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Compounds

Cat No. Product Name
TN6512 Tectol Transferase , Parasite
Tectol 是从Lippia sidoides 中分离的,对人白血病细胞株 HL60 和 CEM 具有显著的抑制作用。它是法尼基转移酶抑制剂,在人和布氏锥虫的IC50分别为 2.09 和 1.73 μM。它具有抗疟原虫活性,是一种中等活性...
T12783 RWJ 50271 Integrin
RWJ 50271 是具有口服活性的选择性LFA-1/ICAM-1相互作用抑制剂,抑制 LFA-1/ICAM-1 介导的细胞粘附,在细胞HL60中的IC50值为 5.0 μM。
T5S1000 Sophoraflavanone G 槐黄烷酮 G,Vexibinol,Kushenol F Apoptosis
Sophoraflavanone G 是从苦参中提取到的一种天然产物,通过抑制 MAPK 相关通路诱导 MDA-MB-231 和 HL-60 细胞凋亡,具有抗肿瘤和抗炎特性。
T2S0357 6-Hydroxycoumarin 6-hydroxychromen-2-one,6-羟基香豆素 Others , Carbonic Anhydrase
6-Hydroxycoumarin 是一种香豆素。其中香豆素具有抗炎,支气管扩张,解热,血管扩张,抗氧化,抗菌,抗真菌,抑菌和抗肿瘤作用。
T14946 Ch55 Ch-55,CH 55,3,5-Di-tert-butylchalcone Retinoid Receptor
Ch55是HL60细胞分化的有效诱导剂(EC50 = 200 nM),与RAR-α和RAR-β受体显示出高亲和力。Ch55可用于有关癌症的研究。
T3774 Gracillin 纤细薯蓣皂苷,山药 cell cycle arrest
Gracillin 是一种甾体皂苷,从植物的根里提取得到,有抗肿瘤作用。
T21165 Pellitorine 墙草碱,Pellitorin,AI3-19560 TRP/TRPV Channel
Pellitorine 是提取自 Piper nigrum 的根的一种化合物。它对 HL60 和 MCT-7 细胞系表现出显著的细胞毒活性。它可用于癌症疾病的研究。
T6588 Mitoxantrone mitozantrone,米托蒽醌 Topoisomerase , PKC
Mitoxantrone 是一种拓扑异构酶 II 的抑制剂,也可抑制蛋白激酶C (PKC),IC50值为8.5 μM。
T60002 Ethyl 2-amino-4-methyl-5-[(3-nitrophenyl)carbamoyl]thiophene-3-carboxylate DC-S239 Histone Methyltransferase
Ethyl 2-amino-4-methyl-5-[(3-nitrophenyl)carbamoyl]thiophene-3-carboxylate 是一种选择性的组蛋白甲基转移酶 SETD7 抑制剂 (IC50 = 4.59 μM),具有...
TN2755 2-Desoxy-4-epi-pulchellin Anti-infection
2-Desoxy-4-epi-pulchellin 是分离自 Polygonum hydropiper 的二氯甲烷可溶部分的一种化合物。
T0974 Novobiocin Sodium 新生霉素钠,Albamycin,Cathomycin,Albamycinsodium Autophagy , ABC , Antibiotic , Potassium Channel , DNA gyrase , Topoisomerase , Antibacterial
Novobiocin sodium 是源自 Streptomyces niveus 的抗生素。 它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。
T0158 Mitoxantrone dihydrochloride 米托蒽醌二盐酸盐,盐酸米托蒽醌,Mitoxantrone 2HCl,NSC-301739,mitozantrone dihydrochloride,Mitoxantrone hydrochloride Topoisomerase , PKC
Mitoxantrone hydrochloride 是一种拓扑异构酶 II 的抑制剂;也可抑制蛋白激酶C (PKC),IC50值为8.5 μM。
T2924 Phloretin 根皮素,RJC 02792,NSC 407292,Dihydronaringenin transporter , SGLT , Endogenous Metabolite
Phloretin 是从苹果树叶中提取的一种查耳酮,具有抗炎、抗氧化和抗癌活性。它是真核尿素转运蛋白抑制剂,可阻断 VacA 介导的尿素和离子转运,有潜力用于类风湿性关节炎和过敏性气道炎症的相关研究。
T73588 8-(4-iodophenyl)-1,3,5,7-tetramethyl BODIPY
8-(4-iodophenyl)-1,3,5,7-tetramethyl BODIPY 是一种新型的 BODIPY 荧光染料,可用于治疗细胞毒性研究。
T6018 Zosuquidar trihydrochloride 唑喹达三盐酸盐,Zosuquidar 3HCl,RS 33295-198 trihydrochloride,LY-335979 trihydrochloride,Zosuquidar (LY335979) 3HCl,RS 33295-198 (D06387) 3HCl P-gp
Zosuquidar trihydrochloride 是一种P-糖蛋白抑制剂,Ki 值为 59 nM。
TN5579 Trigoxyphin A
Trigoxyphin A exhibits strong cytotoxic activity against HL60 (IC(50): 0.27 microM) and A549 (IC(50): 7.5 microM) tumor ...
