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Search Results for " glucocorticoid-receptor "

Targets

100

Compounds

15

Natural Products

12

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T37908 Glucocorticoid receptor agonist-1 Glucocorticoid Receptor
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].
T11417 Glucocorticoid receptor agonist Others
Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.
T67742 EX-A5386 Glucocorticoid receptor modulator-1 Glucocorticoid Receptor
EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.
T74697 Glucocorticoid receptor agonist-2
Glucocorticoid receptor agonist-2 (compound 21) is an glucocorticoid receptor agonist with an IC 50 value of 6.6 nM. Glucocorticoid receptor agonist-2 can be used to synthesize anti-inflammatory ADC molecules. Glucocorti...
T72102 Glucocorticoid receptor modulator 1
Glucocorticoid receptor modulator 1 is a highly potent and orally active non-steroidal selective glucocorticoid receptor modulator with an IC 50 value of 9 nM and 130 nM for NF-κB and AP-1 , respectively. Glucocorticoid ...
T63551 Glucocorticoid receptor-IN-1
Glucocorticoid receptor-IN-1 is a selective regulator of the glucocorticoid receptor (GR) and exhibits anti-inflammatory activity. glucocorticoid receptor-IN-1 has good transcriptional repression, acting on hMMP1 ( IC50:...
T63539 Glucocorticoid receptor-IN-2
Glucocorticoid receptor-IN-2 is a selective regulator of the glucocorticoid receptor (GR) and exhibits anti-inflammatory activity. IC50: 0.171 nM) and also has some transcriptional activating effect on MMTV (EC50: 0.94 n...
T8777 Beclometasone BecloMethasone Glucocorticoid Receptor
Beclometasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma.
T15451 GW-870086 Glucocorticoid Receptor
GW-870086 is an effective anti-inflammatory agent. GW-870086 also plays a role in a glucocorticoid receptor agonist (pIC50: 10.1 in A549 cells expressing NF-κB).
T14377 AZD5423 Glucocorticoid Receptor
AZD5423 is an inhaled, potent, selective, and non-steroidal modulator of glucocorticoid receptor (GR) and it effectively reduces allergen-induced responses in subjects with mild allergic asthma.
T14981 Clobetasone butyrate Glucocorticoid Receptor
Clobetasone butyrate can be used to relieve corticosteroid-responsive dermatoses, including atopic dermatitis and psoriasis. Clobetasone butyrate is a synthetic glucocorticoid. It has topical anti-inflammatory activity e...
T17217 Vamorolone VBP15 Glucocorticoid Receptor , NF-κB
Vamorolone (VBP15) is an orally active dissociative steroidal anti-inflammatory drug and membrane-stabilizer. Vamorolone improves muscular dystrophy without side effects. Vamorolone displays effective NF-κB inhibition an...
T77869 Glucocorticoid receptor agonist-2 Ala-Ala-Mal
Glucocorticoid receptor agonist-2 Ala-Ala-Mal (compound 79) serves as a precursor for synthesizing anti-inflammatory antibody-drug conjugate (ADC) molecules and acts as an active reference for ABBV-3373 [1].
T74116 Glucocorticoid receptor agonist-1 Ala-Ala-Mal
Glucocorticoid receptor agonist-1 Ala-Ala-Mal (compound 88) is a glucocorticosteroid, and an agonist of glucocorticoid receptor . Glucocorticoid receptor agonist-1 Ala-Ala-Mal can be conjugated with Adalimumab to prepar...
T0820 Triamcinolone acetonide Aristogel,Azmacort,Aristoderm Glucocorticoid Receptor
Triamcinolone acetonide (Azmacort) is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as a Corticosteroid Hormone Receptor Agonist. It is an anti-inflammatory glucocorticoid used topically in the ...
T75016 Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal
Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal is a glucocorticoid receptor agonist. Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal can be used in anti-CD40 antibody agent conjugate (ADC) . Glucocortico...
T77835 Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Br
Glucocorticoid Receptor Agonist-1 Phosphate (Gly-Glu-Br) is an antibody-drug conjugate (ADC) linker utilized in the synthesis of ABBV-154, ABBV-927, ABBV-368, and related analogs [1].
