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calmidazolium

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  • Inhibitors & Agonists
    2
    TargetMol | Inhibitors_Agonists
Calmidazolium (cation)
T6826095013-41-5
Calmidazolium (cation) is a powerful inhibitor of or red blood cell Ca -ATPase & Ca transport into inside-out red blood cell vesicles; an antagonist of calmodulin.
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6-8 weeks
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Calmidazolium chloride
R 24571
T1066757265-65-3
Calmidazolium chloride (R 24571) is a calmodulin (CaMK) antagonist with a Kd of 3 nM, which inhibits CaM-dependent phosphodiesterase (IC50 = 0.15 μM) and calmodulin-induced activation of erythrocyte Ca2+-transporting ATPase (IC50 = 0.35 μM). It also induces apoptosis in certain cancer cell lines.
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6-8 weeks
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