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By Target- BCRP
- ABC Transporter(1)
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Results for "
ko-143
" in TargetMol Product Catalog- Inhibitors & Agonists2
CitedMZ82
T200975
MZ82, a derivative of Ko 143, is a potent inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2 BCRP), with an IC50 of approximately 23 nM. Compared to Ko 143, MZ82 exhibits significantly enhanced metabolic stability in liver microsomes and shows marked improvement in mice, along with the ability to penetrate the brain.
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