T75130 Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br
Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br is an Drug-linker conjugates for ADC that can be used as a reaction reagent for the synthesis of anti-CD40 antibody agent conjugates ( ADCs ) [1] .
T6502 Fluocinonide Lidex,Metosyn,Topsyn Glucocorticoid Receptor
Fluocinonide (Topsyn) (Vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent.
T82303 Glucocorticoid receptor agonist-1 phosphate Gly-Glu TFA
Glucocorticoid Receptor Agonist-1 Phosphate Gly-Glu (TFA) serves as a cleavable linker for the synthesis of Antibody-Drug Conjugates (ADCs).
T1163 Betamethasone valerate Betnovate,Betaderm,Betamethasone 17-valerate,Luxiq Glucocorticoid Receptor
Betamethasone valerate (Luxiq) is a synthetic glucocorticoid with metabolic, immunosuppressive and anti-inflammatory actions.
T0261 Amcinonide CL-34699 Glucocorticoid Receptor , Annexin A
Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.
T8396 Prednisone acetate Prednisone 21-acetate Glucocorticoid Receptor
Prednisone acetate (Prednisone 21-acetate) is a glucocorticoid receptor agonist with immunomodulating properties and anti-inflammatory.
T0367 Fluocinolone (Acetonide) Fluocinolone acetonide,Flucort-N Glucocorticoid Receptor
Fluocinolone Acetonide (Flucort-N) is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion, or ointment. It has also been used topically in...
T3316 Fluorometholone Fluoromethalone,Cortilet,Oxylone,Delmeson Glucocorticoid Receptor
Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery. It is marketed under the brand names FML (Allergan) and Flarex (Alcon). Fluorometholone acetate ophthalmic susp...
T0181 Loteprednol etabonate Lotemax,Alrex Glucocorticoid Receptor , Antibacterial , Antibiotic
Loteprednol etabonate (Lotemax) is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.
T1076 Dexamethasone MK 125,Prednisolone F,NSC 34521,Hexadecadrol Glucocorticoid Receptor , Mitophagy , IL Receptor , SARS-CoV , Antibacterial , Antibiotic , Autophagy , Complement System
Dexamethasone (Hexadecadrol) is a glucocorticoid receptor agonist and an IL receptor modulator. Dexamethasone has anti-inflammatory and immunosuppressive activity and induces autophagy. Dexamethasone inhibits LPS-induced...
T1749 AL 082D06 D-06,AL082D06 Glucocorticoid Receptor
AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR(Ki > 10 uM).
T6713 Ulipristal Estrogen/progestogen Receptor , Progesterone Receptor
Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.
TQ0225 Velsecorat AZD7594,AZ13189620 Glucocorticoid Receptor
Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).
T2526 Ciclesonide Zetonna,RPR251526,Omnaris,Alvesco Glucocorticoid Receptor
Ciclesonide (Alvesco)(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.
T0094 Budesonide Entocort,Pulmicort,Rhinocort Glucocorticoid Receptor
Budesonide (Pulmicort), an anti-inflammatory corticosteroid, has shown the effective glucocorticoid activitie and few mineralocorticoid activities. According to reports, Budesonide has extensively inhibitory effects agai...
T1531 Mometasone furoate Sch32088 Glucocorticoid Receptor
Mometasone furoate (Sch32088) is a pregnadienediol derivative ANTI-ALLERGIC AGENT and ANTI-INFLAMMATORY AGENT that is used in the management of ASTHMA and ALLERGIC RHINITIS. It is also used as a topical treatment for ski...
T22367 Methylprednisolone succinate Methylprednisolone hemisuccinate,Methylprednisolone hydrogen succinate Glucocorticoid Receptor
Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory agent.
T21404 Fluticasone furoate Veramyst,Allermist,Avamys,Fluticasone furoate Glucocorticoid Receptor
Fluticasone furoate (Avamys) is a synthetic trifluorinated corticosteroid derived from fluticasone with a Kd of 0.3 nM. Fluticasone furoate has potent anti-inflammatory, anti-asthmatic activity, and low systemic exposure...
