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GPCR/G Protein Adrenergic Receptor

Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma.
Cat No. product name
T1056 Isoprenaline hydrochlorideHOT Isoproterenol is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
T9220 Naftopidil hydrochloride Naftopidil hydrochloride is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenocep...
T3033 Deoxycorticosterone acetate Desoxycorticosterone acetate is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of the adrenocortical...
T0487 Metoprolol tartrate Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.
T0446 Naphazoline hydrochloride Naphazoline hydrochloride is an adrenergic vasoconstrictor agent used as a decongestant.
T1215 Nicardipine hydrochloride Nicardipine Hydrochloride is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nicar...
T2889 Isoferulic acid 3-Hydroxy-4-methoxycinnamic Acid exhibits hypoglycemic properties.
T0766 Promazine hydrochloride Promazine hydrochloride is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. It is primarily used in short-term treatm...
T6703 Tetrahydrozoline HCl Tetrahydrozoline HCl is an imidazoline derivative with alpha receptor agonist activity.
T1045 Trimipramine maleate Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin an...
T1282 Carteolol hydrochloride Carteolol Hydrochloride is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocking agent for be...
T0852 Carbazochrome sodium sulfonate Carbazochrome sodium sulfonate (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.
T1047 Epinephrine bitartrate L-Epinephrine Bitartrate is alpha- and beta-adrenergic receptor stimulator.
T6652 Salbutamol Sulfate Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
T3277 Tulobuterol hydrochloride Tulobuterol hydrochloride is a long-acting beta2-adrenergic receptor agonist.
T2645 Vilanterol Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.
T6662 Scopine Scopine, the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
T1738 Taxifolin Taxifolin is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.
T6505 Formoterol Hemifumarate Formoterol Hemifumarate, an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of chronic obstructive pulmonary disease(C...
T1203 Nadolol Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities. Nadolol competitively blocks beta-1 adrenergic recepto...
T1247 Clonidine hydrochloride Clonidine is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide ...
T3278 Piribedil Piribedil is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
T0317 Buflomedil hydrochloride Buflomedil hydrochloride, a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.
T0165 Urapidil Urapidil, a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
T1012 Acebutolol hydrochloride Acebutolol acts as a cardioselective beta-adrenergic antagonist with little effect on bronchial receptors and has intrinsic sympathomimetic properties. Acebutolo...
T0279 Metaraminol bitartrate Metaraminol bitartrate is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in the...
T0007L (R)-(+)-Atenolol (R)-(+)-Atenolol is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.
T0696 Naftopidil Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
T1071L2 DL-Adrenalin DL-Epinephrine(DL-Adrenaline) is a hormone and a neurotransmitter.
T0993 Methoxamine hydrochloride An alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
T1275 Phentolamine mesilate Phentolamine mesylate is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, ...
T2142 Yohimbine hydrochloride Yohimbine hydrochloride is a plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of ERECTILE DY...
T0088 Urapidil hydrochloride Urapidil hydrochloride is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
T0290 Tizanidine hydrochloride Tizanidine hydrochloride, an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
T0103 Dipivefrin hydrochloride Dipivefrin that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
T1158 Phenoxybenzamine hydrochloride Phenoxybenzamine Hydrochloride is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive and...
T0226 Betaxolol hydrochloride Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induced...
T6408 Betaxolol Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T0197 Terazosin hydrochloride Terazosin, a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a drug of choice for patie...
T0948 Adrenalone hydrochloride Adrenalone hydrochloride, a selective α1-adrenoceptor agonist, is used as a topical hemostatic and vasoconstrictor and used to extend the effect of local anesth...
T0453 Phenylephrine hydrochloride Phenylephrine hydrochloride is a selective agonist of the α1-adrenergic receptor.
T0342 Carvedilol phosphate Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intri...
T6600 Naftopidil DiHCl Naftopidil DiHCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
T0445 Promethazine Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
T1680 Tolazoline hydrochloride Tolazoline is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.
T6688 Synephrine HCl SynephrineHCl (Oxedrine, p-Synephrine) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
T0277 Orciprenaline sulfate Orciprenaline sulfate is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
T1090 Perphenazine Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
T0445L Promethazine hydrochloride Promethazine HCl(NSC-231688), the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mACh receptor, moder...
T0991 Desipramine hydrochloride Desipramine Hydrochloride a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervous system (CNS), d...
T0324 Isoxsuprine hydrochloride Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
T0455 Clozapine Clozapine is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays...
T3284 Carazolol Carazolol is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
T1244 Celiprolol hydrochloride Celiprolol hydrochloride is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity. It is used in the management of ANGINA PE...
T1632 Amitraz AMITRAZ is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic ma...
T0348 Labetalol hydrochloride Labetalol hydrochloride, a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
T0871 Noradrenaline bitartrate Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors. Norepinephrine Bitartrate is a bitartrate salt of norepinephrine, a synthetic phe...
T6860 ICI-118551 Hydrochloride ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
T0076 Paliperidone Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the pr...
T1073 Dronedarone hydrochloride Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
T0031 Ziprasidone hydrochloride monohydrate Ziprasidone(CP88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic activity.
T0735 Pindolol Pindolol is a moderately lipophilic beta blocker (ADRENERGIC BETA-ANTAGONISTS). It is non-cardioselective and has intrinsic sympathomimetic actions, but little m...
T1539 Iloperidone Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
T1567 Olanzapine Olanzapine is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
T0365 Thioridazine hydrochloride Thioridazine, an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selectivity.
