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  • Histone Methyltransferase
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epz 019997

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    3
    TargetMol | Inhibitors_Agonists
gsk3368715 3hcl
GSK3368715(EPZ019997), EPZ019997 3HCl
T223422227587-26-8
GSK3368715, a potent inhibitor of type I protein arginine methyltransferases (PRMT), could inhibit PRMT1, 3, 4, 6 and 8 with Kiapp vaules ranging from 1.5 to 81 nM.
  • Inquiry Price
10-14 weeks
Size
QTY
GSK3368715
EPZ019997
T115001629013-22-4In house
GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s: 3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)). It has strong anti-cancer activity.
  • Inquiry Price
3-6 months
Size
QTY
GSK3368715 dihydrochloride
EPZ019997 dihydrochloride, GSK3368715 2HCl, EPZ019997 2HCl
T11500L1628925-77-8
GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is an orally active and potent inhibitor of type I protein arginine methyltransferases (PRMTs), including PRMT1, PRMT3, PRMT4, PRMT6, and PRMT8. It exhibits anticancer and antitumor activity and can be used to study advanced solid tumors.
  • Inquiry Price
10-14 weeks
Size
QTY