T36963 CAY10503
CAY10503 is a proapoptotic, antiproliferative compound that is able to arrest cell cycle progression in the G0-G1 phase....
TN2835 28-Deoxonimbolide Caspase
28-Deoxonimbolide exhibits potent cytotoxic activity against HL60 leukemia cells.
T4057 Hoechst 33258 trihydrochloride HOE 33258,Bisbenzimide,Hoechst 33258,Pibenzimol,H 33258 trihydrochloride,bisBenzimide H 33258 trihydrochloride Parasite
Hoechst 33258 是一种能够用于 DNA 染色的荧光染料。
T10973 DC41SMe Others
DC41SMe is a DC1 derivative that is cytotoxic to Ramos, Namalwa and HL60 / s with IC50s ranging from 18-25 pM. DC1 is a ...
Tectol
TN6512
synonym:
Target:
RWJ 50271
T12783
synonym:
Target:
Sophoraflavanone G
T5S1000
synonym: 槐黄烷酮 G,Vexibinol,Kushenol F
Target:
6-Hydroxycoumarin
T2S0357
synonym: 6-hydroxychromen-2-one,6-羟基香豆素
Target:
Ch55
T14946
synonym: Ch-55,CH 55,3,5-Di-tert-butylchalcone
Target:
Gracillin
T3774
synonym: 纤细薯蓣皂苷,山药
Target:
Pellitorine
T21165
synonym: 墙草碱,Pellitorin,AI3-19560
Target:
Mitoxantrone
T6588
synonym: mitozantrone,米托蒽醌
Target:
Ethyl 2-amino-4-methyl-5-[(3-nitrophenyl)carbamoyl]thiophene-3-carboxylate
T60002
synonym: DC-S239
Target:
2-Desoxy-4-epi-pulchellin
TN2755
synonym:
Target:
Novobiocin Sodium
T0974
synonym: 新生霉素钠,Albamycin,Cathomycin,Albamycinsodium
Target:
Mitoxantrone dihydrochloride
T0158
synonym: 米托蒽醌二盐酸盐,盐酸米托蒽醌,Mitoxantrone 2HCl,NSC-301739,mitozantrone dihydrochloride,Mitoxantrone hydrochloride
Target:
Phloretin
T2924
synonym: 根皮素,RJC 02792,NSC 407292,Dihydronaringenin
Target:
8-(4-iodophenyl)-1,3,5,7-tetramethyl BODIPY
T73588
synonym:
Target:
Zosuquidar trihydrochloride
T6018
synonym: 唑喹达三盐酸盐,Zosuquidar 3HCl,RS 33295-198 trihydrochloride,LY-335979 trihydrochloride,Zosuquidar (LY335979) 3HCl,RS 33295-198 (D06387) 3HCl
Target:
Trigoxyphin A
TN5579
synonym:
Target:
CAY10503
T36963
synonym:
Target:
28-Deoxonimbolide
TN2835
synonym:
Target:
Hoechst 33258 trihydrochloride
T4057
synonym: HOE 33258,Bisbenzimide,Hoechst 33258,Pibenzimol,H 33258 trihydrochloride,bisBenzimide H 33258 trihydrochloride
Target:
DC41SMe
T10973
synonym:
Target:
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