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Search Result

Search Results for " bradykinin-receptor "

Targets

Bradykinin Receptor

51

Compounds

2

Recombinant Proteins

1

Libraries

Cat No. Product Name Synonyms Targets
TP1181 Bradykinin (2-9) Des-Arg1-bradykinin Bradykinin Receptor
Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin. It is formed by the cleavage action of Aminopeptidase P.
TP1445 [Des-Arg9]-Bradykinin acetate Bradykinin Receptor
[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.
TP1277 Bradykinin Endogenous Metabolite , Bradykinin Receptor
Bradykinin is an inflammatory mediator. It is a peptide that causes blood vessels to dilate (enlarge) via the release of prostacyclin, nitric oxide, and Endothelium-Derived Hyperpolarizing Factor. Bradykinin is a physiol...
T5048 SSR240612 Bradykinin Receptor
SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively).
T22344 Icatibant Acetate Bradykinin Receptor
Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.
T2086 ELN-441958 ELN 441958 Bradykinin Receptor
ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. ELN-441958(ELN 441958) is highly selective for B1 over B2 receptors.
T7645 [Des-Arg9]-Bradykinin [Des-Arg9]-Bradykinin(2TFA) Bradykinin Receptor
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
TP2268L Lys-Bradykinin acetate(342-10-9 free base) Bradykinin Receptor
Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.
T8809 [Des-Arg9]-Bradykinin TFA Bradykinin Receptor
[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.
T33421 MK-0686 MK0686 Bradykinin Receptor
MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.
T36442L (Hyp³)-Bradykinin acetate (Hyp³)-Bradykinin acetate (37642-65-2 Free base) Bradykinin Receptor
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.
TP2075L Bombinakinin M acetate Bombinakinin M acetate(509151-65-9 free base) Bradykinin Receptor
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is approximately 50 times more potent than bradykinin.
TP1918L1 Lys-[Des-Arg9]Bradykinin acetate Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base) Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces p...
TP1918L Lys-[Des-Arg9]Bradykinin,TFA Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa) Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripher...
T34485 Safotibant LF220542,LF 220542,LF 22-0542,LF-220542,LF-22-0542,LF22-0542 Bradykinin Receptor
Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edema.
TP1917L1 Sar-[D-Phe8]-des-Arg9-Bradykinin acetate Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) Bradykinin Receptor
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cl...
T26627L Anatibant 2HCl Anatibant 2HCl(209733-45-9 Free base) Bradykinin Receptor
Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.
TP1933 R715 TFA(185052-09-9 free base) R 715 Bradykinin Receptor
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49). Displays no activity at B2 receptors. Reduces mechanical hypernociception in a mouse model of neuropathic pain. Me...
TP1931L1 [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base) cholecystokinin
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist ...
T4200 Sacubitril hemicalcium salt AHU-377 (hemicalcium salt),AHU377 calcium salt Neprilysin
Sacubitril hemicalcium salt (AHU377 calcium salt) is a potent NEP inhibitor with an IC50 of 5 nM. Sacubitril hemicalcium salt is a component of the heart failure medicine LCZ696. Sacubitril hemicalcium salt is a prodrug ...
T15347 FR167344 free base Others
FR167344 free base is an orally active and nonpeptide antagonist of bradykinin receptor B2. FR167344 free base displays a high-affinity binding to the B2 receptor (IC50: 65 nM). It has no binding affinity for the B1 rece...
T27377 FR190997 FR-190997,FR 190997
FR190997 is an agonist of bradykinin B2 receptor.
T70750 Deltibant
Deltibantis a bradykinin receptor antagonist.
T21060 NPC 567
NPC 567 is an antagonist of the bradykinin receptor.
T69673 Deucrictibant
