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(1)
By Target- GRK
- PKC(1)
- ROCK(1)
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By Target By ResearchField- Cardiovascular System(1)
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Results for "
T14989
" in TargetMol Product Catalog.- Inhibitors & Agonists1
- CMPD101T14989865608-11-3CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM). Which can be used for the study of heart failure. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCα with IC50s of 3.1 μM , 2.3 μM, 1.4 μM and 8.1 μM, respectively.
- $40
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Other Forms of Products
- CMPD101 hydrochloride
T893641941168-71-3CMPD101 hydrochloride is a membrane-permeable small molecule inhibitor of GRK2 and GRK3, exhibiting IC50 values of 18 nM and 5.4 nM, respectively. This compound also inhibits Rho-associated kinase 2 (ROCK-2) and PKCα, with IC50 values of 1.4 μM and 8.1 μM, respectively.- Inquiry Price
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