T6580 Meprednisone SCH 4358,Methylprednisone,NSC 527579,Betanisona,Betapar Glucocorticoid Receptor , Autophagy
Betapar(Meprednisone (Betapar)) is a glucocorticoid and a methylated derivative of prednisone.
T2527 Ulipristal acetate Ulipristal,CDB-2914 Estrogen/progestogen Receptor , Progesterone Receptor , Autophagy
Ulipristal acetate (CDB-2914) is an orally bioavailable, acetate salt of ulipristal, a selective progesterone receptor modulator with anti-progesterone activity. Ulipristal binds to the progesterone receptor (PR), thereb...
T1102 Mifepristone C-1073,RU486,RU 38486 Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , NO Synthase , Autophagy
Mifepristone (C-1073) is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist.
T16079 Mirodenafil SK3530 PDE
Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.
T1127 Beclometasone dipropionate Beclovent,Beclomethasone dipropionate,Beconase,Vancenase Glucocorticoid Receptor
Beclometasone dipropionate (Vancenase) is the dipropionate ester of a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. After cell surface receptor attachment and cell entry, beclomethasone...
T0947L Dexamethasone Phosphate disodium EGP-437,EGP437. Dex-Phos,EGP 437 Glucocorticoid Receptor
Dexamethasone Phosphate disodium (EGP437. Dex-Phos) is a water-soluble form of the synthetic glucocorticoid dexamethasone.
T0208 Prednisolone disodium phosphate Prednisolone phosphate sodium,Prednisolone 21-phosphate disodium Glucocorticoid Receptor
Prednisolone disodium phosphate, a synthetic glucocorticoid, has immunomodulating and anti-inflammatory properties.
T0188 Fluticasone (propionate) CCI-187881,Fluticasone propionate Glucocorticoid Receptor , Virus Protease , Estrogen/progestogen Receptor , Phospholipase , Endogenous Metabolite
Fluticasone propionate (CCI-187881), derived from fluticasone used to remedy asthma and allergic rhinitis, is a high affinity, selective GR (glucocorticoid receptor) agonist.
T1559 Betamethasone dipropionate Diprolene AF,SCH 11460,Betamethasone 17,21-dipropionate,Diprolene,Diprosone Glucocorticoid Receptor
Betamethasone Dipropionate is the 17, 21-dipropionate ester of betamethasone, a synthetic glucocorticoid with metabolic, immunosuppressive and anti-inflammatory actions. Betamethasone dipropionate (SCH 11460) binds to sp...
T0947 Dexamethasone acetate Dexamethasone 21-acetate,Dexamethason acetate,NSC 39471 Glucocorticoid Receptor , Mitophagy , IL Receptor , Annexin A , NOS , Antibacterial , Autophagy
Dexamethasone acetate (NSC 39471) is the acetate salt form of Dexamethasone, a synthetic adrenal corticosteroid with potent anti-inflammatory properties. In addition to binding to specific nuclear steroid receptors, dexa...
TQ0126 Mirodenafil dihydrochloride SK-3530 dihydrochloride PDE
Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.
T4602 Hydrocortisone hemisuccinate Hydrocortisone 21-he,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate Glucocorticoid Receptor , Others , Interleukin
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.
T1573 Flunisolide Rhinalar,Aerobid,Synaclyn Glucocorticoid Receptor
Flunisolide (Rhinalar) is a synthetic corticosteroid with anti-inflammatory and antiallergic properties.
T15102 Dexamethasone palmitate DXP Glucocorticoid Receptor
Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone, shows a 47-fold lower affinity for the glucocorticoid receptor than Dexamethasone. Dexamethasone palmitate is a glucocorticoid receptor agonist and an...
T34383 Rofleponide Glucocorticoid Receptor
Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.

