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Search Result

Search Results for " cannabinoid cb2 receptor "

Targets

Cannabinoid Receptor

43

Compounds

1

Natural Products

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T10696 CB2 modulator 1 Cannabinoid Receptor
CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.
T12306 OMDM-5 Cannabinoid Receptor , Endogenous Metabolite , TRP/TRPV Channel
OMDM-5 is a selective anandamide cellular uptake (ACU)inhibitor(Ki of 4.8 μM).
T12302 OMDM-1 (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide Endogenous Metabolite
OMDM-1 ((Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide) is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor with a Ki of 2.4 μM.
T22009 CB2 receptor agonist 2 ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist Cannabinoid Receptor
CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.
T6527 GW842166X Cannabinoid Receptor
GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor. Phase 2.
T6755 AM1241 Cannabinoid Receptor
AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.
T14302 Olorinab APD 371 Cannabinoid Receptor
Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.
T7375 A-836339 Cannabinoid Receptor
A-836339 acts as a potent cannabinoid receptor full agonist which has a higher affinity for the peripheral CB2 receptor (Ki = 0.64 nM) over the central CB1 receptor (Ki = 270 nM). It displays analgesic, anti-inflammatory...
T7316 LY2828360 Cannabinoid Receptor
LY2828360 is a cannabinoid (CB) receptor 2 agonist (Ki = 40.3 nM). It selectively activates CB2 over CB1 in a GTPγS binding assay (EC50s = 20.1 and >100,000 nM, respectively).
T41231 GP 1a Cannabinoid Receptor , PERK , Arrestin
GP 1a is a potent agonist of cannabinoid receptor 2 (CB2) (EC50=7.1), as shown in cAMP, GTPγS and β-arrestin recruitment assays. GP 1a is approximately 30-fold more selective for CB2 receptors than CB1 receptors and incr...
T37075 CB2R PAM Ec2la Cannabinoid Receptor
CB2R PAM is an orally active cannabinoid type 2 receptor (CB2Rs) positive mutational modulator that enhances CP 55940 and 2-Arachidonylglycerol-stimulated [35S]GTPγS binding to CB2 receptors, but has no effect in the abs...
T3530 Otenabant CP-945598 Cannabinoid Receptor
Otenabant (CP-945598) has been investigated for the treatment of Obesity.
T10697 CB2R-IN-1 Others
CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).
T32336 JWH-149
JWH 149, a synthetic cannabinoid (CB), can potently bind both the central CB1 receptor (Ki = 5.0 nM) and the peripheral CB2 receptor (Ki = 0.73 nM).
T25874 NMP-7 NMP7,NMP 7
NMP-7 is a non-selective CB1 and CB2 cannabinoid receptor agonist that works by blocking T-type calcium channels.
T24218 JTE 7-31
JTE 7-31 is a selective agonist of the cannabinoid receptor. It is a reasonably highly selective CB2 agonist (Ki: 0.088 nM at CB2 vs 11 nM at CB1).
T32341 JWH-251
JWH 251, a cannabimimetic indole, has a high affinity tothe central cannabinoid (CB1) receptor (Ki = 29 nM) and a comparatively modest affinity for the peripheral cannabinoid (CB2) receptor (Ki = 146 nM). JWH 251 can st...
T17027 Tedalinab GRC-10693 Cannabinoid Receptor
Tedalinab is an effective and selective cannabinoid receptor 2 agonist. Tedalinab has the potential for neuropathic pain and osteoarthritis treatment. Tedalinab has >4700-fold functional selectivity for CB2 over CB1.
T24939 Virodhamine trifluoroacetate Virodhamine-trifluoroacetate,Virodhamine trifluoroacetate salt
Virodhamine trifluoroacetate is an antagonist of endogenous cannabinoid receptor mixed that acts by being a full agonist at GPR55 and CB2 and partial antagonist at CB1.
T14504 BAY 38-7271 Cannabinoid Receptor
BAY 38-7271 has strong neuroprotective properties.[1] BAY 38-7271 is selective and highly potent and cannabinoid CB1/CB2 receptor agonist. With Kis of 1.85 nM and 5.96 nM for recombinant human CB1 receptor and CB2 recept...
T29933 AM-1714 UNII-E3OY6PCU04,AM1714
AM-1714 is a reasonable selective agonist for the peripheral cannabinoid receptor CB2. In animal studies, it has been shown to have analgesic and anti-abnormal pain effects.
T32582 LASSBio-881 LASSBio881,LASSBio 881
LASSBio-881 is a non-selective partial agonist of the CB1 and CB2 cannabinoid receptors, as well as an antagonist of the TRPV1 receptor.
T32334 JWH-098
JWH 098, a potent synthetic cannabinoid (CB), can activate the CB1 receptor with a Ki value of 4.5 nM and the CB2 receptor with a Ki value of 1.88 nM. Its effects in cells and animals are still on study.
T32331 JWH 072 JWH072,JWH-072
JWH 072 , known as synthetic cannabinoid (CB), displays a higher affinity to the peripheral CB2 receptor (Ki = 170 nM) than the central CB1 receptor (Ki = 1,050 nM). Its physiological and toxicological properties are sti...
