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Results for "

encequidar

" in TargetMol Product Catalog.
  • Inhibitors & Agonists
    3
    TargetMol | All_Pathways
  • Encequidar
    HM30181A, HM30181
    T8426849675-66-7
    Encequidar (HM30181A) is a potent and selective P-glycoprotein inhibitor.
    • $41
    In Stock
    Size
    QTY
  • Encequidar mesylate
    HM30181A mesylate, HM30181 mesylate
    T11578L849675-87-2
    Encequidar mesylate (HM30181A mesylate) is a competitive P-glycoprotein inhibitor.
    • $35
    In Stock
    Size
    QTY
    TargetMol | Citations Cited
  • Encequidar, HCl
    T68568849675-88-3
    Encequidar, also known as HM-30181, is an oral P-glycoprotein (P-gp) inhibitor developed to enhance the oral bioavailability of P-gp substrate drugs. Encequidar showed the highest potency (IC(50)=0.63nM) among several MDR1 inhibitors, including cycloporin A, XR9576, and GF120918, and effectively blocked transepithelial transport of paclitaxel in MDCK monolayers (IC(50)=35.4nM). Encequidar is currently under clinical trials.
    • $1,520
    1-2 weeks
    Size
    QTY