T0185 Escitalopram Escitalopram is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol upta...
T1540 Doxepin hydrochloride Doxepin Hydrochloride is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mech...
T0031L Ziprasidone hydrochloride Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T0042 Xylometazoline hydrochloride Xylometazoline Hydrochloride is an α-adrenoceptor agonist usually used as nasal decongestant.
T0151 Efloxate Efloxate, a vasodilator, is utilized in the treatment of chronic coronary insufficiency.
T0031L2 Ziprasidone Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T6565 Levobetaxolol HCl Levobetaxolol hydrochloride is a beta-adrenergic receptor inhibitor (beta blocker), used to lower the pressure in the eye in treating conditions such as glaucoma...
T2524 Dexmedetomidine Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect of...
T6241 Quetiapine Fumarate Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
T0162 Quetiapin Quetiapine is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism of quetiapin...
T3232 Higenamine Hydrochloride Higenamine(Hydrochloride) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein...
T1064 Noradrenaline bitartrate monohydrate Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator.
T0210 Tamsulosin hydrochloride Tamsulosin Hydrochloride is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.
T0351 Risperidal Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
T0143 (±)-Bisoprolol hemifumarate Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart, thereb...
T6765 Atipamezole hydrochloride Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochlo...
T6766 Atipamezole Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
T6466 Dexmedetomidine HCl Dexmedetomidine hydrochloride is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE, which is t...
T2535 Ivabradine hydrochloride Ivabradine hydrochloride is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, hy...
T0812 Propranolol hydrochloride Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGIN...
T1433 Ritodrine hydrochloride Ritodrine binds to and activates beta-2 adrenergic receptors of myometrial cells in the uterus, which decreases the intensity and frequency of uterine contractio...
T2320 Indacaterol Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.
T1577 Midodrine hydrochloride Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergic...
T0007 Atenolol Atenolol is a selective β1 receptor antagonist.
T2150 Guanfacine hydrochloride Guanfacine hydrochloride is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.
T1132 Nicergoline Nicergoline is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
T1769 Pardoprunox Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
T0475 Timolol Maleate Timolol is a nonselective beta-adrenergic receptor blocker that is widely used for the therapy of hypertension, angina pectoris and prevention of vascular headac...
T1415 Gemfibrozil Gemfibrozil interacts with peroxisome proliferator-activated receptors (PPARalpha) resulting in PPARalpha-mediated stimulation of fatty acid oxidation and an inc...
T1619 Trazodone hydrochloride Trazodone hydrochloride is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients with major depress...
T2547 Droxidopa Droxidopa is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes of auton...
T6522 Guanabenz Acetate Guanabenz Acetate is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is ...
T1500 Xylazine hydrochloride Xylazine hydrochloride is an adrenergic alpha-2 agonist used as a sedative, analgesic and centrally acting muscle relaxant in veterinary medicine
T0154 Nebivolol hydrochloride Nebivolol hydrochloride is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR through the endothelial L-argin...
T1584 Terbutaline Sulfate Terbutaline sulfate is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
T1671 Mirabegron Mirabegron is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
T0783 Mianserin hydrochloride Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin r...
T3046 BMY 7378 dihydrochloride BMY-7378, α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T1696 2-(1-Piperazinyl)pyrimidine 2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
T2546 Pimozide Pimozide is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic rec...
T1496 Amiodarone hydrochloride Amiodarone hydrochloride is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action by inhibiting POT...
T1050 Prazosin hydrochloride Prazosin Hydrochloride reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism not complete...
T1139 Salbutamol Albuterol stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3', ...
T0970 Anisodamine Anisodamine is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T1504 Silodosin Silodosin is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
T6872 L755507 L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).
T0248 Clorprenaline hydrochloride Clorprenaline Hydrochloride is a beta-2 adrenergic agonist with bronchodilator activity.
T6701 Terazosin hydrochloride dihydrate Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
T5511 L-765314 L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the r...
T14287 Ancarolol Ancarolol is a blocking agent of beta-adrenergic.
T13403 ZK-90055 hydrochloride ZK-90055 hydrochloride is an agonist of β2 adrenergic receptor.
T10778 CGP 20712 A CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
T13285 Vatinoxan hydrochloride Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
T11318 Dopexamine hydrochloride Dopexamine hydrochloride is a β2-adrenergic receptor agonist.
T11286 Fiduxosin Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
T12970 Solabegron Solabegron is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(EC50 : 22 ...
T12829 Salmeterol Salmeterol is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
T12815 (S)-Terazosin (S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor ...
T15042 D2343 D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
T10364 Arbutamine Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure....
T12643 (R)-Terazosin (R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values o...
T7065 Tizanidine Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
T15943 M443 M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
T5134 Vilanterol trifenatate Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7...
T13016 SR59230A SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T13655 DL-Norepinephrine hydrochloride DL-Norepinephrine hydrochloride is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 μM.
T11036 Diacetolol D7 Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
T11015 Midaglizole hydrochloride Midaglizole hydrochloride (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6....
T11010 Detomidine carboxylic acid Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also ...
T10952 Dabuzalgron Dabuzalgron is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicity caused by do...
T12444 Phentolamine Analogue 1 Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
T12402 Penbutolol sulfate Penbutolol sulfate is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.
T12343 Benzquinamide Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
T13804 OPC-28326 OPC-28326 is a selective peripheral vasodilator and an α2-adrenergic receptor angatonist(α2A-, α2B- and α2C-adrenoceptors with Ki of 2040, 285, and 55 nM, ...
