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niraparib metabolite m1

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  • Inhibitors & Agonists
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Niraparib metabolite M1
Niraparib carboxylic acid metabolite M1, M1 metabolite of niraparib
T122291476777-06-6In house
Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1) is the carboxylic acid metabolite of Niraparib. Niraparib is a novel poly (ADP-ribose) polymerase (PARP) inhibitor used in cancer research.
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6-8 weeks
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Niraparib metabolite M1 HCl
Niraparib metabolite M1 HCl (1476777-06-6 Free base), Niraparib carboxylic acid metabolite M1 HCl, M1 metabolite of niraparib HCl
T12229L
Niraparib metabolite M1 HCl is the active metabolite of Niraparib, as a novel targeted ADP ribose polymerase (PARP) inhibitor, it can competitively inhibit PARP1 and PARP2 to block the DNA repair mechanism of tumor cells and thus effectively inhibit the growth and proliferation, which is commonly used in the study of ovarian cancer, fallopian tube cancer and primary peritoneal cancer, and is commonly used in the study of ovarian, fallopian tube and primary peritoneal cancers.
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