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midostaurin-d-5

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  • Inhibitors & Agonists
    2
    TargetMol | Inhibitors_Agonists
  • Isotope Products
    2
    TargetMol | Isotope_Products
Midostaurin-D5
PKC412-D5,CGP 41251-D5
T12036
Midostaurin-D5 is a deuterium labeled Midostaurin.
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7-10 days
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3-Hydroxy Midostaurin-D5
CGP52421-D5
T19119
3-Hydroxy Midostaurin-D5 (CGP52421-D5) is a deuterium-labeled 3-Hydroxy Midostaurin which is a metabolite of PKC412. PKC412 effectively inhibits FMS-like tyrosine kinase-3 (FLT3) autophosphorylation (IC50s: 132 nM and 9.8 μM in culture medium and plasma).
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