neurokinin A(4-10) Neurokinin A(4-10)(TFA) Neurokinin receptor
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
T1743 Aprepitant MK-869,MK-0869,L-754030,Aprepitant` HIV Protease , Antibacterial , Antibiotic , Neurokinin receptor
Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist. The mechanism of action of aprepitant is as a Neurokinin 1 Antagonist, and Cytochrome P450 3A4 Inhibitor, and Cytochrome P450 2C9 Inducer, and C...
T13306L Vapreotide acetate RC-160 acetate,BMY-41606 acetate Neurokinin receptor
Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).
T1790 Fosaprepitant dimeglumine L785298,MK-0517,Fosaprepitant dimeglumine salt Neurokinin receptor
Fosaprepitant dimeglumine (MK-0517) is the dimeglumine salt form of fosaprepitant, the water-soluble, N-phosphorylated prodrug of aprepitant, with antiemetic activity. Upon intravenous administration and rapid conversion...
T3034 Eprazinone dihydrochloride Resplen,Mucitux,Eftapan,NSC 317935,Eprazinone 2HCl Others , Neurokinin receptor
Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.
T7828 [Sar9,Met(O2)11]-Substance P Bhsar-sp,NA Neurokinin receptor
[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.
T7396 Substance P(1-7) Substance P 1-7 Others , Neurokinin receptor
Substance P(1-7) (Substance P 1-7) is the major bioactive metabolite formed after proteolytic degradation of the tachykinin substance P (SP),with anti-inflammatory, anti-nociceptive and anti-hyperalgesic effects
T7631 Eledoisin Related Peptide Eledoisin RP,Eledoisin-Related Peptide,Eledoisin Related Peptide(2TFA) Neurokinin receptor
Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.
TP1363L Neurokinin B acetate(86933-75-7 free base) Neurokinin K Neurokinin receptor
Neurokinin B acetate(86933-75-7 free base) is the acetate form of Neurokinin B, which belongs to the tachykinin family. Neurokinin binds to neurokinin receptor 1 (NK1R), nk2r and NK3R, and mediates its biological effects...
TP1385 Neurokinin A(4-10) TFA(97559-35-8 free base) Neurokinin A(4-10) TFA Neurokinin receptor
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].
T68068 Ezlopitant CJ 11974,CJ-11974,CJ11974 Neurokinin receptor
Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.
T69140 Burapitant SSR 240600 Neurokinin receptor
Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.
T68068L (R)-CJ 11974 Neurokinin receptor
(R)-CJ 11974 is a novel non-peptide neurokinin NK1 substance P receptor antagonist with potential analgesic activity that can be used to study chemotherapy-induced vomiting.
TP1851L Scyliorhinin II acetate Neurokinin receptor
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.
T19518L Physalaemin acetate Neurokinin receptor
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.
T25616 Lanepitant 2HCl LY303870 dihydrochloride,LY 303870 dihydrochloride,LY-303870 dihydrochloride,Lanepitant dihydrochloride Neurokinin receptor
Lanepitant 2HCl is a non-peptide neurokinin-1 receptor antagonist with analgesic and anti-inflammatory activity.Lanepitant 2HCl inhibits the binding of Substance P to the neurokinin-1 receptor, inhibits neurogenic inflam...
T16114 Pavinetant AZD4901,MLE-4901,AZD2624 MEK
Pavinetant is a small molecule orally active and selective neurokinin-3 (NK3) receptor antagonist for the treatment of hot flashes and polycystic ovarian syndrome (PCOS), which is a potential compound for the treatment o...
T3724 Rolapitant hydrochloride Rolapitant HCl Neurokinin receptor
Rolapitant (SCH619734) hydrochloride is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a K i of 0.66 nM. Rolapitant hydrochloride (Rolapitant HCl) does not interact with CY...
T9417L Gamma-preprotachykinin amide (72-92) acetate gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base) Others
gamma-preprotachykinin amide (72-92) acetate is a 21 amino acid peptide belonging to the tachykinin (TK) family and including neurokinin A (NKA) in its C-terminal sequence. gamma-preprotachykinin amide (72-92) acetate po...
T68556 GW679769
GW679769 is a neurokinin-1 receptor antagonist.
T20148 L 659,877 L 659877,L-659,877,L-659877,L659,877,L659877
L 659,877 is an antagonist of the Tachykinin and neurokinin-2 receptor.
T70587 CJ-12255
CJ-12255 is a Neurokinin-1 Receptor Antagonist.
T76427 (D-Pro2,D-Trp6,8,Nle10)-Neurokinin B
(D-Pro2,D-Trp6,8,Nle10)-Neurokinin B functions as a competitive antagonist to the Neurokinin B receptor, exhibiting a pA2 value of 5.5. Notably, it does not affect Substance P or Neurokinin A [1].
T69295 DNK 333
DNK 333 is a dual neurokinin NK1/NK2 receptor antagonist.
T34799 Telmapitant
Telmapitant is an antagonist of the neurokinin NK1 receptor.
T29210 ZD6021 ZD-6021,ZD 6021
ZD6021 is an antagonist of neurokinin 1 receptor.
T16406 Orvepitant maleate GW823296 maleate Neurokinin receptor
Orvepitant maleate is an effective, selective, and well-tolerated neurokinin-1 receptor (NK-1) antagonist (pKi: 10.2 for human neurokinin-1 receptor). Orvepitant maleate has the potential for depressive disorder and chro...
T27175 Dilopetine Citrate E-6006 Citrate,E-6039,E6039,E 6039
Dilopetine Citrate, a tachykinin receptor modulator and a neurokinin receptor modulator, is used potentially for the treatment of depression.
T24359 L 743310 L-743310,L743310,L743,310,L 743,310,L-743,310
L 743310 is an antagonist of the neurokinin-1 receptor.
T24447 Men 10208 Men-10208,Thr-asp-tyr-trp-val-trp-trp-arg-NH2,Men10208
Men 10208 is an antagonist of the neurokinin A receptor.
T29157 WIN 51,708 WIN51,708,WIN-51,708
WIN 51,708 is an antagonist of neurokinin-1 receptor.

