Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T0165	Urapidil	34661-75-1	100%
T0165	Urapidil, a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
T1180	Blonanserin	132810-10-7	100%
T1180	Blonanserin is an atypical antipsychotic approved in Japan in January, 2008. Relative to many other antipsychotics, blonanserin has an improved tolerability prof...
T1012	Acebutolol hydrochloride	34381-68-5	100%
T1012	Acebutolol acts as a cardioselective beta-adrenergic antagonist with little effect on bronchial receptors and has intrinsic sympathomimetic properties. Acebutolo...
T0151	Efloxate	119-41-5	100%
T0151	Efloxate, a vasodilator, is utilized in the treatment of chronic coronary insufficiency.
TP1238L	ACTH 1-14 acetate(25696-21-3 free base)	TP1238L	100%
TP1238L	ACTH (1-14) is a fragment of adrenocorticotrophin, which regulates cortisol and androgen production.Adrenocorticotropic hormone (ACTH), also known as corticotrop...
T0173	Nylidrin hydrochloride	849-55-8	100%
T0173	Nylidrin hydrochloride was an effective inhibitor of the IgG1-mediated release of histamine from passively sensitized guinea pig lung slices, and of the IgE-medi...
T23253	RS 100329	1215654-26-4	100%
T23253	RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.
T6662	Scopine	498-45-3	100%
T6662	Scopine, the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
T0172	Maprotiline hydrochloride	10347-81-6	100%
T0172	Maprotiline hydrochloride is a bridged-ring tetracyclic antidepressant that is both mechanistically and functionally similar to the tricyclic antidepressants, in...
T0871	Noradrenaline bitartrate	69815-49-2	100%
T0871	Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors. Norepinephrine Bitartrate is a bitartrate salt of norepinephrine, a synthetic pheny...
T5134	Vilanterol trifenatate	503070-58-4	100%
T5134	Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, ...
T0342	Carvedilol phosphate hemihydrate	610309-89-2	100%
T0342	Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intri...
T1158	Phenoxybenzamine hydrochloride	63-92-3	100%
T1158	Phenoxybenzamine Hydrochloride is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive and...
T2320	Indacaterol	312753-06-3	100%
T2320	Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.
T8595	Practolol	6673-35-4	94.31%
T8595	Practolol is a selective β-adrenoceptor blocker.
TN1015	Meranzin	23971-42-8	95.08%
TN1015	Meranzin is an absorbed bioactive compound from the Traditional Chinese Medicine (TCM) Chaihu-Shugan-San (CSS). Meranzin, isolated from leaves of Murraya exotica...
T0445L	Promethazine hydrochloride	58-33-3	95.36%
T0445L	Promethazine HCl(NSC-231688), the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mACh receptor, moder...
T8580	Bupranolol	14556-46-8	95.85%
T8580	Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic....
T37906	Dibenamine hydrochloride	55-43-6	96.43%
T37906	Dibenamine hydrochloride is a competitive and irreversible adrenergic blocking agent and is known to modify the pharmacological effects of epinephrine. Dibenamin...
T6765	Atipamezole hydrochloride	104075-48-1	96.71%
T6765	Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochlor...