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By Target- BCRP
- ABC Transporter(1)
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Results for "
ko143
" in TargetMol Product Catalog- Inhibitors & Agonists2
CitedABCG2-IN-1
T795132559759-40-7
ABCG2-IN-1 (compound K2), an analog of Ko143, is an orally active inhibitor of ABCG2 with an IC50 of 0.13 μM, demonstrating favorable oral pharmacokinetics in mice and showing promise for further research [1].
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