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Results for "

mk 0457

" in TargetMol Product Catalog.
  • Inhibitors & Agonists
    2
    TargetMol | All_Pathways
  • Tozasertib
    VX 680, MK-0457
    T2509639089-54-6
    Tozasertib (MK-0457) is a pan-Aurora kinase inhibitor (Kis: 0.6/18/4.6 nM for Aurora A/Aurora B/Aurora C). It shows selectivity against more than 190 different kinases.
    • $40
    In Stock
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    TargetMol | Citations Cited
  • Tozasertib lactate
    T68415899827-04-4
    Tozasertib lactate is a potent and selective small-molecule inhibitor of the Aurora kinases which suppresses tumor growth by inducing apoptosis in tumor cells in which Aurora kinases are overexpressed.
    • $1,520
    6-8 weeks
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