T13470 (±)-Methotrimeprazine (D6) (±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
T11786 KUL 7211 racemate KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
TN2267 Tetrahydroalstonine Tetrahydroalstonine and Raubasine preferentially block the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogenou...
TN5061 Stephanine l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
TP1238L ACTH 1-14 acetate(25696-21-3 free base) ACTH (1-14) is a fragment of adrenocorticotrophin, which regulates cortisol and androgen production.Adrenocorticotropic hormone (ACTH), also known as corticotrop...
T8899 Metipranolol Metipranolol is a β-adrenergic receptor antagonist that is given orally for the treatment of hypertension and also applied topically to the cornea for treating ...
T8738 LUN42518 HCl 47142-51-8(free base) LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.
T8810 Terbutaline Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol
T20570 Labetalol Labetalol is a mixed alpha/beta-adrenergic antagonist.It is used to treat high blood pressure. It can be given by mouth for long term hypertension management or ...
T21446 Rotigotine Hydrochloride Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
T8696 Propranolol HCl Propranolol hydrochloride is a blocker of β1 and β2 adrenergic receptor
T21066 Norepinephrine bitartrate salt Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
T21147 Clenbuterol Clenbuterol is a substituted phenylaminoethanol that has β2 adrenomimetic properties at very low doses, and is used as a bronchodilator in asthma.
T8663 Nifenalol.HCl Nifenalol is a antagonist of β-adrenergic receptor.
T23283 RX 821002 hydrochloride α2-adrenoceptor antagonist
TN4882 Quinine HCl Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T16759 Ritanserin Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adren...
TN4323 Isorauhimbine 3-Epi-alpha-yohimbine(Isorauhimbine) has alpha adrenoceptor blocking activities,it also has cardiovascular effects.
TN3507 Beta-Yohimbine Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
TN3368 Akuammigine Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
TN3364 Agrimonolide Agrimonolide is a potential α1 adrenergic receptor antagonist, it exerts anti-inflammatory activity, at least in part, via suppressing LPS-induced activation of...
T8595 Practolol Practolol is a selective β-adrenoceptor blocker.
T8580 Bupranolol Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic...
T22406 Prazosin Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T22275 Bisoprolol Bisoprolol is a cardioselective β1-adrenergic blocker used for secondary prevention of heart failure, myocardial, angina pectorisinfarction (MI) and mild to mod...
T17310 Phenylephrine Phenylephrine is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
T11894 Lusaperidone Lusaperidone is an α2 adrenergic receptor antagonist, with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively.
T16769 Ro 363 RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
T8348 Phentolamine Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
TN1922 Meranzin hydrate Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-h...
T6422 Brimonidine Tartrate Brimonidine tartrate is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pressure associated with...
T6579 Medetomidine HCl Medetomidine is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
T3165 Metoprolol Succinate Metoprolol succinate is a selective adrenergic beta-1 blocking agent that is commonly used to treat ANGINA PECTORIS; HYPERTENSION; and CARDIAC ARRHYTHMIAS.
T1459 Cisatracurium besylate Cisatracurium Besylate is a nondepolarizing skeletal muscle relaxant for intravenous administration.
T0394 Moxisylyte hydrochloride Moxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
T0483 Sotalol hydrochloride Sotalol Hydrochloride is the hydrochloride salt form of sotalol, an ethanolamine derivative with Class III antiarrhythmic and antihypertensive properties.
T6653 Salmeterol Xinafoate Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstru...
T1287 Synephrine Synephrine is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
T2306 Brexpiprazole Brexpiprazole is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.
T6464 Detomidine HCl Detomidine HCl produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
T1327 Nortriptyline hydrochloride Nortriptyline hydrochloride is a metabolite of AMITRIPTYLINE that is also used as an antidepressive agent. Nortriptyline is used in major depression, dysthymia, ...
T6519 Gramine Gramine, a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for ...
T3457 Olodaterol Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors lo...
T6663 Scopine HCl Scopine HCl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
T4429 Rauwolscine hydrochloride Rauwolscine, a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potent...
T0137 Mirtazapine Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T0173 Nylidrin hydrochloride Nylidrin hydrochloride was an effective inhibitor of the IgG1-mediated release of histamine from passively sensitized guinea pig lung slices, and of the IgE-medi...
T0397 Tetryzoline Tetrahydrozoline, an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of the eye resulted...
T1446 Bambuterol hydrochloride Bambuterol, a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
T0091 Alfuzosin hydrochloride Alfuzosin hydrochloride is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).
T1503 Esmolol hydrochloride Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instan...
T0115 Idazoxan hydrochloride Idazoxan hydrochloride is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
T0101 Doxazosin mesylate Doxazosin mesylate(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
T1239 Indacaterol maleate Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
T2580 Formoterol Arformoterol is an adrenergic β-2 receptor agonist with a prolonged duration of action. It is used to manage asthma and in the treatment of chronic obstructive ...
T0447 Carvedilol Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intri...
T1071L DL-Adrenaline Hydrochloride DL-Adrenaline Hydrochloride is the hydrochloride salt of the naturally occurring sympathomimetic amine with vasoconstricting, intraocular pressure-reducing activ...
T2226 Pergolide mesylate salt PERGOLIDE MESYLATE is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due to...
TN1797 Isorhoifolin Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
T7045 Clonidine Clonidine is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide-...
T8358 Fenoterol Fenoterol is an  agonist of  β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.