Deucrictibant is a bradykinin receptor antagonist.
T70576 NPC 17731
NPC 17731 is a bradykinin receptor antagonist.
T70574 NPC 17761
NPC 17761 is a bradykinin receptor antagonist.
T63241 Fulimetibant
Fulimetibant is a bradykinin receptor antagonist.
T80117 Lys-(Des-Arg9,Leu8)-Bradykinin Bradykinin Receptor
Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].
T25895 NVP-SAA164 SAA 164,SAA164,SAA-164,NVP SAA164
NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.
T25555 JMV-1645 JMV1645,JMV 1645
JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.
T24065 FK-3657 FK 3657,FK3657,FR-173657,FR 173657,FR173657
FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.
T15547 Icatibant HOE 140 Others
Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).
TP2076 [Phe8Ψ(CH-NH)-Arg9]-Bradykinin
Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage. 5-fold more potent and exhibits a more prolonged duration of action than bradykinin in vivo.
TP2075 Bombinakinin M
Potent bradykinin receptor agonist. Highly selective for mammalian arterial smooth muscle bradykinin receptors, displaying ~ 50-fold greater potency than bradykinin. Elicits dose-dependent contractile effects in smooth m...
TP2268 Lys-Bradykinin Others
Endogenous bradykinin receptor agonist
T80072 Des-Arg9-[Leu8]-Bradykinin acetate Bradykinin Receptor
Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].
T76385 [Tyr8] Bradykinin
[Tyr8] Bradykinin, a B2 kinin receptor agonist, not only stimulates ERK1/2 phosphorylation but also serves as an internal standard [1].
TP1918 Lys-[Des-Arg9]Bradykinin
Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. ...
T76212 B 9430
B 9430 is a potent bradykinin B1/B2 receptor antagonist [1] .
T27790 Labradimil RMP-7,ALK-01-040,Receptor-mediated permeabiliser-7,DRG0182,DRG 0182,DRG-0182
Labradimil is a bradykinin B2 receptor agonist. Labradimil increases the permeability of human brain microvascular endothelial cell monolayers. Labradimil enhances delivery of hydrophilic chemotherapeutics and increases ...
T83500 [Des-Arg10]-HOE I40
[Des-Arg10]-HOE 140 is a bioactive peptide that functions as a potent B1 bradykinin receptor antagonist.
T38544 Fasitibant chloride MEN16132 free base,Fasitibant chloride
Fasitibant chloride (MEN16132 free base) is a powerful and specific nonpeptide antagonist of the bradykinin B2 receptor (B2R). This compound effectively reduces joint pain and mitigates joint edema in a rat model of Carr...
T73646 Lys-[Des-Arg9]Bradykinin TFA
Lys-[Des-Arg9]Bradykinin TFA is a naturally occurring kinin that serves as a potent and highly selective agonist for the bradykinin B1 receptor, demonstrating binding affinities (K i values) of 0.12 nM, 1.7 nM, and 0.23 ...
TP1931 [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
Broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradyki...
TP1917 Sar-[D-Phe8]-des-Arg9-Bradykinin
Potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cleavage. Exhibits hypotensive and angiogenic ac...
TP1999 MEN 11270
Peptide antagonist of the B2 bradykinin receptor (pKi = 10.3); conformationally constrained cyclized analog of HOE 140. Blocks hypotension and bronchoconstriction in vivo. Displays selectivity for B2 over 29 other recept...
T26627 Anatibant LF16-0687,LF-16-0687,LF 160687,LF 16-0687,LF-160687
Anatibant is a potent non-peptide bradykinin B2 receptor antagonist. Anatibant reduces intracranial hypertension and histopathological damage after experimental traumatic brain injury.
TP2126 R 892
Potent and selective bradykinin B1 receptor antagonist (ID50 values are 2.8 and > 600 nM at B1 and B2 receptors respectively). Exhibits no intrinsic agonist activity and is resistant to aminopeptidase and kininase II (AC...
TP1662 Galanin Receptor Ligand M35
The chimeric peptide M35 [galanin (1-13)-bradykinin(2-9) amide] is a high-affinity galanin receptor ligand acting as a galanin receptor antagonist in the rat spinal cord, rat hippocampus and isolated mouse pancreatic isl...

