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Results for "

mdv 3100

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    5
    TargetMol | Inhibitors_Agonists
  • Isotope Products
    2
    TargetMol | Isotope_Products
Enzalutamide
MDV3100
T6002915087-33-1
Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP) that activates autophagy, exhibits antitumor activity, and is commonly used in treating desmoplasia-resistant prostate cancer.
  • $40
In Stock
Size
QTY
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TargetMol | Citations Cited
N-desmethyl Enzalutamide
N-desmethyl MDV 3100
T194501242137-16-1
N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and secondary pharmacodynamics of similar potency to Enzalutamide and circulates at approximately the same plasma concentrations as enzalutamide.
  • $29
In Stock
Size
QTY
Enzalutamide-d3
MDV3100 D3
T112081443331-82-5
Enzalutamide D3 is a deuterium labeled Enzalutamide . Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells.
  • $108
5 days
Size
QTY
Enzalutamide carboxylic acid
T82171242137-15-0
Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
  • $60
In Stock
Size
QTY
N-desmethyl Enzalutamide D6
N-desmethyl MDV 3100 D6
T19449
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
  • $596
7-10 days
Size
QTY