T8143 Bevantolol hydrochloride Bevantolol hydrochloride is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.
T8149 Dobutamine (hydrochloride) Dobutamine (hydrochloride) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
T8304 Anisodamine Hydrobromide Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
TCS2185 Yohimbine Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T7164 Levalbuterol tartrate Levosalbutamol tartrate is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
T7160 Lofexidine Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
T5471 GUANABENZ GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
T5450 DL-071-IT DL 071-IT is a potent non-selective beta-adrenoceptor antagonist. DL 071 IT showed intrinsic sympathomimetic activity and weak membrane stabilizing activity.
T5327 Amezinium (methylsulfate) Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition of noradrenaline and tyramine uptake.
T5159 BI 1744 hydrochloride Olodaterol is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and a...
T4963 Higenamine Higenamine is a novel α1 -adrenoceptor antagonist.
T3996 Dapiprazole Hydrochloride Dapiprazole Hydrochloride is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors in the smooth muscle of blood vessels (arteries, a...
T5035 Methoxyphenamine Hydrochloride Methoxyphenamine is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.
T5028 Landiolol hydrochloride Landiolol is an ultra-short-acting β1 selective adrenoceptor antagonist.
T5105 1-(2-Pyridyl)piperazine 1-(2-Pyridyl)piperazine is a selective α2-adrenoceptor antagonists. 1-(2-Pyridyl)piperazine shows sympatholytic activity. 1-(2-Pyridyl)piperazine is also a meta...
T4983 Isoetharine mesylate salt Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T4S0998 Trifolirhizin Trifolirhizin exerts varying degrees of inhibition on tyrosinase-dependent melanin biosynthesis, and therefore, are candidates as skin-whitening agents.Trifolirh...
T7079 Batefenterol Batefenterol (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hβ2-ad...
T4548 Procaterol hydrochloride Short-acting β2-adrenergic receptor agonist used to treat asthma.
T7046 Xylazine Xylazine is α2-adrenergic receptor agonist.
T7044 Norepinephrine Norepinephrine can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression of vascula...
T5S2178 Fargesin 1. Fargesin as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Fargesin improves d...
T4560 Alprenolol Alprenolol is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1A and 5-HT1B.
T4526 Piperoxan hydrochloride Piperoxan hydrochloride is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered.
T0172 Maprotiline hydrochloride Maprotiline hydrochloride is a bridged-ring tetracyclic antidepressant that is both mechanistically and functionally similar to the tricyclic antidepressants, in...
Isoprenaline hydrochloride HOT
T1056CAS 51-30-9
Isoproterenol is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
Naftopidil hydrochloride
T9220CAS 1164469-60-6
Naftopidil hydrochloride is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenocep...
Deoxycorticosterone acetate
T3033CAS 56-47-3
Desoxycorticosterone acetate is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of the adrenocortical...
Metoprolol tartrate
T0487CAS 56392-17-7
Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.
Naphazoline hydrochloride
T0446CAS 550-99-2
Naphazoline hydrochloride is an adrenergic vasoconstrictor agent used as a decongestant.
Nicardipine hydrochloride
T1215CAS 54527-84-3
Nicardipine Hydrochloride is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nicar...
Isoferulic acid
T2889CAS 537-73-5
3-Hydroxy-4-methoxycinnamic Acid exhibits hypoglycemic properties.
Promazine hydrochloride
T0766CAS 53-60-1
Promazine hydrochloride is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. It is primarily used in short-term treatm...
Tetrahydrozoline HCl
T6703CAS 522-48-5
Tetrahydrozoline HCl is an imidazoline derivative with alpha receptor agonist activity.
Trimipramine maleate
T1045CAS 521-78-8
Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin an...
Carteolol hydrochloride
T1282CAS 51781-21-6
Carteolol Hydrochloride is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocking agent for be...
Carbazochrome sodium sulfonate
T0852CAS 51460-26-5
Carbazochrome sodium sulfonate (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.
Epinephrine bitartrate
T1047CAS 51-42-3
L-Epinephrine Bitartrate is alpha- and beta-adrenergic receptor stimulator.
Salbutamol Sulfate
T6652CAS 51022-70-9
Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
Tulobuterol hydrochloride
T3277CAS 56776-01-3
Tulobuterol hydrochloride is a long-acting beta2-adrenergic receptor agonist.
Vilanterol
T2645CAS 503068-34-6
Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.
Scopine
T6662CAS 498-45-3
Scopine, the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
Taxifolin
T1738CAS 480-18-2
Taxifolin is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.
Formoterol Hemifumarate
T6505CAS 43229-80-7
Formoterol Hemifumarate, an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of chronic obstructive pulmonary disease(C...
Nadolol
T1203CAS 42200-33-9
Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities. Nadolol competitively blocks beta-1 adrenergic recepto...
Clonidine hydrochloride
T1247CAS 4205-91-8
Clonidine is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide ...
Piribedil
T3278CAS 3605-01-4
Piribedil is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
Buflomedil hydrochloride
T0317CAS 35543-24-9
Buflomedil hydrochloride, a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.
Urapidil
T0165CAS 34661-75-1
Urapidil, a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
Acebutolol hydrochloride
T1012CAS 34381-68-5
Acebutolol acts as a cardioselective beta-adrenergic antagonist with little effect on bronchial receptors and has intrinsic sympathomimetic properties. Acebutolo...
Metaraminol bitartrate
T0279CAS 33402-03-8
Metaraminol bitartrate is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in the...
