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Compounds

Cat No. Product Name
T8433 HQNO Mitochondrial Metabolism
HQNO 是一种电子传递链抑制剂,对 complex III 的Kd 值为 64 nM,由P. aeruginosa 产生的。它是许多物种的线粒体NDH-2的有效抑制剂。
T5337 IACS-010759 IACS 10759,IACS10759,IACS-10759 Apoptosis , Mitochondrial Metabolism , Others
IACS010759 是一种口服有效的线粒体氧化磷酸化复合物 I 抑制剂。它在依赖 OXPHOS 的脑癌和急性髓性白血病模型中抑制增殖并诱导细胞凋亡,有研究复发/难治性 AML 和实体瘤潜力。
T9169 MPP+ iodide Mitochondrial Metabolism , Autophagy
MPP+ iodide 是一种 5-羟色胺转运体的高亲和力底物,也是一种神经毒素 MPTP 的有毒代谢物,通过选择性破坏黑质多巴胺能神经元,在动物模型中引起帕金森病症状。它被多巴胺转运体吸收进入多巴胺能神经元,通过影响呼吸链复合体 I 对线...
T0239 Lonidamine Diclondazolic Acid,DICA,AF1890,氯尼达明 Hexokinase , Apoptosis , Mitochondrial Metabolism
Lonidamine 是一种抗肿瘤药物,是己糖激酶、线粒体丙酮酸载体和质膜单羧酸转运蛋白抑制剂,同时也抑制线粒体复合物 II。
T9714 Atpenin A5 Potassium Channel
Atpenin A5 是高度特异性的complex II 抑制剂,IC50为 ~10 nM。Dolastatin 10也是有效的mKATP 通道激动剂,具有心脏保活的作用。
T4446 Tebufenpyrad MK239,吡螨胺,Pyranica,Comanche Mitochondrial Metabolism
Tebufenpyrad 是一种重要的农业化学杀螨剂,其作用类似于已知的线粒体毒物 rotenone。
T19714 Fenpyroximate Others
Fenpyroximate 是一种有效的杀螨剂。
T9491 Pyraclostrobin Antifungal , Antibacterial
Pyraclostrobin 是一种球果苷杀菌剂,可诱导 3T3-L1 细胞内甘油三酯的积累,还可抑制真菌和哺乳动物细胞的线粒体复合物 III 。
T10404 ATP synthase inhibitor 1 ATPase
ATP synthase inhibitor 1 是 F1/FO-ATP 合酶复合物 c 亚基的有效抑制剂,抑制线粒体通透性转换孔的开放。
T5114 Pyridaben Calcium Channel , Parasite
Pyridaben 是一种METI 杀螨剂,可抑制复合物 I 处的线粒体电子转运。它对多种螨虫具有活性,通过滤纸接触给药,在 25 mg/mL、100 mg/mL 和 200 mg/mL 的剂量下,分别诱导 100% 的C. malacce...
T14346 Aumitin Autophagy , Others
Aumitin 是一种基于二氨基嘧啶的自噬抑制剂,以剂量依赖性抑制饥饿和雷帕霉素诱导的自噬,IC50分别为 0.12 μM 和 0.24 μM。它通过靶向复合物 I 抑制线粒体呼吸。
T36141 Boscalid Mitochondrial Metabolism
Boscalid 是一种广谱羧酰胺类杀菌剂,通过与线粒体复合物 II/琥珀酸脱氢酶的泛醌位点结合来抑制真菌呼吸。
T62238 AMPK activator 4 AMPK
AMPK activator 4 是一种有效且具有选择性的AMPK激活剂,不抑制线粒体复合物 I。AMPK activator 4 选择性地激活肌肉组织中的 AMPK且剂量依赖性地改善正常小鼠的糖耐量,显著降低 db/db 糖尿病小鼠的空腹...
T27516 GW844520
GW844520 is a potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. fal...
TMPY-03511 COX5B Protein, Human, Recombinant (His Tag)
Cytochrome C oxidase (COX) is the terminal enzyme of the mitochondrial respiratory chain. It is a multi-subunit enzyme...
T34472 S1QEL S1-QEL,S-1QEL,S1QEL1.1,S1 QEL,S 1QEL
S1QEL is a suppressor of mitochondrial respiratory complex I site IQ electron leak which suppresses superoxide and/or H2...
T68508 Ametoctradin
Ametoctradin is a new Oomycete-specific fungicide and a potent Qo site inhibitor of the mitochondrial respiration comple...
T70032 NCI-006
NCI-006 is a potent new inhibitor of lactate dehydrogenase (LDH) that disrupts tumor growth in mice. LDH inhibition slow...
T26573 AG311 AG-311,AG 311
AG311 is an inhibitor of complex I and hypoxia-induced HIF-1α stabilization. In vitro, AG311 induces rapid necrosis in n...
T14293 Annonacin Others
Annonacin is an Acetogenin and promotes cytotoxicity via a pathway inhibiting the mitochondrial complex and it is the ac...
HQNO
T8433
synonym:
Target:
IACS-010759
T5337
synonym: IACS 10759,IACS10759,IACS-10759
Target:
MPP+ iodide
T9169
synonym:
Target:
Lonidamine
T0239
synonym: Diclondazolic Acid,DICA,AF1890,氯尼达明
Target:
Atpenin A5
T9714
synonym:
Target:
Tebufenpyrad
T4446
synonym: MK239,吡螨胺,Pyranica,Comanche
Target:
Fenpyroximate
T19714
synonym:
Target:
Pyraclostrobin
T9491
synonym:
Target:
ATP synthase inhibitor 1
T10404
synonym:
Target:
Pyridaben
T5114
synonym:
Target:
Aumitin
T14346
synonym:
Target:
Boscalid
T36141
synonym:
Target:
AMPK activator 4
T62238
synonym:
Target:
GW844520
T27516
synonym:
Target:
COX5B Protein, Human, Recombinant (His Tag)
TMPY-03511
synonym:
Target:
S1QEL
T34472
synonym: S1-QEL,S-1QEL,S1QEL1.1,S1 QEL,S 1QEL
Target:
Ametoctradin
T68508
synonym:
Target:
NCI-006
T70032
synonym:
Target:
AG311
T26573
synonym: AG-311,AG 311
Target:
Annonacin
T14293
synonym:
Target:
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