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Compounds

Cat No. Product Name
T12580 PTUPB Epoxide Hydrolase , COX
PTUPB 是强效的sEH(IC50:0.9 μM)和COX-2(IC50:1.26 μM)的双向抑制剂。
T27061 CP-24879 hydrochloride CP-24879 HCl Others
CP-24879 hydrochloride 是选择性的 delta5D/delta6D 联合抑制剂。它能显著降低肝细胞内脂质积聚和炎症损伤。它在脂肪-1 和 ω-3 处理的肝细胞中表现出优越的抗脂肪变性和抗炎作用,可用于非酒精性脂肪性肝炎...
T14301 Apararenone MT-3995 Glucocorticoid Receptor
Apararenone 是一种新型的、非甾体类盐皮质激素受体 (mineralocorticoid receptor) 拮抗剂,正在开发用于糖尿病性肾病和非酒精性脂肪性肝炎的研究。
T31964 Glycolithocholic acid 甘氨石胆酸,Lithocholylglycine,Lithocholic acid glycine conjugate Others
Glycolithocholic acid 属于内源性代谢产物,是甘氨酸结合的次级胆汁酸。它可用于诊断非酒精性脂肪性肝炎,溃疡性结肠炎和原发性硬化性胆管炎。
T65815 H-Asp(OtBu)-OtBu HCl Amino Acids and Derivatives
H-Asp(OtBu)-OtBu HCl 是一种天冬氨酸衍生物,可能用于研究神经功能的比较和非酒精类肝炎类代谢性疾病。
T9186 Ervogastat PF-06865571 Transferase
Ervogastat 是一种有效且耐受性良好的二酰基甘油酰基转移酶 2 抑制剂。 Ervogastat 可降低非酒精性脂肪性肝炎 (NASH) 中的脂肪变性和肝脏甘油三酯水平。
T64334 Glycolithocholic acid, sodium salt Others
Glycolithocholic acid, sodium salt 是 Glycolithocholic acid 的钠盐。Glycolithocholic acid 是一种甘氨酸结合的次级胆汁酸。Glycolithocholic aci...
T67974 Berberine ursodeoxycholate HTD1801,BUDCA
Berberine ursodeoxycholate 是一种口服有效的降血脂剂 ,是 Berberine 和 Ursodeoxycholic acid 的一种离子盐。Berberine ursodeoxycholate 具有广泛的代谢活性...
T2601 Vidofludimus 4sc-101,SC12267 Dehydrogenase , DNA/RNA Synthesis , Interleukin
Vidofludimus 是一种新型的二氢乳清酸脱氢酶 (DHODH) 小分子抑制剂,可在不影响淋巴细胞增殖的条件下抑制IL-17的分泌。
T17236 Volixibat SHP626,LUM002 Others
Volixibat is a highly selective and competitive apical sodium-dependent bile acid transporter inhibitor. Volixibat has t...
T11448 GOAT-IN-1 Others
GOAT-IN-1 is an inhibitor of ghrelin O-acyltransferase (GOAT), which could be useful for the prophylaxis or treatment of...
T35801 ML-262
ML-262 is an inhibitor of hepatic lipid droplet formation (IC50 = 6.4 nM in murine AML-12 cells), which is associated wi...
T62029 ML261
ML261 是肝脂滴形成的抑制剂,IC50值为 69.7 nM。ML261 在非酒精性脂肪性肝病 (NAFLD) 和炎症中具有研究价值。
T35443 1-Palmitoyl-2-Stearoyl-3-Oleoyl-rac-glycerol
1-Palmitoyl-2-stearoyl-3-oleoyl-rac-glycerol is a triacylglycerol that contains palmitic , stearic , and oleic acid at t...
T77175 Efruxifermin
Efruxifermin 是一种Fc-FGF21融合蛋白(人IgG1Fc 结构域连接到修饰的人 FGF21)。与天然人FGF21相比,Efruxifermin 的半衰期延长,受体亲和力增强。Efruxifermin 可用于非酒精性脂肪性肝炎...
T74421 Pemvidutide
Pemvidutide 是一种GLP-1R/GCGR 双重激动剂,可导致体重、肝脏脂肪和血清脂质的显著降低。Pemvidutide 可用于非酒精性脂肪性肝炎 (NASH) 和肥胖症的研究。
T21978 P-nitro-Pifithrin-α
p-nitro-Pifithrin-α is a cell-permeable analog of pifithrin-α, a potent p53 inhibitor. It suppresses p53-mediated TGF-β1...
T35636 SHS4121705
SHS4121705 is an orally bioavailable mitochondrial uncoupler.1It increases oxygen consumption rate in L6 rat myoblast ce...
T63777 QH536
QH536 是 HMGCR 的有效降解剂 (EC50: 0.22 μM)。QH536 表现出抗炎效果,并没有诱导胆固醇在细胞内积聚的副作用。QH536 能够用于研究心血管疾病和非酒精性脂肪性肝炎。
T72889 FXR agonist 4
FXR agonist4 是法尼酯 X 受体 (FXR) 激动剂,EC50值为 1.05 μM。FXR agonist4 有效改善 DIO 小鼠高脂血症、肝脏脂肪变性、胰岛素抵抗和肝脏炎症。FXR agonist4 可用于非酒精性脂肪性肝...
PTUPB
T12580
synonym:
Target:
CP-24879 hydrochloride
T27061
synonym: CP-24879 HCl
Target:
Apararenone
T14301
synonym: MT-3995
Target:
Glycolithocholic acid
T31964
synonym: 甘氨石胆酸,Lithocholylglycine,Lithocholic acid glycine conjugate
Target:
H-Asp(OtBu)-OtBu HCl
T65815
synonym:
Target:
Ervogastat
T9186
synonym: PF-06865571
Target:
Glycolithocholic acid, sodium salt
T64334
synonym:
Target:
Berberine ursodeoxycholate
T67974
synonym: HTD1801,BUDCA
Target:
Vidofludimus
T2601
synonym: 4sc-101,SC12267
Target:
Volixibat
T17236
synonym: SHP626,LUM002
Target:
GOAT-IN-1
T11448
synonym:
Target:
ML-262
T35801
synonym:
Target:
ML261
T62029
synonym:
Target:
1-Palmitoyl-2-Stearoyl-3-Oleoyl-rac-glycerol
T35443
synonym:
Target:
Efruxifermin
T77175
synonym:
Target:
Pemvidutide
T74421
synonym:
Target:
p-nitro-Pifithrin-α
T21978
synonym:
Target:
SHS4121705
T35636
synonym:
Target:
QH536
T63777
synonym:
Target:
FXR agonist 4
T72889
synonym:
Target:
1 2