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Search Result

Search Results for "proteasome in 1"

Libraries

Protease Inhibitor Library HIF-1 Signaling Pathway Compound Library NF-κB Signaling Compound Library
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Compounds

Cat No. Product Name
T12561 Proteasome-IN-1 Proteasome
Proteasome-IN-1 is an inhibitor of proteasome.
T12818 S119-8 Influenza Virus
S119-8 是一种广谱甲型和乙型流感病毒抑制剂，抑制多种乙型流感病毒和耐奥司他韦的甲型流感病毒。
T2S1837 Steviol 甜菊醇,Hydroxydehydrostevic acid,NSC 226902 Others
Steviol 是一种甜菊糖甙的主要代谢物。它能降低 AQP2 的表达，并促进 AQP2 的降解，从而减缓肾囊肿的生长。
T76243 Proteasome-activating peptide 1 TFA
Proteasome-activating peptide 1 TFA 是一种肽，是一种有效的蛋白酶体激活剂。Proteasome-activating peptide 1 TFA 可增加胰凝乳蛋白酶样蛋白酶体催化活性，从而提高体外和培养中...
T16795 Rpn11-IN-1 Capzimin intermediate Others
Rpn11-IN-1 is an effective and selective inhibitor of proteasome subunit Rpn11 (IC50: 390 nM).
T63321 20S Proteasome activator 1
20S Proteasome activator 1 是 20S 蛋白酶的有效激活剂，能够作用于胰蛋白酶样位点 (IC50: 0.3 μM)、胰凝乳蛋白酶样位点 (IC50: 0.7 μM)和半胱天冬酶位点 (IC50: 1.8 μM)。2...
T62255 20S Proteasome-IN-4
20S Proteasome-IN-4 (Compound 7) 是一种能透过血脑屏障的、寄生虫选择性的、具有口服活性的20Sproteasome 抑制剂，对T. b. brucei20S 蛋白酶体的IC50为 6.3 nM。20S Pro...
T72762 Proteasome-IN-4
Proteasome-IN-4 是一种良好的非共价 proteasome 抑制剂 (IC50= 8.39 nM)。Proteasome-IN-4 对 RPMI-8226、MM-1S 和 MV-4-11 细胞系具有较强的抗增殖活性。Prote...
T68869 TP-110
TP-110 is a new proteasome inhibitor, which shows potent growth inhibition in various tumor cell lines. Treatment with T...
T40255 VCP/p97 inhibitor-1 VCP/p97 inhibitor-1
VCP/p97 inhibitor-1, a highly effective compound, inhibits VCP/p97 (also known as Cdc48, CDC-48, or Ter94) with an IC 50...
T69880 YW2065
YW2065 has excellent anti-colorectal cancer effects in vitro and in vivo. YW2065 achieves its inhibitory activity for Wn...
T75870 PR-39 TFA
PR-39 TFA 是富含脯氨酸和精氨酸的天然抗菌肽，是一种非竞争性，可逆和变构的蛋白酶体 (proteasome) 抑制剂。PR-39 TFA 可逆地结合到蛋白酶体的 α7 亚基上，并通过泛素-蛋白酶体途径阻断 NF-κB 抑制剂 IκB...
T74878 Enzyme-IN-1
Enzyme-IN-1 (compound 1) 是一种基于肽的 N 端亲核试剂 (Ntn) 水解酶抑制剂。具体来说，Enzyme-IN-1 抑制 20S 蛋白酶体的糜胰蛋白酶样活性 (CT-L)。Enzyme-IN-1 可能具有潜在的抗炎...
T74755 TUS-007
TUS-007 是一种 CANDDY 分子，由蛋白酶体抑制剂修饰而成。然而，TUS-007 几乎不能抑制蛋白酶体活性。TUS-007 也是一种口服有效的KRASG12D/V 降解剂。TUS-007 可用于 KRAS G12D/V 无细胞化学...
T18543 Phthalimide-PEG4-MPDM-OH Others
Phthalimide-PEG4-MPDM-OH, a PROTAC linker with a PEGs composition, has applications in the synthesis of various PROTACs....
T75488 Leptosphaerodione
Leptosphaerodione，可从 Remotididymellasp. 中分离得到，是一种有效的泛素-蛋白酶体系统 (UPS) 抑制剂。Leptosphaerodione 在 HeLa 细胞中具有细胞毒性，IC50为 3.2 μM。...
T18544 Phthalimide-PEG4-PDM-OTBS Others
Phthalimide-PEG4-PDM-OTBS is a PROTAC linker comprised of polyethylene glycols (PEGs). This compound is utilized in the ...
T35481 DD 03-171
Potent and selective BTK Degrader (IC50 = 5.1 nM); degrades BTK in a proteasome- and CRBN-dependent manner. Suppresses B...
T17646 Boc-C1-PEG3-C4-OBn Others
Boc-C1-PEG3-C4-OBn (PROTAC Linker 15) is a PEG-based PROTAC linker employed in the synthesis of various PROTACs, includi...
T17647 Boc-C1-PEG3-C4-OH Others
Boc-C1-PEG3-C4-OH is an Alkyl/ether-based PROTAC linker utilized in the synthesis of PROTACs, which are characterized by...
Proteasome-IN-1
T12561
synonym:
Target:
S119-8
T12818
synonym:
Target:
Steviol
T2S1837
synonym: 甜菊醇,Hydroxydehydrostevic acid,NSC 226902
Target:
Proteasome-activating peptide 1 TFA
T76243
synonym:
Target:
Rpn11-IN-1
T16795
synonym: Capzimin intermediate
Target:
20S Proteasome activator 1
T63321
synonym:
Target:
20S Proteasome-IN-4
T62255
synonym:
Target:
Proteasome-IN-4
T72762
synonym:
Target:
TP-110
T68869
synonym:
Target:
VCP/p97 inhibitor-1
T40255
synonym: VCP/p97 inhibitor-1
Target:
YW2065
T69880
synonym:
Target:
PR-39 TFA
T75870
synonym:
Target:
Enzyme-IN-1
T74878
synonym:
Target:
TUS-007
T74755
synonym:
Target:
Phthalimide-PEG4-MPDM-OH
T18543
synonym:
Target:
Leptosphaerodione
T75488
synonym:
Target:
Phthalimide-PEG4-PDM-OTBS
T18544
synonym:
Target:
DD 03-171
T35481
synonym:
Target:
Boc-C1-PEG3-C4-OBn
T17646
synonym:
Target:
Boc-C1-PEG3-C4-OH
T17647
synonym:
Target:
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