Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • CDK
    (2)
Filter
Search Result
Results for "

lerociclib

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    2
    TargetMol | Inhibitors_Agonists
lerociclib
G1T-38, G1T38, G1T 38
T113451628256-23-4
Lerociclib (G1T38) is a selective and highly potent CDK4 6 inhibitor with anticancer and antitumor activity, inhibits CDK4 CyclinD1 and CDK6 CyclinD3, and inhibits tumor growth in an animal model of endocrine-resistant breast cancer. Due to the poor solubility, for animal studies, the salt form T11345L is recommended.
  • Inquiry Price
8-10 weeks
Size
QTY
Lerociclib dihydrochloride
G1T38 dihydrochloride
T11345L2097938-59-3
Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective CDK4 CDK6 inhibitor, with IC50 values of 2 nM for CDK6 CyclinD3 and 1 nM for CDK4 CyclinD1.
  • Inquiry Price
Size
QTY
TargetMol | Inhibitor Sale