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(4)
By Target- GRK
- Aurora Kinase(1)
- Dopamine Receptor(1)
- ERK(1)
- PKA(1)
- ROCK(1)
- Others(2)
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Results for "
grk-2 inhibitor
" in TargetMol Product Catalog- Inhibitors & Agonists4
GRK2 Inhibitor
βARK1 Inhibitor
T2546424269-96-3
GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).
- $139
Size
QTY
GRK2 Inhibitor 2
T799132592436-21-8
GRK2 Inhibitor 2 (Compound 8h), with an IC50 of 19 nM for GRK2 and 137 nM for Aurora-A, enhances β-AR-mediated cAMP accumulation in GRK2-overexpressing HEK293 cells. It is utilized in congestive heart failure (HF) research [1].
- Inquiry Price
Size
QTY
GSK180736A
GSK180736
T3513817194-38-0
GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 μM) and >100-fold selectivity over other GRKs. It is a weak inhibitor of PKA (IC50: 30 μM), but highly effective against ROCK1 (IC50: 100 nM).
- $35
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QTY
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