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brexpiprazole s oxide

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  • Inhibitors & Agonists
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Brexpiprazole S-oxide
DM-3411
T106121191900-51-2
Brexpiprazole S-oxide (DM-3411), a primary metabolite of Brexpiprazole, acts as a partial agonist of human 5-HT1A and dopamine receptors with Ki values of 0.12 nM and 0.3 nM, respectively.
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3-6 months
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Brexpiprazole S-oxide D8
DM-3411 D8
T106112748605-29-8
Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium-labeled Brexpiprazole S-oxide, the primary metabolite of Brexpiprazole, which is a partial agonist of human 5-HT1A and dopamine receptors (Kis: 0.12 nM and 0.3 nM).
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