Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • P2Y Receptor
    (6)
  • 5-HT Receptor
    (1)
  • Apoptosis
    (1)
  • Autophagy
    (1)
  • Epigenetic Reader Domain
    (1)
  • P2X Receptor
    (1)
  • Others
    (5)
Filter
Search Result
Results for "

p2y4 receptor

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    16
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    1
    TargetMol | Peptide_Products
PPTN
T125301160271-30-6In house
PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.
  • Inquiry Price
6-8 weeks
Size
QTY
PPTN hydrochloride
T635341992047-65-0In house
PPTN hydrochloride is a potent, high-affinity, competitive, and highly selective P2Y14 receptor antagonist (KB: 434 pM) with no agonist or antagonist activity at P2Y1, P2Y2, P2Y4, P2Y6, P2Y11, P2Y12, or P2Y13 receptors, exhibiting anti-inflammatory and anti-immune effects.
  • Inquiry Price
6-8 weeks
Size
QTY
Indophagolin
T89461207660-00-1
Indophagolin is a potent, indoline-containing autophagy inhibitor with an IC50 of 140 nM, and it antagonizes the purinergic receptor P2X4 as well as P2X1 and P2X3 with IC50s of 2.71, 2.40, and 3.49 μM, respectively.
  • Inquiry Price
Size
QTY
TargetMol | Inhibitor Sale
MRS2698
T16139934014-05-8
MRS2698 is an effective and highly selective agonist of the P2Y2 receptor (EC50: 8 nM). MRS2698 also is >300-fold P2Y2-selective versus the P2Y4 and P2Y6 receptors.
  • Inquiry Price
3-6 months
Size
QTY
PSB-1114 tetrasodium
T166721657025-60-9
PSB-1114 tetrasodium shows >50-fold selectivity versus the P2Y4 (EC50: 9.3 μM) and P2Y6 (EC50: 7.0 μM) receptors. PSB-1114 tetrasodium is an effective, enzymatically stable, and subtype-selective P2Y2 receptor agonist (EC50: 134 nM) .
  • Inquiry Price
8-10 weeks
Size
QTY
UTPγS trisodium salt
T234991266569-94-1
P2Y2 and P2Y4 receptor agonist
  • Inquiry Price
10-14 weeks
Size
QTY
MRS 4062 triethylammonium salt
MRS-4062,MRS4062,MRS 4062
T280961309871-50-8
MRS 4062 triethylammonium salt is a selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively).
  • Inquiry Price
Size
QTY
MRS2179
MRS 2179,MRS-2179
T28099101204-49-3
MRS2179 is a competitive P2Y1 receptor antagonist (Kb = 100 nM) with no appreciable activity at P2Y2, P2Y4, or P2Y6 at concentrations up to 30 µM, or at P2Y12 and P2Y13. It inhibits ADP-induced platelet shape change and aggregation (pA2 = 6.55) in vitro a
  • Inquiry Price
6-8 weeks
Size
QTY
MRS 2578
T6172711019-86-2
MRS2578, an effective P2Y6 receptor antagonist with IC50 of 37 nM, shows insignificant inhibition at P2Y1, P2Y2, P2Y4, and P2Y11 receptors.
  • Inquiry Price
Size
QTY
MRS2179 tetrasodium hydrate
T64078
MRS2179 tetrasodium hydrate, a competitive antagonist of the P2Y1 receptor, acts on the turkey P2Y1 receptor (Kb: 102 nM, pA2: 6.99) and exhibits an inhibitory effect on platelet aggregation. IC50: 1.15 μM), P2X3 (IC50: 12.9 μM), P2X2, P2X4, P2Y2, P2Y4 and P2Y6 receptors.
  • Inquiry Price
10-14 weeks
Size
QTY
PSB-1114 triethylamine
T78080
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50 of 9.3 μM) and P2Y6 (EC50 of 7.0 μM) receptors [1].
  • Inquiry Price
Size
QTY
4-Thiouridine 5′-triphosphate tetralithium
4-Thio-UTP tetralithium
T7919620188-72-1
4-Thiouridine 5′-triphosphate tetralithium (4-Thio-UTP), a potent P2Y2 and P2Y4 receptor agonist, exhibits EC50 values of 35 nM for hP2Y2 and 350 nM for hP2Y4. It is utilized in crosslinking experiments and labeling of transcriptional complexes [1] [2].
  • Inquiry Price
8-10 weeks
Size
QTY
4-Thiouridine 5′-triphosphate disodium
4-Thio-UTP tetrasodium
T7919768507-49-3
4-Thiouridine 5′-triphosphate (4-Thio-UTP) tetrasodium functions as a potent agonist at P2Y 2 and P2Y 4 receptors, with half-maximal effective concentrations (EC50s) of 35 nM for hP2Y 2 and 350 nM for hP2Y 4. This compound is applicable in studies involving crosslinking experiments and labeling of the transcriptional complex [1] [2].
  • Inquiry Price
Size
QTY
UDP-β-S sodium
Uridine-5' O-(2-thiodiphosphate)
T83803
UDP-β-S, serving as a specific agonist for the purinergic P2Y6 receptor, effectively promotes inositol phosphate accumulation in 1321N1 cells containing P2Y6 receptors, with an EC50 value of 28 nM. This selectivity is evident when compared to its effects on cells expressing P2Y1, P2Y2, or P2Y4 receptors, where a concentration of 10 µM is used. Additionally, at a concentration of 1 µM, UDP-β-S stimulates DNA synthesis in isolated rat aorta smooth muscle cells.
  • Inquiry Price
3-6 months
Size
QTY
Rp-2'-Deoxyuridine-5'-O-(1-thiotriphosphate) sodium
Rp-dUTP-α-S
T83833
Rp-2'-Deoxyuridine-5'-O-(1-thiotriphosphate) (Rp-dUTP-α-S), a sulfur-containing nucleotide isomer and purinergic P2Y2 receptor agonist, preferentially promotes inositol phosphate accumulation in 1321N1 astrocytoma cells with P2Y2 receptors (EC50 = 12.5 µM) compared to those expressing P2Y4 receptors at a concentration of 10 µM.
  • Inquiry Price
3-6 months
Size
QTY
Uridine adenosine tetraphosphate
UP4A
T8950010527-48-7
Uridine adenosine tetraphosphate (UP4A) acts primarily as an endothelium-derived vasoconstrictor, exerting its effects mainly through the P2X1 receptor, and potentially through the P2Y2 and P2Y4 receptors as well. It is utilized in research related to cardiovascular diseases.
  • Inquiry Price
Size
QTY