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vactosertib hydrochloride

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Vactosertib Hydrochloride
TEW-7197 Hydrochloride, NOV1301 Hydrochloride, NOV 1301 Hydrochloride, EW-7197 Hydrochloride
T152621352610-25-3
Vactosertib Hydrochloride (EW-7197 Hydrochloride) is an orally active and highly efficient ATP-competitive ALK5 (activin receptor-like kinase 5) inhibitor, a TGF-β receptor I inhibitor with anti-metastatic and anticancer properties. It sensitizes pancreatic cancer cells to gemcitabine by inhibiting their viability.
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1-2 weeks
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TargetMol
Vactosertib
TEW-7197, EW-7197
T64961352608-82-2
Vactosertib (EW-7197) is an orally bioavailable inhibitor of the serine/threonine kinase, transforming growth factor (TGF)-beta receptor type 1 (TGFBR1), also known as activin receptor-like kinase 5 (ALK5), with potential antineoplastic activity.
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