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Search Result

Search Results for " adenosine a1 receptor "

Targets

Adenosine Receptor

75

Compounds

4

Natural Products

2

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T14127 Adenosine A1 receptor activator T62 Adenosine Receptor
Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also reduces hypersensitivity in models of inflammatory and nerve...
T22466 Adenosine receptor A1 antagonist 5 cAMP
Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure.
T7683 Adenosine amine congener ADAC Adenosine Receptor
Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.
T27076 8-Cyclopentyl-1,3-dimethylxanthine CPT Adenosine Receptor
8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.
T12160 N6-Cyclohexyladenosine CHA Adenosine Receptor
N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm. N6-Cyclohexyladenosine exerts anticonvulsant effects and protects against neuronal death. CHA was also found to inhibit the pressor ...
T17023 Tecadenoson CVT-510 Adenosine Receptor
Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
T70722 N 0861 Adenosine Receptor
N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.
TQ0125 Capadenoson BAY 68-4986 Adenosine Receptor
Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.
T15655 KFM19 Adenosine Receptor
KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.
T29112 VPC171 VPC 171,VPC-171 Adenosine Receptor
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
T22744 DPCPX PD 116948 Adenosine Receptor
DPCPX (PD 116948) is an A1 adenosine receptor antagonist
T34914 Trabodenoson INNO-8875,INO-8875,PJ875,PJ-875,INNO 8875,INNO8875,PJ 875 Adenosine Receptor
Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.
T27323 FK-453 FK453,FK 453 Adenosine Receptor
FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.
T21519 CCPA 2-chloro-N(6)cyclopentyladenosine,2-CHLORO-N-CYCLOPENTYLADENOSINE Adenosine Receptor
CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor
T23347 SDZ WAG 994 Adenosine Receptor
SDZ WAG 994 is an A1 adenosine receptor agonist.
T16263 N6-Cyclopentyladenosine UK-80882,CPA Adenosine Receptor
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of 2.3 nM, 790 nM, and 43 nM for human A1, A2A, and A3 recepto...
T37792 A2A receptor antagonist 1 CPI-444 analog,A2A receptor antagonist 1 Adenosine Receptor
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
T16140 MRS 1754 Adenosine Receptor
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
T28748 Selodenoson RG14202,DTI0009,DTI-0009,RG-14202,DT-009,DT009 Adenosine Receptor
Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.
T39039 FSCPX Adenosine Receptor
FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency. Additionally, FSCPX can effectively decrease the interstitial adenosine level in the ...
T17117 Tonapofylline BG 9928 Adenosine Receptor
Tonapofylline is an orally active and selective antagonist of the A1 adenosine receptor (Ki: 7.4 nM for human A1). Tonapofylline can be used in studies about heart failure.
T67972L Amp579 TFA Amp579 TFA(213453-89-5 Free base) Adenosine Receptor
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.
T14944 CGS 15943 PI3K , Adenosine Receptor
CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM , respectively.
T6441 CGS 21680 Hydrochloride CGS 21680 HCl Adenosine Receptor
CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.
T16782 Rolofylline KW-3902,MK-7418,KF-15372 Adenosine Receptor
Rolofylline (KW-3902) is a selective adenosine A1 receptor antagonist used in the study of acute congestive heart failure and renal dysfunction, and in the study of neurodegenerative disorders.
T16136 MRS-1706 Adenosine Receptor
MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.
T16808 Runcaciguat Others , Guanylate cyclase
Runcaciguat is a soluble guanylate cyclase stimulator. Runcaciguat combines with selective partial adenosine A1 receptor agonists and can be used in studies about cardiovascular and renal diseases.
T2671 Regadenoson CVT-3146,Lexiscan Adenosine Receptor
Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadenoson selectively binds to and activates the A2A adenosine re...
T6884 Namodenoson 2-Cl-IB-MECA,CF-102 Adenosine Receptor
Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.
T22489 2'-MeCCPA 2-Chloro-N-cyclopentyl-2′-C-methyladenosine HCV Protease , Adenosine Receptor
2'-MeCCPA is a potent and highly selective A1 adenosine receptor (A1AR) agonist with a K-value of 1.8 nM for AR.2'-MeCCPA inhibits trichostatin-stimulated adenylate cyclase activity with an IC value of 13.1 nM.2'-MeCCPA ...
T6979 SCH 58261 SCH58261 Adenosine Receptor
SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.
T14506 BAY 60-6583 Others , Adenosine Receptor
BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3 receptors.BAY 60-6583 is cardioprotective in a model of myocardial...
T23202 PSB 36 Others
A1 adenosine receptor antagonist
T23130 PD 81723 Others
Allosteric potentiator at the adenosine A1 receptor
T27861 LUF5831 LUF 5831,LUF-5831
LUF5831 is an agonist of adenosine A1 receptor.
T70067 IRFI-165
IRFI-165 is an adenosine A1 receptor inhibitor
T27862 LUF5981 LUF-5981,LUF 5981
LUF5981 is a selective agonist of human adenosine A1 receptor.
T69450 DU172
DU172 is the tyrosine-targeted covalent adenosine A1 receptor antagonist.
T24384 L-97-1 L97-1,L 97-1
L-97-1 is an antagonist of the adenosine A1 receptor.
T23964 Dansyl-NECA DansylNECA
Dansyl-NECA is a selective agonist of fluorescent adenosine A1 receptor.
T31086 CPFPX [18F]CPFPX
CPFPX is a highly selective radioactive ligand for the A1 adenosine receptor (A1AR).
T28446 PQ-69 PQ69,PQ 69
PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.
T70827 MDL-102234
MDL-102234 is an adenosine A1 receptor antagonist.
T26565 Adentri BG-9719,BG9719,BG 9719,CVT124,CVT-124,CVT 124
Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.
T70667 KF 20274
KF 20274 is an adenosine A1 antagonist; purinergic receptor antagonist.
T24526 Neladenoson dalanate HCl Neladenoson dalanate hydrochloride
Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).
T26621 AMP-579 RPR100579,RPR 100579,AMP 579,RPR-100579
AMP-579 is an adenosine A1 receptor agonist. AMP-579 also acts as a A2b-adenosine receptor agonist in human 293 cells and rabbit hearts.
T14015 ST4206 Others
ST4206 is an antagonist of adenosine A2A. For adenosine A2A receptor and adenosine A1 receptor, the Kis values are 12 nM and 197 nM , respectively.
T26737 Bamifylline Hydrochloride BAX-2793Z,AC 3810,AC-3810,BAX2793Z,BAX 2793Z
Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.
T31068 CP-608039 UNII-A1LB8I4247
CP-608039 is a selective adenosine A3 receptor agonist for both human A3 and human A1 receptors.

