Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • Cannabinoid Receptor
    (1)
  • Others
    (2)
Filter
Search Result
Results for "

hcb1r

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    3
    TargetMol | Inhibitors_Agonists
Taranabant
MK-0364
T13080L701977-09-5
Taranabant (MK-0364) is a selective and potent cannabinoid 1 (CB1) receptor inverse agonist used in the study of obesity and nicotine dependence.
  • Inquiry Price
10-14 weeks
Size
QTY
GAT564
T61180
GAT564 (Compound 15d) is a highly effective allosteric modulator of the cannabinoid 1 receptor (CB1R), with EC50 values of 87 nM for cAMP and 320 nM for β-arrestin2. It significantly enhances the binding of orthosteric ligands to hCB1R and exhibits remarkable efficacy as a topical agent, significantly reducing intraocular pressure (IOP) in an ocular normotensive murine model of glaucoma [1].
  • Inquiry Price
10-14 weeks
Size
QTY
cbr agonist-2
T62584
CBR Agonist-2 is a CB1 agonist (CB1R; CB1 ligand) with an EC50 of 960 nM and Ki of 970 nM, making it a promising tool for studying diseases related to the endogenous cannabinoid system involving hCB1R.
  • Inquiry Price
10-14 weeks
Size
QTY