Compounds

Substance P
TP1087
Synonym: Neurokinin P
Target: Endogenous Metabolite, Neurokinin receptor
Neurokinin A
TP1008
Synonym: α-Neurokinin,Substance K,Neuromedin L
Target: Neurokinin receptor
Senktide
T7633
Synonym:
Target: Neurokinin receptor
SB 218795
T23316
Synonym:
Target: Neurokinin receptor
SB-222200
T16849
Synonym:
Target: Neurokinin receptor
Men 10376 TFA(135306-85-3,free)
TP1086
Synonym: Men 10376 TFA,Neurokinin-2 receptor antagonist TFA
Target: Neurokinin receptor
Maropitant
T7209
Synonym:
Target: Neurokinin receptor
GR-73632
TP1572
Synonym:
Target: Neurokinin receptor
Elinzanetant
T38144
Synonym:
Target: Neurokinin receptor
Fezolinetant
T15278
Synonym: ESN-364
Target: Neurokinin receptor
Talnetant
T7549
Synonym: SB 223412
Target: Neurokinin receptor
Neurokinin Receptor (393-407), rat
T76429
Synonym:
Target:
L-732138
T8235
Synonym:
Target: Neurokinin receptor
[Lys5,MeLeu9,Nle10]-NKA(4-10)
TP1883
Synonym:
Target: Neurokinin receptor
Tradipitant
T17156
Synonym: VLY-686,LY686017
Target: Neurokinin receptor
Substance P (7-11)
T7554
Synonym: Substance P 7-11(TFA)
Target: Others, Neurokinin receptor
Men 10376
T16038
Synonym: Neurokinin-2 receptor antagonist
Target: CDK
Netupitant
T6905
Synonym: Ro 67-31898/000,CID 6451149
Target: Neurokinin receptor
Rolapitant
T3716
Synonym: SCH619734
Target: Neurokinin receptor
Neurokinin A(4-10)
T7559
Synonym: Neurokinin A(4-10)(TFA)
Target: Neurokinin receptor
Aprepitant
T1743
Synonym: MK-869,MK-0869,L-754030,Aprepitant`
Target: HIV Protease, Antibacterial, Antibiotic, Neurokinin receptor
Vapreotide acetate
T13306L
Synonym: RC-160 acetate,BMY-41606 acetate
Target: Neurokinin receptor
Fosaprepitant dimeglumine
T1790
Synonym: L785298,MK-0517,Fosaprepitant dimeglumine salt
Target: Neurokinin receptor
Eprazinone dihydrochloride
T3034
Synonym: Resplen,Mucitux,Eftapan,NSC 317935,Eprazinone 2HCl
Target: Others, Neurokinin receptor
[Sar9,Met(O2)11]-Substance P
T7828
Synonym: Bhsar-sp,NA
Target: Neurokinin receptor
Substance P(1-7)
T7396
Synonym: Substance P 1-7
Target: Others, Neurokinin receptor
Eledoisin Related Peptide
T7631
Synonym: Eledoisin RP,Eledoisin-Related Peptide,Eledoisin Related Peptide(2TFA)
Target: Neurokinin receptor
Neurokinin B acetate(86933-75-7 free base)
TP1363L
Synonym: Neurokinin K
Target: Neurokinin receptor
Neurokinin A(4-10) TFA(97559-35-8 free base)
TP1385