Compounds

Adenosine A1 receptor activator T62
T14127
Synonym:
Target: Adenosine Receptor
Adenosine receptor A1 antagonist 5
T22466
Synonym:
Target: cAMP
Adenosine amine congener
T7683
Synonym: ADAC
Target: Adenosine Receptor
8-Cyclopentyl-1,3-dimethylxanthine
T27076
Synonym: CPT
Target: Adenosine Receptor
N6-Cyclohexyladenosine
T12160
Synonym: CHA
Target: Adenosine Receptor
Tecadenoson
T17023
Synonym: CVT-510
Target: Adenosine Receptor
N 0861
T70722
Synonym:
Target: Adenosine Receptor
Capadenoson
TQ0125
Synonym: BAY 68-4986
Target: Adenosine Receptor
KFM19
T15655
Synonym:
Target: Adenosine Receptor
VPC171
T29112
Synonym: VPC 171,VPC-171
Target: Adenosine Receptor
DPCPX
T22744
Synonym: PD 116948
Target: Adenosine Receptor
Trabodenoson
T34914
Synonym: INNO-8875,INO-8875,PJ875,PJ-875,INNO 8875,INNO8875,PJ 875
Target: Adenosine Receptor
FK-453
T27323
Synonym: FK453,FK 453
Target: Adenosine Receptor
CCPA
T21519
Synonym: 2-chloro-N(6)cyclopentyladenosine,2-CHLORO-N-CYCLOPENTYLADENOSINE
Target: Adenosine Receptor
SDZ WAG 994
T23347
Synonym:
Target: Adenosine Receptor
N6-Cyclopentyladenosine
T16263
Synonym: UK-80882,CPA
Target: Adenosine Receptor
A2A receptor antagonist 1
T37792
Synonym: CPI-444 analog,A2A receptor antagonist 1
Target: Adenosine Receptor
MRS 1754
T16140
Synonym:
Target: Adenosine Receptor
Selodenoson
T28748
Synonym: RG14202,DTI0009,DTI-0009,RG-14202,DT-009,DT009
Target: Adenosine Receptor
FSCPX
T39039
Synonym:
Target: Adenosine Receptor
Tonapofylline
T17117
Synonym: BG 9928
Target: Adenosine Receptor
Amp579 TFA
T67972L
Synonym: Amp579 TFA(213453-89-5 Free base)
Target: Adenosine Receptor
CGS 15943
T14944
Synonym:
Target: PI3K, Adenosine Receptor
CGS 21680 Hydrochloride
T6441
Synonym: CGS 21680 HCl
Target: Adenosine Receptor
Rolofylline
T16782
Synonym: KW-3902,MK-7418,KF-15372
Target: Adenosine Receptor
MRS-1706
T16136
Synonym:
Target: Adenosine Receptor
Runcaciguat
T16808
Synonym:
Target: Others, Guanylate cyclase
Regadenoson
T2671
Synonym: CVT-3146,Lexiscan
Target: Adenosine Receptor
Namodenoson
T6884
Synonym: 2-Cl-IB-MECA,CF-102
Target: Adenosine Receptor
2'-MeCCPA
T22489
Synonym: 2-Chloro-N-cyclopentyl-2′-C-methyladenosine
Target: HCV Protease, Adenosine Receptor
SCH 58261
T6979
Synonym: SCH58261
Target: Adenosine Receptor
BAY 60-6583
T14506
Synonym:
Target: Others, Adenosine Receptor
PSB 36
T23202
Synonym:
Target: Others
PD 81723
T23130
Synonym:
Target: Others
LUF5831
T27861
Synonym: LUF 5831,LUF-5831
Target:
IRFI-165
T70067
Synonym:
Target:
LUF5981
T27862
Synonym: LUF-5981,LUF 5981
Target:
DU172
T69450
Synonym:
Target:
L-97-1
T24384
Synonym: L97-1,L 97-1
Target:
Dansyl-NECA
T23964
Synonym: DansylNECA
Target:
CPFPX
T31086
Synonym: [18F]CPFPX
Target:
PQ-69
T28446
Synonym: PQ69,PQ 69
Target:
MDL-102234
T70827
Synonym:
Target:
Adentri
T26565
Synonym: BG-9719,BG9719,BG 9719,CVT124,CVT-124,CVT 124
Target:
KF 20274
T70667
Synonym:
Target:
Neladenoson dalanate HCl
T24526
Synonym: Neladenoson dalanate hydrochloride
Target:
AMP-579
T26621
Synonym: RPR100579,RPR 100579,AMP 579,RPR-100579
Target:
ST4206
T14015
Synonym:
Target: Others
Bamifylline Hydrochloride
T26737
Synonym: BAX-2793Z,AC 3810,AC-3810,BAX2793Z,BAX 2793Z
Target:
CP-608039
T31068
Synonym: UNII-A1LB8I4247
Target:
1 2
Cat No. Product Name Synonyms Targets
TN2247 Swertisin Adenosine Receptor
Swertisin, a novel herbal biomolecule, shows a strong antihyperglycemic action. Swertisin is an adenosine A1 receptor antagonist, is known to have antidiabetic, anti-inflammatory and antioxidant effects.
T2133 Adenosine monophosphate 5'-Adenylic acid,AMP,Adenosine 5'-monophosphate Endogenous Metabolite , AMPK
Adenosine monophosphate (AMP) is a purine ribonucleoside 5'-monophosphates and a key cellular metabolite in signal transduction and regulation of energy homeostasis.It has a role as an EC 3.1.3.11 (fructose-bisphosphatas...
T10822 Cirsimarin Cirsitakaoside Adenosine Receptor
Cirsimarin (Cirsitakaoside) is a flavonoid isolated from Microtea debilis. It shows a potent antilipogenic effect and decreases adipose tissue deposition in mice. Cirsimarin has antagonist activity on the adenosine A1 re...
T5940 Proxyphylline 7-(2-Hydroxypropyl)theophylline PDE , Adenosine Receptor
Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor. Proxyphylline acts as a cardiac stimulant, vasodilator and bronchodilator.

Natural Products

Swertisin
TN2247
Synonym:
Target: Adenosine Receptor
Adenosine monophosphate
T2133
Synonym: 5'-Adenylic acid,AMP,Adenosine 5'-monophosphate
Target: Endogenous Metabolite, AMPK
Cirsimarin
T10822
Synonym: Cirsitakaoside
Target: Adenosine Receptor
Proxyphylline
T5940
Synonym: 7-(2-Hydroxypropyl)theophylline
Target: PDE, Adenosine Receptor

Recombinant Proteins

Species：
Human (2)
Expression System：
HEK293 (1)
in vitro E. coli expression system (1)
Tag：
(1)
N-terminal 10xHis-tagged (1)
Cat No. Product Name Species Expression System
TMPH-00892 A1AR Protein, Human, Recombinant (His) Human in vitro E. coli expression system
Receptor for adenosine. The activity of this receptor is mediated by G proteins which inhibit adenylyl cyclase.
TMPK-00861 A2AR Protein-VLP, Human, Recombinant Human HEK293
Adenosine is a neuromodulator in the adult central nervous system. Membrane-bound receptors for adenosine have been identified and cDNAs for A1, A2a, A2b, and A3 adenosine receptor subtypes have been cloned recently.Expr...
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