(R)-(+)-Atenolol
T0007LCAS 56715-13-0
(R)-(+)-Atenolol is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.
Naftopidil
T0696CAS 57149-07-2
Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
DL-Adrenalin
T1071L2CAS 329-65-7
DL-Epinephrine(DL-Adrenaline) is a hormone and a neurotransmitter.
Methoxamine hydrochloride
T0993CAS 61-16-5
An alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
Phentolamine mesilate
T1275CAS 65-28-1
Phentolamine mesylate is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, ...
Yohimbine hydrochloride
T2142CAS 65-19-0
Yohimbine hydrochloride is a plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of ERECTILE DY...
Urapidil hydrochloride
T0088CAS 64887-14-5
Urapidil hydrochloride is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
Tizanidine hydrochloride
T0290CAS 64461-82-1
Tizanidine hydrochloride, an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
Dipivefrin hydrochloride
T0103CAS 64019-93-8
Dipivefrin that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
Phenoxybenzamine hydrochloride
T1158CAS 63-92-3
Phenoxybenzamine Hydrochloride is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive and...
Betaxolol hydrochloride
T0226CAS 63659-19-8
Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induced...
Betaxolol
T6408CAS 63659-18-7
Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
Terazosin hydrochloride
T0197CAS 63074-08-8
Terazosin, a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a drug of choice for patie...
Adrenalone hydrochloride
T0948CAS 62-13-5
Adrenalone hydrochloride, a selective α1-adrenoceptor agonist, is used as a topical hemostatic and vasoconstrictor and used to extend the effect of local anesth...
Phenylephrine hydrochloride
T0453CAS 61-76-7
Phenylephrine hydrochloride is a selective agonist of the α1-adrenergic receptor.
Carvedilol phosphate
T0342CAS 610309-89-2
Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intri...
Naftopidil DiHCl
T6600CAS 57149-08-3
Naftopidil DiHCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
Promethazine
T0445CAS 60-87-7
Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
Tolazoline hydrochloride
T1680CAS 59-97-2
Tolazoline is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.
Synephrine HCl
T6688CAS 5985-28-4
SynephrineHCl (Oxedrine, p-Synephrine) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
Orciprenaline sulfate
T0277CAS 5874-97-5
Orciprenaline sulfate is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
Perphenazine
T1090CAS 58-39-9
Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
Promethazine hydrochloride
T0445LCAS 58-33-3
Promethazine HCl(NSC-231688), the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mACh receptor, moder...
Desipramine hydrochloride
T0991CAS 58-28-6
Desipramine Hydrochloride a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervous system (CNS), d...
Isoxsuprine hydrochloride
T0324CAS 579-56-6
Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
Clozapine
T0455CAS 5786-21-0
Clozapine is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays...
Carazolol
T3284CAS 57775-29-8
Carazolol is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
Celiprolol hydrochloride
T1244CAS 57470-78-7
Celiprolol hydrochloride is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity. It is used in the management of ANGINA PE...
Amitraz
T1632CAS 33089-61-1
AMITRAZ is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic ma...
Labetalol hydrochloride
T0348CAS 32780-64-6
Labetalol hydrochloride, a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
Noradrenaline bitartrate
T0871CAS 69815-49-2
Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors. Norepinephrine Bitartrate is a bitartrate salt of norepinephrine, a synthetic phe...
ICI-118551 Hydrochloride
T6860CAS 1217094-53-5
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
Paliperidone
T0076CAS 144598-75-4
Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the pr...
Dronedarone hydrochloride
T1073CAS 141625-93-6
Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
Ziprasidone hydrochloride monohydrate
T0031CAS 138982-67-9
Ziprasidone(CP88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic activity.
Pindolol
T0735CAS 13523-86-9
Pindolol is a moderately lipophilic beta blocker (ADRENERGIC BETA-ANTAGONISTS). It is non-cardioselective and has intrinsic sympathomimetic actions, but little m...
Iloperidone
T1539CAS 133454-47-4
Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
Olanzapine
T1567CAS 132539-06-1
Olanzapine is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
Thioridazine hydrochloride
T0365CAS 130-61-0
Thioridazine, an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selectivity.
Escitalopram
T0185CAS 128196-01-0
Escitalopram is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol upta...
Doxepin hydrochloride
T1540CAS 1229-29-4
Doxepin Hydrochloride is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mech...
Ziprasidone hydrochloride
T0031LCAS 122883-93-6
Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
Xylometazoline hydrochloride
T0042CAS 1218-35-5
Xylometazoline Hydrochloride is an α-adrenoceptor agonist usually used as nasal decongestant.
Efloxate
T0151CAS 119-41-5
Efloxate, a vasodilator, is utilized in the treatment of chronic coronary insufficiency.
Ziprasidone
T0031L2CAS 146939-27-7
Ziprasidone is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
Levobetaxolol HCl
T6565CAS 116209-55-3
Levobetaxolol hydrochloride is a beta-adrenergic receptor inhibitor (beta blocker), used to lower the pressure in the eye in treating conditions such as glaucoma...
Dexmedetomidine
T2524CAS 113775-47-6
Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect of...
Quetiapine Fumarate
T6241CAS 111974-72-2
Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
Quetiapin
T0162CAS 111974-69-7
Quetiapine is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism of quetiapin...
Higenamine Hydrochloride
T3232CAS 11041-94-4
Higenamine(Hydrochloride) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein...
