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Nitracrine dihydrochloride is an acridine antineoplastic agent used in mammary and ovarian tumors. It inhibits RNA synthesis.

OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of 2040, 285, and 55 nM, respectively.

Phlorizin (Phloridzin) is a non-selective SGLT inhibitor found in apple, for hSGLT1( Ki=300 nM) and hSGLT2( Ki=39 nM) .

Trimelamol (CB10-375; NSC283162) is an efficient acid-catalyzed DNA interstrand cross-linker with low neurotoxicity due to its limited penetration of the blood-brain barrier. It exhibits antitumor activity and can overcome platinum resistance. Trimelamol is utilized in research concerning lung and ovarian cancers.

N-Trifluoroacetyladriamycin is a metabolite of Valrubicin (N-trifluoroacetyladriamycin-14-valerate, trade name Valstar). Valrubicin is a chemotherapy drug utilized to treat bladder cancer. Valrubicin is the anthracycline doxorubicin analog and is administ

Valopicitabine, a NS5B inhibitor, is used potentially for the treatment of HCV infection.