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GPCR/G Protein GNRH Receptor

GNRH Receptor

The gonadotropin-releasing hormone receptor (GnRHR), also known as the luteinizing hormone releasing hormone receptor (LHRHR), is a member of the seven-transmembrane, G-protein coupled receptor (GPCR) family. It is the receptor of gonadotropin-releasing hormone (GnRH). The GnRHR is expressed on the surface of pituitary gonadotrope cells as well as lymphocytes, breast, ovary, and prostate.
Cat No. product name
T10988L Degarelix acetate(214766-78-6 free base) Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
TP1307 Buserelin Acetate (57982-77-1 free base) Buserelin Acetate is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
T3630 Relugolix Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential an...
T1494 Alarelin Alarelin acetate is a synthetic GnRH agonist.
T4102 Goserelin acetate Goserelin acetate is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
T5018 Leuprorelin Leuprolide is an agonist at pituitary GnRH receptors.GnRH receptor Leuprorelin is a gonadotrophin-releasing hormone (GnRH) analogue used to treat a wide range of...
T5021 Leuprolide Acetate (53714-56-0 free base) Leuprolide is an agonist at pituitary GnRH receptors. Leuprorelin is a gonadotropin-releasing hormone (GnRH) analog used to treat a wide range of sex hormone-rel...
T5520 Cetrorelix( x acetate) Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
T5031 Elagolix sodium Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
T10988 Degarelix Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
TP2337 Ganirelix Acetate Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
T10217L Abarelix Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
T11174 (R)-Elagolix (R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable de...
T21309 Nafarelin acetate(76932-56-4 free base) Nafarelin acetate is a GnRH agonist that acts as an analog of GnRH. Nafarelin causes a decrease in the pituitary secretion of gonadotropins luteinizing hormone (...
T21410 Triptorelin acetate(57773-63-4 free base) Triptorelin Acetate is used as a GnRH agonist. It decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH) ...
T5520L Cetrorelix diacetate Cetrorelix diacetate is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the ...
TP1700L LGnRH-III, lamprey acetate(147859-97-0 free base) LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion of...
TP1434L Lecirelin acetate(61012-19-9 free base) Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts....
TP2323L Deslorelin acetate(57773-65-6 free base) Deslorelin acetate is a gonadotropin releasing hormone super-agonist (GnRH agonist)
T1480 Danazol Danazol is a synthetic steroid with antigonadotropic and anti-estrogenic activities that acts as an anterior pituitary suppressant by inhibiting the pituitary ou...
Degarelix acetate(214766-78-6 free base)
T10988LCAS T10988L
Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
Buserelin Acetate (57982-77-1 free base)
TP1307CAS 68630-75-1
Buserelin Acetate is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
Relugolix
T3630CAS 737789-87-6
Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential an...
Alarelin
T1494CAS 79561-22-1
Alarelin acetate is a synthetic GnRH agonist.
Goserelin acetate
T4102CAS 145781-92-6
Goserelin acetate is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
Leuprorelin
T5018CAS 53714-56-0
Leuprolide is an agonist at pituitary GnRH receptors.GnRH receptor Leuprorelin is a gonadotrophin-releasing hormone (GnRH) analogue used to treat a wide range of...
Leuprolide Acetate (53714-56-0 free base)
T5021CAS 74381-53-6
Leuprolide is an agonist at pituitary GnRH receptors. Leuprorelin is a gonadotropin-releasing hormone (GnRH) analog used to treat a wide range of sex hormone-rel...
Cetrorelix( x acetate)
T5520CAS 145672-81-7
Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
Elagolix sodium
T5031CAS 832720-36-2
Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
Degarelix
T10988CAS 214766-78-6
Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
Ganirelix Acetate
TP2337CAS 123246-29-7
Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
Abarelix
T10217LCAS 183552-38-7
Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
(R)-Elagolix
T11174CAS 834153-87-6
(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable de...
Nafarelin acetate(76932-56-4 free base)
T21309CAS 76932-60-0
Nafarelin acetate is a GnRH agonist that acts as an analog of GnRH. Nafarelin causes a decrease in the pituitary secretion of gonadotropins luteinizing hormone (...
Triptorelin acetate(57773-63-4 free base)
T21410CAS 140194-24-7
Triptorelin Acetate is used as a GnRH agonist. It decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH) ...
Cetrorelix diacetate
T5520LCAS 130143-01-0
Cetrorelix diacetate is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the ...
LGnRH-III, lamprey acetate(147859-97-0 free base)
TP1700LCAS TP1700L
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion of...
Lecirelin acetate(61012-19-9 free base)
TP1434LCAS TP1434L
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts....
Deslorelin acetate(57773-65-6 free base)
TP2323LCAS TP2323L
Deslorelin acetate is a gonadotropin releasing hormone super-agonist (GnRH agonist)
Danazol
T1480CAS 17230-88-5
Danazol is a synthetic steroid with antigonadotropic and anti-estrogenic activities that acts as an anterior pituitary suppressant by inhibiting the pituitary ou...