Noradrenaline bitartrate monohydrate
T1064CAS 108341-18-0
Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator.
Tamsulosin hydrochloride
T0210CAS 106463-17-6
Tamsulosin Hydrochloride is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.
Risperidal
T0351CAS 106266-06-2
Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
(±)-Bisoprolol hemifumarate
T0143CAS 104344-23-2
Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart, thereb...
Atipamezole hydrochloride
T6765CAS 104075-48-1
Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochlo...
Atipamezole
T6766CAS 104054-27-5
Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
Dexmedetomidine HCl
T6466CAS 145108-58-3
Dexmedetomidine hydrochloride is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE, which is t...
Ivabradine hydrochloride
T2535CAS 148849-67-6
Ivabradine hydrochloride is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, hy...
Propranolol hydrochloride
T0812CAS 318-98-9
Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGIN...
Ritodrine hydrochloride
T1433CAS 23239-51-2
Ritodrine binds to and activates beta-2 adrenergic receptors of myometrial cells in the uterus, which decreases the intensity and frequency of uterine contractio...
Indacaterol
T2320CAS 312753-06-3
Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.
Midodrine hydrochloride
T1577CAS 3092-17-9
Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergic...
Atenolol
T0007CAS 29122-68-7
Atenolol is a selective β1 receptor antagonist.
Guanfacine hydrochloride
T2150CAS 29110-48-3
Guanfacine hydrochloride is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.
Nicergoline
T1132CAS 27848-84-6
Nicergoline is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
Pardoprunox
T1769CAS 269718-84-5
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
Timolol Maleate
T0475CAS 26921-17-5
Timolol is a nonselective beta-adrenergic receptor blocker that is widely used for the therapy of hypertension, angina pectoris and prevention of vascular headac...
Gemfibrozil
T1415CAS 25812-30-0
Gemfibrozil interacts with peroxisome proliferator-activated receptors (PPARalpha) resulting in PPARalpha-mediated stimulation of fatty acid oxidation and an inc...
Trazodone hydrochloride
T1619CAS 25332-39-2
Trazodone hydrochloride is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients with major depress...
Droxidopa
T2547CAS 23651-95-8
Droxidopa is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes of auton...
Guanabenz Acetate
T6522CAS 23256-50-0
Guanabenz Acetate is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is ...
Xylazine hydrochloride
T1500CAS 23076-35-9
Xylazine hydrochloride is an adrenergic alpha-2 agonist used as a sedative, analgesic and centrally acting muscle relaxant in veterinary medicine
Nebivolol hydrochloride
T0154CAS 152520-56-4
Nebivolol hydrochloride is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR through the endothelial L-argin...
Terbutaline Sulfate
T1584CAS 23031-32-5
Terbutaline sulfate is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
Mirabegron
T1671CAS 223673-61-8
Mirabegron is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
Mianserin hydrochloride
T0783CAS 21535-47-7
Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin r...
BMY 7378 dihydrochloride
T3046CAS 21102-95-4
BMY-7378, α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
2-(1-Piperazinyl)pyrimidine
T1696CAS 20980-22-7
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
Pimozide
T2546CAS 2062-78-4
Pimozide is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic rec...
Amiodarone hydrochloride
T1496CAS 19774-82-4
Amiodarone hydrochloride is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action by inhibiting POT...
Prazosin hydrochloride
T1050CAS 19237-84-4
Prazosin Hydrochloride reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism not complete...
Salbutamol
T1139CAS 18559-94-9
Albuterol stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3', ...
Anisodamine
T0970CAS 17659-49-3
Anisodamine is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
Silodosin
T1504CAS 160970-54-7
Silodosin is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
L755507
T6872CAS 159182-43-1
L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).
Clorprenaline hydrochloride
T0248CAS 6933-90-0
Clorprenaline Hydrochloride is a beta-2 adrenergic agonist with bronchodilator activity.
Terazosin hydrochloride dihydrate
T6701CAS 70024-40-7
Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
L-765314
T5511CAS 189349-50-6
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the r...
Ancarolol
T14287CAS 75748-50-4
Ancarolol is a blocking agent of beta-adrenergic.
ZK-90055 hydrochloride
T13403CAS 84638-81-3
ZK-90055 hydrochloride is an agonist of β2 adrenergic receptor.
CGP 20712 A
T10778CAS 105737-62-0
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
Vatinoxan hydrochloride
T13285CAS 130466-38-5
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
Dopexamine hydrochloride
T11318CAS 86484-91-5
Dopexamine hydrochloride is a β2-adrenergic receptor agonist.
Fiduxosin
T11286CAS 208993-54-8
Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
Solabegron
T12970CAS 252920-94-8
Solabegron is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(EC50 : 22 ...
Salmeterol
T12829CAS 89365-50-4
Salmeterol is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
(S)-Terazosin
T12815CAS 109351-33-9
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor ...
D2343
T15042CAS 72734-63-5
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
Arbutamine
T10364CAS 128470-16-6
Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure....
(R)-Terazosin
T12643CAS 109351-34-0
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values o...
Tizanidine
T7065CAS 51322-75-9
Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
M443
T15943CAS 1820684-31-8
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
Vilanterol trifenatate
T5134CAS 503070-58-4
Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7...
SR59230A
T13016CAS 174689-39-5
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
DL-Norepinephrine hydrochloride
T13655CAS 55-27-6
DL-Norepinephrine hydrochloride is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 μM.
Diacetolol D7
T11036CAS 1346604-19-0
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
Midaglizole hydrochloride
T11015CAS 79689-25-1
Midaglizole hydrochloride (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6....
