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Results for "

lurasidone

" in TargetMol Product Catalog.
  • Inhibitors & Agonists
    16
    TargetMol | All_Pathways
  • Isotope Products
    9
    TargetMol | Isotope_Products
  • Reference Standards
    3
    TargetMol | Standard_Products
Lurasidone
SM-13496
T21337367514-87-2
Lurasidone (SM-13496) is an antagonist of dopamine D2 and 5-HT7 receptors (IC50 = 1.68 and 0.495 nM, respectively) and a partial agonist of the 5-HT1A receptor (IC50 = 6.75 nM).
  • $39
In Stock
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TargetMol | Citations Cited
Lurasidone D8 Hydrochloride
SM-13496 D8
T11892
Lurasidone-D8 hydrochloride is an inhibitor of Dopamine D2, 5-HT2A, 5-HT7, 5-HT1A and noradrenaline α2C, and is the deuterium labeled Lurasidone Hydrochloride (T1735).
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Lurasidone metabolite 14326
T11893186204-33-1
Lurasidone metabolite 14326, an active metabolite of the atypical antipsychotic Lurasidone, functions effectively in the body.
  • $839
35 days
Size
QTY
Lurasidone metabolite 14326 hydrochloride
Lurasidone metabolite 14326 hydrochloride (186204-33-1 free base)
T11893L
Lurasidone metabolite 14326 hydrochloride, an active metabolite of the atypical antipsychotic Lurasidone, maintains its significant function in pharmacological efficacy.
  • Inquiry Price
3-6 months
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Lurasidone Metabolite 14283 hydrochloride
T13760186204-32-0
Lurasidone Metabolite 14283 hydrochloride is a major active metabolite of Lurasidone.
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3-6 months
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Lurasidone Metabolite 14283-D8
T19406
Lurasidone Metabolite 14283-D8 is the deuterium labeled Lurasidone Metabolite 14283 (T13760).
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Lurasidone Metabolite 14326-D8
T19407
Lurasidone Metabolite 14326-D8 is the deuterium labeled Lurasidone Metabolite 14326 (T11893).
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Lurasidone Inactive Metabolite 14283-D8
5α/6α-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers)
TMIH-0315
Lurasidone Inactive Metabolite 14283-D8 is a deuterated compound of Lurasidone Inactive Metabolite 14283 (T86832). Lurasidone Inactive Metabolite 14283 has a CAS number of 186204-31-9.
  • $857
7-10 days
Size
QTY
Lurasidone Inactive Metabolite 14326-D8
5β/6β-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers)
TMIH-0316
Lurasidone Inactive Metabolite 14326-D8 is a deuterated compound of Lurasidone Inactive Metabolite 14326 (T11893). Lurasidone Inactive Metabolite 14326 has a CAS number of 186204-33-1.
  • $857
7-10 days
Size
QTY
Lurasidone hydrochloride
SM-13496 Hydrochloride, Lurasidone HCl
T1735367514-88-3
Lurasidone hydrochloride (Lurasidone HCl) is a thiazole derivative and atypical antipsychotic agent that functions as a dopamine D2 receptor antagonist; serotonin 5-HT2 receptor antagonist, serotonin 5-HT7 receptor antagonist, an antagonist of the adrenergic α2A and α2C receptors, as well as a partial serotonin 5-HT1A receptor agonist. It is used in the treatment of schizophrenia and bipolar disorder.
  • $35
In Stock
Size
QTY
TargetMol | Citations Cited
Lurasidone metabolite 14283
T86832186204-31-9
Lurasidone metabolite 14283, an active metabolite of lurasidone, can be utilized in antipsychotic research [1].
  • $1,120
35 days
Size
QTY
lurasidone-D8
TMIH-03131132654-54-6
lurasidone-D8 is a deuterated compound of lurasidone (TMSM-3492).
  • $889
7-10 days
Size
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Lurasidone-D8 hydrochloride
TMIH-0314
Lurasidone-D8 hydrochloride is a deuterated compound of Lurasidone hydrochloride. Lurasidone hydrochloride has a CAS number of 367514-88-3. Lurasidone hydrochloride (T1735) is a thiazole derivative and atypical antipsychotic agent that functions as a dopamine D2 receptor antagonist; serotonin 5-HT2 receptor antagonist, serotonin 5-HT7 receptor antagonist, an antagonist of the adrenergic α2A and α2C receptors, as well as a partial serotonin 5-HT1A receptor agonist. It is used in the treatment of schizophrenia and bipolar disorder.
  • $445
7-10 days
Size
QTY
Lurasidone (Standard)
TMSM-3492367514-87-2
Lurasidone (Standard) is a reference standard for research and analysis in studies involving Lurasidone. Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6.75 nM).
  • $153
7-10 days
Size
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Lurasidone-[D4] Hydrochloride (Standard)
TMSM-6522
Lurasidone-[D4] Hydrochloride (Standard) is a reference standard of Lurasidone-[D4] Hydrochloride intended for quantitative analysis, quality control, and related biochemical research applications.
  • $612
4-6 weeks
Size
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Lurasidone-[D8] Hydrochloride (Standard)
TMSM-6523
Lurasidone-[D8] Hydrochloride (Standard) is a reference standard of Lurasidone-[D8] Hydrochloride intended for quantitative analysis, quality control, and related biochemical research applications.
  • $563
7-10 days
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QTY