Compounds

Glucocorticoid receptor agonist-1
T37908
Synonym:
Target: Glucocorticoid Receptor
Glucocorticoid receptor agonist
T11417
Synonym:
Target: Others
EX-A5386
T67742
Synonym: Glucocorticoid receptor modulator-1
Target: Glucocorticoid Receptor
Glucocorticoid receptor agonist-2
T74697
Synonym:
Target:
Glucocorticoid receptor modulator 1
T72102
Synonym:
Target:
Glucocorticoid receptor-IN-1
T63551
Synonym:
Target:
Glucocorticoid receptor-IN-2
T63539
Synonym:
Target:
Beclometasone
T8777
Synonym: BecloMethasone
Target: Glucocorticoid Receptor
GW-870086
T15451
Synonym:
Target: Glucocorticoid Receptor
AZD5423
T14377
Synonym:
Target: Glucocorticoid Receptor
Clobetasone butyrate
T14981
Synonym:
Target: Glucocorticoid Receptor
Vamorolone
T17217
Synonym: VBP15
Target: Glucocorticoid Receptor, NF-κB
Glucocorticoid receptor agonist-2 Ala-Ala-Mal
T77869
Synonym:
Target:
Glucocorticoid receptor agonist-1 Ala-Ala-Mal
T74116
Synonym:
Target:
Triamcinolone acetonide
T0820
Synonym: Aristogel,Azmacort,Aristoderm
Target: Glucocorticoid Receptor
Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal
T75016
Synonym:
Target:
Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Br
T77835
Synonym:
Target:
Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br
T75130
Synonym:
Target:
Fluocinonide
T6502
Synonym: Lidex,Metosyn,Topsyn
Target: Glucocorticoid Receptor
Glucocorticoid receptor agonist-1 phosphate Gly-Glu TFA
T82303
Synonym:
Target:
Betamethasone valerate
T1163
Synonym: Betnovate,Betaderm,Betamethasone 17-valerate,Luxiq
Target: Glucocorticoid Receptor
Amcinonide
T0261
Synonym: CL-34699
Target: Glucocorticoid Receptor, Annexin A
Prednisone acetate
T8396
Synonym: Prednisone 21-acetate
Target: Glucocorticoid Receptor
Fluocinolone (Acetonide)
T0367
Synonym: Fluocinolone acetonide,Flucort-N
Target: Glucocorticoid Receptor
Fluorometholone
T3316
Synonym: Fluoromethalone,Cortilet,Oxylone,Delmeson
Target: Glucocorticoid Receptor
Loteprednol etabonate
T0181
Synonym: Lotemax,Alrex
Target: Glucocorticoid Receptor, Antibacterial, Antibiotic
Dexamethasone
T1076
Synonym: MK 125,Prednisolone F,NSC 34521,Hexadecadrol
Target: Glucocorticoid Receptor, Mitophagy, IL Receptor, SARS-CoV, Antibacterial, Antibiotic, Autophagy, Complement System
AL 082D06
T1749
Synonym: D-06,AL082D06
Target: Glucocorticoid Receptor
Ulipristal
T6713
Synonym:
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Velsecorat
TQ0225
Synonym: AZD7594,AZ13189620
Target: Glucocorticoid Receptor
Ciclesonide
T2526
Synonym: Zetonna,RPR251526,Omnaris,Alvesco
Target: Glucocorticoid Receptor
Budesonide
T0094
Synonym: Entocort,Pulmicort,Rhinocort
Target: Glucocorticoid Receptor
Mometasone furoate
T1531
Synonym: Sch32088
Target: Glucocorticoid Receptor
Methylprednisolone succinate
T22367
Synonym: Methylprednisolone hemisuccinate,Methylprednisolone hydrogen succinate
Target: Glucocorticoid Receptor
Fluticasone furoate
T21404
Synonym: Veramyst,Allermist,Avamys,Fluticasone furoate
Target: Glucocorticoid Receptor
Meprednisone
T6580
Synonym: SCH 4358,Methylprednisone,NSC 527579,Betanisona,Betapar
Target: Glucocorticoid Receptor, Autophagy
Ulipristal acetate
T2527
Synonym: Ulipristal,CDB-2914
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Autophagy
Mifepristone
T1102
Synonym: C-1073,RU486,RU 38486
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, NO Synthase, Autophagy
Mirodenafil
T16079
Synonym: SK3530
Target: PDE
Beclometasone dipropionate
T1127
Synonym: Beclovent,Beclomethasone dipropionate,Beconase,Vancenase
Target: Glucocorticoid Receptor
Dexamethasone Phosphate disodium
T0947L
Synonym: EGP-437,EGP437. Dex-Phos,EGP 437