Detomidine carboxylic acid
T11010CAS 115664-39-6
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also ...
Dabuzalgron
T10952CAS 219311-44-1
Dabuzalgron is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicity caused by do...
Phentolamine Analogue 1
T12444CAS 47142-51-8
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
Penbutolol sulfate
T12402CAS 38363-32-5
Penbutolol sulfate is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.
Benzquinamide
T12343CAS 63-12-7
Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
OPC-28326
T13804CAS 167626-17-7
OPC-28326 is a selective peripheral vasodilator and an α2-adrenergic receptor angatonist(α2A-, α2B- and α2C-adrenoceptors with Ki of 2040, 285, and 55 nM, ...
(±)-Methotrimeprazine (D6)
T13470CAS 1189805-51-3
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
KUL 7211 racemate
T11786CAS 911196-40-2
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
Tetrahydroalstonine
TN2267CAS 6474-90-4
Tetrahydroalstonine and Raubasine preferentially block the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogenou...
Stephanine
TN5061CAS 517-63-5
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
ACTH 1-14 acetate(25696-21-3 free base)
TP1238LCAS TP1238L
ACTH (1-14) is a fragment of adrenocorticotrophin, which regulates cortisol and androgen production.Adrenocorticotropic hormone (ACTH), also known as corticotrop...
Metipranolol
T8899CAS 22664-55-7
Metipranolol is a β-adrenergic receptor antagonist that is given orally for the treatment of hypertension and also applied topically to the cornea for treating ...
LUN42518 HCl 47142-51-8(free base)
T8738CAS T8738
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.
Terbutaline
T8810CAS 23031-25-6
Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol
Labetalol
T20570CAS 36894-69-6
Labetalol is a mixed alpha/beta-adrenergic antagonist.It is used to treat high blood pressure. It can be given by mouth for long term hypertension management or ...
Rotigotine Hydrochloride
T21446CAS 125572-93-2
Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
Propranolol HCl
T8696CAS 3506-09-0
Propranolol hydrochloride is a blocker of β1 and β2 adrenergic receptor
Norepinephrine bitartrate salt
T21066CAS 3414-63-9
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
Clenbuterol
T21147CAS 37148-27-9
Clenbuterol is a substituted phenylaminoethanol that has β2 adrenomimetic properties at very low doses, and is used as a bronchodilator in asthma.
nifenalol.HCl
T8663CAS 5704-60-9
Nifenalol is a antagonist of β-adrenergic receptor.
RX 821002 hydrochloride
T23283CAS 109544-45-8
α2-adrenoceptor antagonist
Quinine HCl
TN4882CAS 130-89-2
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
Ritanserin
T16759CAS 87051-43-2
Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adren...
Isorauhimbine
TN4323CAS 483-09-0
3-Epi-alpha-yohimbine(Isorauhimbine) has alpha adrenoceptor blocking activities,it also has cardiovascular effects.
beta-Yohimbine
TN3507CAS 549-84-8
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor block...
Akuammigine
TN3368CAS 642-17-1
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
Agrimonolide
TN3364CAS 21499-24-1
Agrimonolide is a potential α1 adrenergic receptor antagonist, it exerts anti-inflammatory activity, at least in part, via suppressing LPS-induced activation of...
Practolol
T8595CAS 6673-35-4
Practolol is a selective β-adrenoceptor blocker.
Bupranolol
T8580CAS 14556-46-8
Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic...
Prazosin
T22406CAS 19216-56-9
Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
Bisoprolol
T22275CAS 66722-44-9
Bisoprolol is a cardioselective β1-adrenergic blocker used for secondary prevention of heart failure, myocardial, angina pectorisinfarction (MI) and mild to mod...
Phenylephrine
T17310CAS 59-42-7
Phenylephrine is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
Lusaperidone
T11894CAS 214548-46-6
Lusaperidone is an α2 adrenergic receptor antagonist, with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively.
Ro 363
T16769CAS 74513-77-2
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
Phentolamine
T8348CAS 50-60-2
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
Meranzin hydrate
TN1922CAS 5875-49-0
Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-h...
Brimonidine Tartrate
T6422CAS 70359-46-5
Brimonidine tartrate is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pressure associated with...
Medetomidine HCl
T6579CAS 86347-15-1
Medetomidine is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
Metoprolol Succinate
T3165CAS 98418-47-4
Metoprolol succinate is a selective adrenergic beta-1 blocking agent that is commonly used to treat ANGINA PECTORIS; HYPERTENSION; and CARDIAC ARRHYTHMIAS.
Cisatracurium besylate
T1459CAS 96946-42-8
Cisatracurium Besylate is a nondepolarizing skeletal muscle relaxant for intravenous administration.
Moxisylyte hydrochloride
T0394CAS 964-52-3
Moxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
Sotalol hydrochloride
T0483CAS 959-24-0
Sotalol Hydrochloride is the hydrochloride salt form of sotalol, an ethanolamine derivative with Class III antiarrhythmic and antihypertensive properties.
Salmeterol Xinafoate
T6653CAS 94749-08-3
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstru...
Synephrine
T1287CAS 94-07-5
Synephrine is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
Brexpiprazole
T2306CAS 913611-97-9
Brexpiprazole is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.
