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Results for "
molibresib besylate
" in TargetMol Product Catalog- Inhibitors & Agonists1
Molibresib besylate
I-BET 762 besylate, GSK 525762C
T11472L1895049-20-3
Molibresib besylate (GSK 525762C) is a selective and potent inhibitor of the bromodomain and extra-terminal (BET) family of proteins with potential anticancer activity for the study of refractory hematologic malignant diseases.Molibresib besylate generates reactive oxygen species (ROS), which potentiate ATM activation.
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T114721260530-25-3
GSK 525768A, the inactive enantiomer of GSK525762A, exhibits no activity towards BET.
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I-BET 762, GSK525762, GSK 525762A
T19061260907-17-2
Molibresib (GSK525762) is an inhibitor of BET proteins (IC50: about 35 nM).
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