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(3)
By Target- Histamine Receptor
- Apoptosis(1)
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Results for "
h3lr
" in TargetMol Product Catalog.- Inhibitors & Agonists3
- Clobenpropit dihydrobromideT8439145231-35-2Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
- $38
SizeQTY - ProxyfanProxifanT23190177708-09-7Proxyfan (Proxifan) is a high-affinity protean antagonist/agonist of histamine H3 receptors with a full spectrum of pharmacological activity ranging from full agonist to full inverse agonist(antagonist), depending on the competition between constitutively active and resting H3 receptors within a given tissue or brain region.Proxyfan acts as a neutral antagonist in the feeding-associated ventral medial nucleus of the hypothalamus, and as a agonist in the basolateral amygdala of the rat (BLA).
- $293
SizeQTY - Proxyfan OxalateT883571620017-81-3Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.
- $1,730
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