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gs 626510

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  • Inhibitors & Agonists
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    TargetMol | Inhibitors_Agonists
GS-626510
T154191637770-13-8
GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2 3 4; IC50: 83 nM and 78 nM for BD1 and BD2).
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6-8 weeks
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