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  • Melanocortin Receptor
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Results for "

mc2r

" in TargetMol Product Catalog.
  • Inhibitors & Agonists
    4
    TargetMol | All_Pathways
  • Recombinant Protein
    1
    TargetMol | Recombinant_Protein
  • Atumelnant
    CRN04894, CRN 04894
    T860912392970-97-5
    Atumelnant (CRN04894) is a selective and potent MC2R antagonist that inhibits ACTH-stimulated corticosterone secretion in a dose-dependent manner for the study of congenital adrenocortical hyperplasia (CAH) and Cushing's disease (CD).
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    10-14 weeks
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  • Dersimelagon
    MT-7117
    T253101835256-48-8
    Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values ​​of 8.16, 3.91, 1.14, and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m), and rat (r) MC1R, respectively. Dersimelagon exhibits good affinity for hMC1R and hMC4R, with Ki values ​​of 2.26 and 32.9 nM, respectively. Dersimelagon can be used in the study of skin pigmentation[1].
    • $72
    In Stock
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  • ATMW-2
    T203063
    ATMW-2 is an antagonist engineered using NeuralGenThesis (NGT) technology, specifically targeting the melanocortin 2 receptor (MC2R).
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    Inquiry
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  • GPS1573
    T888802445822-54-6
    GPS1573 is a non-competitive antagonist of the melanocortin 2 receptor (MC2R) that blocks the ACTH-stimulated activity of MC2R in a dose-dependent manner (IC50=66 nM). Due to its high selectivity in antagonizing MC2R, GPS1573 is utilized for research in Cushings disease.
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