Compounds

Bradykinin (2-9)
TP1181
Synonym: Des-Arg1-bradykinin
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin acetate
TP1445
Synonym:
Target: Bradykinin Receptor
Bradykinin
TP1277
Synonym:
Target: Endogenous Metabolite, Bradykinin Receptor
SSR240612
T5048
Synonym:
Target: Bradykinin Receptor
Icatibant Acetate
T22344
Synonym:
Target: Bradykinin Receptor
ELN-441958
T2086
Synonym: ELN 441958
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin
T7645
Synonym: [Des-Arg9]-Bradykinin(2TFA)
Target: Bradykinin Receptor
Lys-Bradykinin acetate(342-10-9 free base)
TP2268L
Synonym:
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin TFA
T8809
Synonym:
Target: Bradykinin Receptor
MK-0686
T33421
Synonym: MK0686
Target: Bradykinin Receptor
(Hyp³)-Bradykinin acetate
T36442L
Synonym: (Hyp³)-Bradykinin acetate (37642-65-2 Free base)
Target: Bradykinin Receptor
Bombinakinin M acetate
TP2075L
Synonym: Bombinakinin M acetate(509151-65-9 free base)
Target: Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin acetate
TP1918L1
Synonym: Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base)
Target: Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin,TFA
TP1918L
Synonym: Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa)
Target: Bradykinin Receptor
Safotibant
T34485
Synonym: LF220542,LF 220542,LF 22-0542,LF-220542,LF-22-0542,LF22-0542
Target: Bradykinin Receptor
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
TP1917L1
Synonym: Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base)
Target: Bradykinin Receptor
Anatibant 2HCl
T26627L
Synonym: Anatibant 2HCl(209733-45-9 Free base)
Target: Bradykinin Receptor
R715 TFA(185052-09-9 free base)
TP1933
Synonym: R 715
Target: Bradykinin Receptor
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
TP1931L1
Synonym: [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base)
Target: cholecystokinin
Sacubitril hemicalcium salt
T4200
Synonym: AHU-377 (hemicalcium salt),AHU377 calcium salt
Target: Neprilysin
FR167344 free base
T15347
Synonym:
Target: Others
FR190997
T27377
Synonym: FR-190997,FR 190997
Target:
Deltibant
T70750
Synonym:
Target:
NPC 567
T21060
Synonym:
Target:
Deucrictibant
T69673
Synonym:
Target:
NPC 17731
T70576
Synonym:
Target:
NPC 17761
T70574
Synonym:
Target:
Fulimetibant
T63241
Synonym:
Target:
Lys-(Des-Arg9,Leu8)-Bradykinin
T80117
Synonym:
Target: Bradykinin Receptor
NVP-SAA164
T25895
Synonym: SAA 164,SAA164,SAA-164,NVP SAA164
Target:
JMV-1645
T25555
Synonym: JMV1645,JMV 1645
Target:
FK-3657
T24065
Synonym: FK 3657,FK3657,FR-173657,FR 173657,FR173657
Target:
Icatibant
T15547
Synonym: HOE 140
Target: Others
[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
TP2076
Synonym:
Target:
Bombinakinin M
TP2075
Synonym:
Target:
Lys-Bradykinin
TP2268
Synonym:
Target: Others
Des-Arg9-[Leu8]-Bradykinin acetate
T80072
Synonym:
Target: Bradykinin Receptor
[Tyr8] Bradykinin
T76385
Synonym:
Target:
Lys-[Des-Arg9]Bradykinin
TP1918
Synonym:
Target:
B 9430
T76212
Synonym:
Target:
Labradimil
T27790
Synonym: RMP-7,ALK-01-040,Receptor-mediated permeabiliser-7,DRG0182,DRG 0182,DRG-0182
Target:
[Des-Arg10]-HOE I40
T83500
Synonym:
Target:
Fasitibant chloride
T38544
Synonym: MEN16132 free base,Fasitibant chloride
Target:
Lys-[Des-Arg9]Bradykinin TFA
T73646
Synonym:
Target:
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
TP1931
Synonym:
Target:
Sar-[D-Phe8]-des-Arg9-Bradykinin
TP1917
Synonym:
Target:
MEN 11270
TP1999
Synonym:
Target:
Anatibant
T26627
Synonym: LF16-0687,LF-16-0687,LF 160687,LF 16-0687,LF-160687
Target:
R 892
TP2126
Synonym:
Target:
Galanin Receptor Ligand M35
TP1662
Synonym:
Target:
1 2

Recombinant Proteins

Species：
Human (1)
Paguma larvata (1)
Expression System：
Baculovirus-Insect Cells (1)
HEK293 (1)
Tag：
C-terminal hFc-tagged (1)
His (1)
Cat No. Product Name Species Expression System
TMPH-03081 ACE2 Protein, Paguma larvata, Recombinant (hFc) Paguma larvata HEK293
Essential counter-regulatory carboxypeptidase of the renin-angiotensin hormone system that is a critical regulator of blood volume, systemic vascular resistance, and thus cardiovascular homeostasis. Converts angiotensin ...
TMPY-00410 EPHX2 Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
Genetic variation in EPHX2 was significantly associated with risk of incident CHD in Caucasians, implicating EPHX2 as a potential cardiovascular disease-susceptibility gene. Single nucleotide polymorphisms (SNPs) in the ...
Cat No. Product Name
L7110 Anti-Hypertension Compound Library

719 compounds
719 hypertension-related small molecules for high-throughput and high-content screening.

Libraries

Anti-Hypertension Compound Library
L7110
Compounds: 719
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