Target: Glucocorticoid Receptor
Prednisolone disodium phosphate
T0208
Synonym: Prednisolone phosphate sodium,Prednisolone 21-phosphate disodium
Target: Glucocorticoid Receptor
Fluticasone (propionate)
T0188
Synonym: CCI-187881,Fluticasone propionate
Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite
Betamethasone dipropionate
T1559
Synonym: Diprolene AF,SCH 11460,Betamethasone 17,21-dipropionate,Diprolene,Diprosone
Target: Glucocorticoid Receptor
Dexamethasone acetate
T0947
Synonym: Dexamethasone 21-acetate,Dexamethason acetate,NSC 39471
Target: Glucocorticoid Receptor, Mitophagy, IL Receptor, Annexin A, NOS, Antibacterial, Autophagy
Mirodenafil dihydrochloride
TQ0126
Synonym: SK-3530 dihydrochloride
Target: PDE
Hydrocortisone hemisuccinate
T4602
Synonym: Hydrocortisone 21-he,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate
Target: Glucocorticoid Receptor, Others, Interleukin
Flunisolide
T1573
Synonym: Rhinalar,Aerobid,Synaclyn
Target: Glucocorticoid Receptor
Dexamethasone palmitate
T15102
Synonym: DXP
Target: Glucocorticoid Receptor
Rofleponide
T34383
Synonym:
Target: Glucocorticoid Receptor
1 2
Cat No. Product Name Synonyms Targets
T1560 Prednisolone Predonine,Hydroretrocortine,Metacortandralone Glucocorticoid Receptor , Endogenous Metabolite
Prednisolone (Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
T1614 Hydrocortisone Cortisol Glucocorticoid Receptor , Endogenous Metabolite
Hydrocortisone (Cortisol) is a glucocorticoid hormone secreted by the adrenocortex. Hydrocortisone agonizes the glucocorticoid receptor, which promotes proteolytic metabolism, gluconeogenesis, capillary wall stabilizatio...
T1168 Desonide Tridesilon,Locapred,Prednacinolone Glucocorticoid Receptor
Desonide (Prednacinolone) is a synthetic glucocorticosteroid for topical use, with anti-inflammatory activity. Desonide binds to glucocorticoid receptors in the cytoplasm, and the ligand-receptor complex is translocated ...
T0798 Triamcinolone Fluoxyprednisolone,Aristocort,Rodinolone Glucocorticoid Receptor , COX
Triamcinolone (Aristocort) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. Upon cell entry, triamcinolone binds to and activates the glucocorticoid receptor, which leads to transloca...
T2810 (20S)-Protopanaxatriol 20(S)-APPT,g-PPT Apoptosis , Estrogen Receptor/ERR , Glucocorticoid Receptor , Estrogen/progestogen Receptor , Liver X Receptor
(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid receptor.
T2884 Cortisone Kendall's compound E,17-Hydroxy-11-dehydrocorticosterone Glucocorticoid Receptor , Endogenous Metabolite
Cortisone (17-Hydroxy-11-dehydrocorticosterone) is a corticosteroid with potent glucocorticoid activity.
T0034 Cortisone acetate Cortisone 21-acetate,NSC 49420 Glucocorticoid Receptor , Endogenous Metabolite
Cortisone Acetate is the acetate salt form of cortisone, a synthetic or semisynthetic analog of the naturally occurring cortisone hormone produced by the adrenal glands with anti-inflammatory and immunomodulating propert...
T1261 Medroxyprogesterone Acetate Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,Farlutin,Medroxyprogesterone (acetate) Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , Endogenous Metabolite
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally or by intramuscular injection and has also been...
T1243 Hydrocortisone acetate Cortisol 21-acetate,Hydrocortisone 21-acetate Glucocorticoid Receptor , Annexin A , Endogenous Metabolite
Hydrocortisone acetate (Cortisol 21-acetate) is the synthetic acetate salt form of hydrocortisone, a corticosteroid with anti-inflammatory and immunosuppressive properties.