T38912 Vicasinabin
Vicasinabin, a potent agonist of cannabinoid receptor 2 (CB2), exhibits promising potential for researching chronic pain, atherosclerosis, regulation of bone mass, neuroinflammation, and related human diseases.
T30903 CHM-081 CHM 081
JWH 081, a cannabimimetic aminoalkylindole, has a high-affinity to the central cannabinoid (CB1) receptor (Ki =1.2 nM) and ten-fold reduced affinity to the peripheral cannabinoid (CB2) receptor (Ki = 12.4 nM). JWH 081-N-...
T32338 JWH-182 JWH182
JWH 182, a potent synthetic cannabinoid (CB) can activate the central CB1 receptor and the peripheral CB2 receptor with a Ki value of 0.65 nM and 1.1 nM, respectively. Its effects in cells and animals have not evaluated.
T36566 Amauromine
Amauromine is a neutral antagonist of the cannabinoid (CB) receptor CB1 that is selective for CB1 (Ki = 178 nM; Kb = 66.6 nM) over CB2, with no activity at CB2 receptors at concentrations up to 10 μM. It is also an antag...
T38049 Glycerophospho-N-Palmitoyl Ethanolamine
N-Acylated ethanolamines (NAE) are naturally-occurring lipids that have diverse bioactivities. For example, arachidonoyl ethanolamide (AEA) is an endogenous neurotransmitter that evokes cellular responses by activating t...
T38199 (±)-WIN 55,212 (mesylate)
(±)-WIN 55,212-2 is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki value of 62.3 and 3.3 nM for human recombinant central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, respectively....
T68247 PSB-KD107
PSB-KD107 is an agonist of the Cannabinoid-Activated Orphan G‑Protein-Coupled Receptor GPR18. PSB-KD107 displayed significantly higher potency and efficacy than THC, determined in a GPR18-dependent β-arrestin recruitment...
T38147 (S)-AM1241 (S)-AM1241
(S)-AM1241 binds to cannabinoid (CB) receptors and is selective for the CB2 over the CB1 receptor (Kis = 658 and >10,000 nM, respectively, in a membrane assay using human receptors). (S)-1241 acts as an agonist at human,...
T38030 (R)-AM1241 (R)-AM1241
(R)-AM1241 binds to cannabinoid (CB) receptors and has greater than 100-fold selectivity for the CB2 over the CB1 receptor (Kis = 15 and 5,000 nM, respectively, in a membrane assay using human receptors). (R)-AM1241 acts...
T21914 (S)-SLV 319
Ibipinabant (SLV319) is a potent, selective, and orally active antagonist of the cannabinoid CB1 receptor, demonstrating a K i of 7.8 nM and exhibiting over 1000-fold selectivity for CB1 compared to CB2 (K i =7943 nM). I...
T62132 S-777469
S-777469 is a selective, orally active agonist of the cannabinoid type 2 receptor (CB2) (Ki: 36 nM). s-777469 significantly inhibited compound 48/80-induced scratching behaviour in mice in a dose-dependent manner. s-7774...
T27809 LEI-101
LEI-101 is a potent, selective, and orally bioavailable cannabinoid CB2 receptor agonist, with a pEC 50 of 8 for hCB2, and a pK i of less than 4 for hERG. LEI-101 is ~100-fold more potent in binding to CB2 receptors than...
T38138 ACEA 2'-chloro-AEA,Arachidonoyl 2'-Chloroethylamide
Arachidonoyl 2-chloroethylamide (ACEA) is a potent and selective cannabinoid (CB) receptor 1 agonist with Ki values of 1.4 and >2,000 nM for CB1 and CB2 receptors, respectively. In whole animal experiments, ACEA induces ...
T71963 (−)-WIN 55,212-3 mesylate
(−)-WIN 55,212-3 mesylate is an aminoalkylindole derivative which acts as a competitive neutral antagonist of the human cannabinoid CB2 receptor, blocking both the stimulating action of CP 55,940 and the inverse agonism ...
T79577 CB2 PET Radioligand 1 Cannabinoid Receptor
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.7 nM). It is synthesized via Cu-mediated 18F-fluorination an...
T23099 O-2050 Others
O-2050 is a high affinity cannabinoid CB 1 receptor antagonist with a K i of 2.5 nM. O-2050 inhibits cannabinoid CB 2 receptor with Ki of 0.2 nM. O-2050 decreased food intake in mice and caused locomotor stimulation in m...
T69612 PSB-KD477
PSB-KD477 is an Agonist of the Cannabinoid-Activated Orphan G-Protein-Coupled Receptor GPR18. PSB-KD477 displayed significantly higher potency and efficacy than THC, determined in a GPR18-dependent β-arrestin recruitment...
T35408 (±)10(11)-EDP Ethanolamide
(±)10(11)-EDP ethanolamide is an ω-3 endocannabinoid epoxide and cannabinoid (CB) receptor agonist (EC50s = 0.43 and 22.5 nM for CB1 and CB2 receptors, respectively). It is produced though direct epoxygenation of docosah...
T35468 (±)19(20)-EDP Ethanolamide
(±)19(20)-EDP ethanolamide is an ω-3 endocannabinoid epoxide and cannabinoid (CB) receptor agonist (EC50s = 108 and 280 nM for CB1 and CB2, respectively). It is produced through direct epoxygenation of docosahexaenoyl et...