Detomidine HCl
T6464CAS 90038-01-0
Detomidine HCl produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
Nortriptyline hydrochloride
T1327CAS 894-71-3
Nortriptyline hydrochloride is a metabolite of AMITRIPTYLINE that is also used as an antidepressive agent. Nortriptyline is used in major depression, dysthymia, ...
Gramine
T6519CAS 87-52-5
Gramine, a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for ...
Olodaterol
T3457CAS 868049-49-4
Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors lo...
Scopine HCl
T6663CAS 85700-55-6
Scopine HCl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
Rauwolscine hydrochloride
T4429CAS 6211-32-1
Rauwolscine, a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potent...
Mirtazapine
T0137CAS 85650-52-8
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
Nylidrin hydrochloride
T0173CAS 849-55-8
Nylidrin hydrochloride was an effective inhibitor of the IgG1-mediated release of histamine from passively sensitized guinea pig lung slices, and of the IgE-medi...
Tetryzoline
T0397CAS 84-22-0
Tetrahydrozoline, an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of the eye resulted...
Bambuterol hydrochloride
T1446CAS 81732-46-9
Bambuterol, a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
Alfuzosin hydrochloride
T0091CAS 81403-68-1
Alfuzosin hydrochloride is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).
Esmolol hydrochloride
T1503CAS 81161-17-3
Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instan...
Idazoxan hydrochloride
T0115CAS 79944-56-2
Idazoxan hydrochloride is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
Doxazosin mesylate
T0101CAS 77883-43-3
Doxazosin mesylate(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
Indacaterol maleate
T1239CAS 753498-25-8
Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
Formoterol
T2580CAS 73573-87-2
Arformoterol is an adrenergic β-2 receptor agonist with a prolonged duration of action. It is used to manage asthma and in the treatment of chronic obstructive ...
Carvedilol
T0447CAS 72956-09-3
Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intri...
DL-Adrenaline Hydrochloride
T1071LCAS 329-63-5
DL-Adrenaline Hydrochloride is the hydrochloride salt of the naturally occurring sympathomimetic amine with vasoconstricting, intraocular pressure-reducing activ...
Pergolide mesylate salt
T2226CAS 66104-23-2
PERGOLIDE MESYLATE is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due to...
Isorhoifolin
TN1797CAS 552-57-8
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
Clonidine
T7045CAS 4205-90-7
Clonidine is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide-...
Fenoterol
T8358CAS 13392-18-2
Fenoterol is an  agonist of  β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.
Bevantolol hydrochloride
T8143CAS 42864-78-8
Bevantolol hydrochloride is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.
Dobutamine (hydrochloride)
T8149CAS 49745-95-1
Dobutamine (hydrochloride) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
Anisodamine Hydrobromide
T8304CAS 55449-49-5
Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
Yohimbine
TCS2185CAS 146-48-5
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
Levalbuterol tartrate
T7164CAS 661464-94-4
Levosalbutamol tartrate is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
Lofexidine
T7160CAS 31036-80-3
Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
GUANABENZ
T5471CAS 5051-62-7
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
DL-071-IT
T5450CAS 55104-39-7
DL 071-IT is a potent non-selective beta-adrenoceptor antagonist. DL 071 IT showed intrinsic sympathomimetic activity and weak membrane stabilizing activity.
Amezinium (methylsulfate)
T5327CAS 30578-37-1
Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition of noradrenaline and tyramine uptake.
BI 1744 hydrochloride
T5159CAS 869477-96-3
Olodaterol is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and a...
Higenamine
T4963CAS 5843-65-2
Higenamine is a novel α1 -adrenoceptor antagonist.
Dapiprazole Hydrochloride
T3996CAS 72822-13-0
Dapiprazole Hydrochloride is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors in the smooth muscle of blood vessels (arteries, a...
Methoxyphenamine Hydrochloride
T5035CAS 5588-10-3
Methoxyphenamine is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.
Landiolol hydrochloride
T5028CAS 144481-98-1
Landiolol is an ultra-short-acting β1 selective adrenoceptor antagonist.
1-(2-Pyridyl)piperazine
T5105CAS 34803-66-2
1-(2-Pyridyl)piperazine is a selective α2-adrenoceptor antagonists. 1-(2-Pyridyl)piperazine shows sympatholytic activity. 1-(2-Pyridyl)piperazine is also a meta...
Isoetharine mesylate salt
T4983CAS 7279-75-6
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
Trifolirhizin
T4S0998CAS 6807-83-6
Trifolirhizin exerts varying degrees of inhibition on tyrosinase-dependent melanin biosynthesis, and therefore, are candidates as skin-whitening agents.Trifolirh...
Batefenterol
T7079CAS 743461-65-6
Batefenterol (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hβ2-ad...
Procaterol hydrochloride
T4548CAS 81262-93-3
Short-acting β2-adrenergic receptor agonist used to treat asthma.
Xylazine
T7046CAS 7361-61-7
Xylazine is α2-adrenergic receptor agonist.
Norepinephrine
T7044CAS 51-41-2
Norepinephrine can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression of vascula...
Fargesin
T5S2178CAS 31008-19-2
1. Fargesin as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Fargesin improves d...
Alprenolol
T4560CAS 13655-52-2
Alprenolol is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1A and 5-HT1B.
Piperoxan hydrochloride
T4526CAS 135-87-5
Piperoxan hydrochloride is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered.
Maprotiline hydrochloride
T0172CAS 10347-81-6
Maprotiline hydrochloride is a bridged-ring tetracyclic antidepressant that is both mechanistically and functionally similar to the tricyclic antidepressants, in...