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am-251

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    2
    TargetMol | Inhibitors_Agonists
AM251
T1915183232-66-8
AM251 is a effective CB1 receptor antagonist (IC50 Ki: 8 7.49 nM) that displays 306-fold selectivity over CB2 receptors; also effective GPR55 agonist (EC50: 39 nM).
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Tocrifluor T1117
T234641186195-59-4
Fluorescent form of AM 251, CB1 receptor antagonist
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