Synonym: Neurokinin A(4-10) TFA
Target: Neurokinin receptor
Ezlopitant
T68068
Synonym: CJ 11974,CJ-11974,CJ11974
Target: Neurokinin receptor
Burapitant
T69140
Synonym: SSR 240600
Target: Neurokinin receptor
(R)-CJ 11974
T68068L
Synonym:
Target: Neurokinin receptor
Scyliorhinin II acetate
TP1851L
Synonym:
Target: Neurokinin receptor
Physalaemin acetate
T19518L
Synonym:
Target: Neurokinin receptor
Lanepitant 2HCl
T25616
Synonym: LY303870 dihydrochloride,LY 303870 dihydrochloride,LY-303870 dihydrochloride,Lanepitant dihydrochloride
Target: Neurokinin receptor
Pavinetant
T16114
Synonym: AZD4901,MLE-4901,AZD2624
Target: MEK
Rolapitant hydrochloride
T3724
Synonym: Rolapitant HCl
Target: Neurokinin receptor
gamma-preprotachykinin amide (72-92) acetate
T9417L
Synonym: gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base)
Target: Others
GW679769
T68556
Synonym:
Target:
L 659,877
T20148
Synonym: L 659877,L-659,877,L-659877,L659,877,L659877
Target:
CJ-12255
T70587
Synonym:
Target:
(D-Pro2,D-Trp6,8,Nle10)-Neurokinin B
T76427
Synonym:
Target:
DNK 333
T69295
Synonym:
Target:
Telmapitant
T34799
Synonym:
Target:
ZD6021
T29210
Synonym: ZD-6021,ZD 6021
Target:
Orvepitant maleate
T16406
Synonym: GW823296 maleate
Target: Neurokinin receptor
Dilopetine Citrate
T27175
Synonym: E-6006 Citrate,E-6039,E6039,E 6039
Target:
L 743310
T24359
Synonym: L-743310,L743310,L743,310,L 743,310,L-743,310
Target:
Men 10208
T24447
Synonym: Men-10208,Thr-asp-tyr-trp-val-trp-trp-arg-NH2,Men10208
Target:
WIN 51,708
T29157
Synonym: WIN51,708,WIN-51,708
Target:
1 2
Cat No. Product Name Synonyms Targets
T8789 N-Acetyl-L-tryptophan N-acetyltryptophan Endogenous Metabolite , Neurokinin receptor
N-Acetyl-L-tryptophan (N-acetyltryptophan) is an inhibitor of neurokinin 1 receptor (NK1-receptor, NK1R).

Natural Products

N-Acetyl-L-tryptophan
T8789
Synonym: N-acetyltryptophan
Target: Endogenous Metabolite, Neurokinin receptor

Recombinant Proteins

Species：
Human (1)
Expression System：
E. coli (1)
Tag：
N-6His (1)
Cat No. Product Name Species Expression System
TMPJ-01379 TAC3 Protein, Human, Recombinant (His) Human E. coli
Tachykinin 3 (TAC3) is a secreted protein that belongs to the Tachykinin family. Tachykinins are active peptides that excite neurons and evoke behavioral responses; they are potent vasodilators and secretagogues, and con...
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