T2748 Cortodoxone 11-Deoxycortisol,cortexolone,17α,21-dihydroxyprogesterone,Reichstein's substance S,11-Desoxycortisol Glucocorticoid Receptor , Endogenous Metabolite
Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.
T0948L Corticosterone 17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,Corticosterone (From plants) Glucocorticoid Receptor , Endogenous Metabolite
Corticosterone (Kendall's compound B) is a sensitive inhibitor of monoamine transport.
T1683 Actriol Epiestriol Glucocorticoid Receptor
Actriol (Epiestriol) is always used as Glucocorticoid Receptor agonist.
T6343 Geldanamycin NSC 122750 HSP , Influenza Virus , Tyrosine Kinases , Antibacterial , Antibiotic
Geldanamycin, an HSP90 inhibitor (Kd: 1.2 μM), specifically disrupts glucocorticoid receptor (GR)/HSP association.
T1429 17α-Hydroxyprogesterone Hydroxyprogesterone,17-OHP,17-Hydroxyprogesterone Estrogen/progestogen Receptor , Progesterone Receptor , Endogenous Metabolite
17α-Hydroxyprogesterone (17-OHP) is a physiological progestin that is produced during glucocorticoid and steroid hormone synthesis and is increased during the third trimester of pregnancy. Hydroxyprogesterone binds to th...
TN3537 Braylin IL Receptor , TNF , NF-κB
Braylin has anti-inflammatory, antinociceptive and immunomodulatory effects, which possibly act through the glucocorticoid receptor activation and by inhibition of the transcriptional activity of NF-κB. Braylin is also ...

Natural Products

Prednisolone
T1560
Synonym: Predonine,Hydroretrocortine,Metacortandralone
Target: Glucocorticoid Receptor, Endogenous Metabolite
Hydrocortisone
T1614
Synonym: Cortisol
Target: Glucocorticoid Receptor, Endogenous Metabolite
Desonide
T1168
Synonym: Tridesilon,Locapred,Prednacinolone
Target: Glucocorticoid Receptor
Triamcinolone
T0798
Synonym: Fluoxyprednisolone,Aristocort,Rodinolone
Target: Glucocorticoid Receptor, COX
(20S)-Protopanaxatriol
T2810
Synonym: 20(S)-APPT,g-PPT
Target: Apoptosis, Estrogen Receptor/ERR, Glucocorticoid Receptor, Estrogen/progestogen Receptor, Liver X Receptor
Cortisone
T2884
Synonym: Kendall's compound E,17-Hydroxy-11-dehydrocorticosterone
Target: Glucocorticoid Receptor, Endogenous Metabolite
Cortisone acetate
T0034
Synonym: Cortisone 21-acetate,NSC 49420
Target: Glucocorticoid Receptor, Endogenous Metabolite
Medroxyprogesterone Acetate
T1261
Synonym: Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,Farlutin,Medroxyprogesterone (acetate)
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, Androgen Receptor, Endogenous Metabolite
Hydrocortisone acetate
T1243
Synonym: Cortisol 21-acetate,Hydrocortisone 21-acetate
Target: Glucocorticoid Receptor, Annexin A, Endogenous Metabolite
Cortodoxone
T2748
Synonym: 11-Deoxycortisol,cortexolone,17α,21-dihydroxyprogesterone,Reichstein's substance S,11-Desoxycortisol
Target: Glucocorticoid Receptor, Endogenous Metabolite
Corticosterone
T0948L
Synonym: 17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,Corticosterone (From plants)
Target: Glucocorticoid Receptor, Endogenous Metabolite
Actriol
T1683
Synonym: Epiestriol
Target: Glucocorticoid Receptor
Geldanamycin
T6343
Synonym: NSC 122750
Target: HSP, Influenza Virus, Tyrosine Kinases, Antibacterial, Antibiotic
17α-Hydroxyprogesterone
T1429
Synonym: Hydroxyprogesterone,17-OHP,17-Hydroxyprogesterone
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite
Braylin
TN3537
Synonym:
Target: IL Receptor, TNF, NF-κB

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-06836 NR3C1 Protein, Human, Recombinant (His) Human E. coli
NR3C1 (Nuclear Receptor Subfamily 3 Group C Member 1) is a Protein Coding gene. This gene encodes glucocorticoid receptor, which can function both as a transcription factor that binds to glucocorticoid response elements ...