Compounds

CB2 modulator 1
T10696
Synonym:
Target: Cannabinoid Receptor
OMDM-5
T12306
Synonym:
Target: Cannabinoid Receptor, Endogenous Metabolite, TRP/TRPV Channel
OMDM-1
T12302
Synonym: (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide
Target: Endogenous Metabolite
CB2 receptor agonist 2
T22009
Synonym: ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist
Target: Cannabinoid Receptor
GW842166X
T6527
Synonym:
Target: Cannabinoid Receptor
AM1241
T6755
Synonym:
Target: Cannabinoid Receptor
Olorinab
T14302
Synonym: APD 371
Target: Cannabinoid Receptor
A-836339
T7375
Synonym:
Target: Cannabinoid Receptor
LY2828360
T7316
Synonym:
Target: Cannabinoid Receptor
GP 1a
T41231
Synonym:
Target: Cannabinoid Receptor, PERK, Arrestin
CB2R PAM
T37075
Synonym: Ec2la
Target: Cannabinoid Receptor
Otenabant
T3530
Synonym: CP-945598
Target: Cannabinoid Receptor
CB2R-IN-1
T10697
Synonym:
Target: Others
JWH-149
T32336
Synonym:
Target:
NMP-7
T25874
Synonym: NMP7,NMP 7
Target:
JTE 7-31
T24218
Synonym:
Target:
JWH-251
T32341
Synonym:
Target:
Tedalinab
T17027
Synonym: GRC-10693
Target: Cannabinoid Receptor
Virodhamine trifluoroacetate
T24939
Synonym: Virodhamine-trifluoroacetate,Virodhamine trifluoroacetate salt
Target:
BAY 38-7271
T14504
Synonym:
Target: Cannabinoid Receptor
AM-1714
T29933
Synonym: UNII-E3OY6PCU04,AM1714
Target:
LASSBio-881
T32582
Synonym: LASSBio881,LASSBio 881
Target:
JWH-098
T32334
Synonym:
Target:
JWH 072
T32331
Synonym: JWH072,JWH-072
Target:
Vicasinabin
T38912
Synonym:
Target:
CHM-081
T30903
Synonym: CHM 081
Target:
JWH-182
T32338
Synonym: JWH182
Target:
Amauromine
T36566
Synonym:
Target:
Glycerophospho-N-Palmitoyl Ethanolamine
T38049
Synonym:
Target:
(±)-WIN 55,212 (mesylate)
T38199
Synonym:
Target:
PSB-KD107
T68247
Synonym:
Target:
(S)-AM1241
T38147
Synonym: (S)-AM1241
Target:
(R)-AM1241
T38030
Synonym: (R)-AM1241
Target:
(S)-SLV 319
T21914
Synonym:
Target:
S-777469
T62132
Synonym:
Target:
LEI-101
T27809
Synonym:
Target:
ACEA
T38138
Synonym: 2'-chloro-AEA,Arachidonoyl 2'-Chloroethylamide
Target:
(−)-WIN 55,212-3 mesylate
T71963
Synonym:
Target:
CB2 PET Radioligand 1
T79577
Synonym:
Target: Cannabinoid Receptor
O-2050
T23099
Synonym:
Target: Others
PSB-KD477
T69612
Synonym:
Target:
(±)10(11)-EDP Ethanolamide
T35408
Synonym:
Target:
(±)19(20)-EDP Ethanolamide
T35468
Synonym:
Target:
Cat No. Product Name Synonyms Targets
TN2268 Tetrahydromagnolol Cannabinoid Receptor , GPR , GABA Receptor
Tetrahydromagnolol can activate cannabinoid (CB) receptors.

Natural Products

Tetrahydromagnolol
TN2268
Synonym:
Target: Cannabinoid Receptor, GPR, GABA Receptor

Recombinant Proteins

Species：
Human (1)
Expression System：
HEK293 (1)
Tag：
Tag Free (1)
Cat No. Product Name Species Expression System
TMPY-06623 CB2/CNR2 Protein, Human, Recombinant Human HEK293
Genetic variants within the CNR2 gene encoding the cannabinoid receptor CB2 are associated with osteoporosis and low bone mineral density (BMD) in case-control studies. There is a possibility that genetic variants of the...
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