TMPJ-00110 GITR/TNFRSF18 Protein, Mouse, Recombinant (hFc & His) Mouse Human Cells
Tumor necrosis factor receptor superfamily member 18(Gitr) contains 3 TNFR-Cys repeats and it have four isforms.IsformA、isformB and isformC is single-pass type I membrane protein and isformD is a secreted protein. The p...
TMPH-00776 Griffithsin Protein, Griffithsia sp., Recombinant (X31S, His & Myc) Griffithsia sp. Baculovirus
Catalyzes the conversion of cortisol to the inactive metabolite cortisone. Modulates intracellular glucocorticoid levels, thus protecting the nonselective mineralocorticoid receptor from occupation by glucocorticoids.
TMPY-01117 MRAP Protein, Human, Recombinant (hFc) Human HEK293
MRAP (Melanocortin 2 Receptor Accessory Protein) is a Protein Coding gene. This gene encodes a melanocortin receptor-interacting protein. It belongs to the MRAP family. MRAP, which contains a single transmembrane domain,...
TMPK-00132 GITR/TNFRSF18 Protein, Human, Recombinant (aa 26-161, His & Avi), Biotinylated Human HEK293
GITR (glucocorticoid-induced tumor necrosis factor receptor), also known as AITR and TNFRSF18, is a 40 kDa transmembrane glycoprotein that functions in immune regulation.GIRT is a receptor for TNFSF18. Seems to be involv...
TMPK-00133 GITR/TNFRSF18 Protein, Human, Recombinant (aa 26-161, His) Human HEK293
GITR (glucocorticoid-induced tumor necrosis factor receptor), also known as AITR and TNFRSF18, is a 40 kDa transmembrane glycoprotein that functions in immune regulation.GIRT is a receptor for TNFSF18. Seems to be involv...
TMPY-03259 Calreticulin Protein, Human, Recombinant (His) Human HEK293
Calreticulin is a multifunctional protein. It acts as a main Ca(2+)-binding (storage) protein in the lumen of the endoplasmic reticulum. Calreticulin binds Ca2+ ions (a second messenger in signal transduction), rendering...
TMPK-01086 GITR/TNFRSF18 Protein, Mouse, Recombinant (aa 22-153, His) Mouse HEK293
GITR (glucocorticoid-induced tumor necrosis factor receptor), also known as AITR and TNFRSF18, is a 40 kDa transmembrane glycoprotein that functions in immune regulation.GIRT is a receptor for TNFSF18. Seems to be involv...
TMPK-01260 GITR/TNFRSF18 Protein, Cynomolgus, Recombinant (aa 20-156, His) Cynomolgus HEK293
GITR (glucocorticoid-induced tumor necrosis factor receptor), also known as AITR and TNFRSF18, is a 40 kDa transmembrane glycoprotein that functions in immune regulation.GIRT is a receptor for TNFSF18. Seems to be involv...
TMPY-03258 Calreticulin Protein, Human, Recombinant (hFc) Human HEK293
Calreticulin is a multifunctional protein. It acts as a main Ca(2+)-binding (storage) protein in the lumen of the endoplasmic reticulum. Calreticulin binds Ca2+ ions (a second messenger in signal transduction), rendering...
TMPY-06327 Calreticulin Protein, Human, Recombinant Human HEK293
Calreticulin is a multifunctional protein. It acts as a main Ca(2+)-binding (storage) protein in the lumen of the endoplasmic reticulum. Calreticulin binds Ca2+ ions (a second messenger in signal transduction), rendering...
TMPY-01383 PRMT6 Protein, Human, Recombinant (His & Flag) Human HEK293
Protein arginine N-methyltransferase 6, also known as Histone-arginine N-methyltransferase PRMT6, PRMT6, and HRMT1L6, is a member of the protein arginine N-methyltransferase family and PRMT6 subfamily. PRMT6 is highly ex...
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