Home Tools
Log in
Cart

Search Result

Search Results for "monoamine transporter"

Targets

Compounds

Cat No. Product Name
T7147 Valbenazine NBI-98854 Monoamine Transporter
Valbenazine 是一种高度选择性的囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,Ki 为 110-190 nM,用于治疗迟发性运动障碍。
T22714 Decynium 22 Others
Decynium 22 是有机阳离子转运蛋白和单胺转运蛋白的抑制剂,具有抗抑郁作用。
T7563 NBI-98782 (+)-α-二氢丁苯那嗪,[2R-(2a,3b,11bb)]-1,3,4,6,7,11b-六氢-9,10-二甲氧基-3-异丁基-2H-苯并[a]喹嗪-2-醇,(+)-α-DHTBZ,(+)-α-Dihydrotetrabenazine,(+)-DTBZ Monoamine Transporter
NBI-98782 是一种囊泡单胺转运蛋白 (VMAT2) 抑制剂,Ki 为0.97nM。
T3534 Tetrabenazine Racemate 丁苯那嗪外消旋体,丁苯那嗪,TETRABENAZINE,Nitoman,Ro 1-9569 Racemate,Rubigen Monoamine Transporter
Tetrabenazine Racemate 是一种选择性和可逆的囊泡单胺转运蛋白 2 (VMAT-2) 抑制剂。它阻断神经递质吸收到肾上腺素能储存囊泡中,并已被用作囊泡运输系统的高亲和力标记。
T0791 Reserpine 利血平,Serpivite,Serpalan,Serpasil Monoamine Transporter , Potassium Channel , Autophagy , Others , MRP
Reserpine 是一种从催吐萝芙木的根中发现的生物碱。它抑制去甲肾上腺素吸收到储存囊泡中,导致中枢和外周轴突末端的儿茶酚胺和血清素耗尽。它可作为抗高血压药和抗精神病药以及研究工具。
T23070 Nisoxetine hydrochloride Monoamine Transporter , Sodium Channel , Norepinephrine
Nisoxetine hydrochloride 是一种去甲肾上腺素转运蛋白 (NET) 抑制剂,Kd 值为 0.76 nM。它是抗抑郁药和局部麻药,可以阻断电压门控性钠通道。
T1993 J-147 J147 Monoamine Oxidase , Epigenetic Reader Domain , Dopamine Receptor
J147 是一种高效的、具有口服活性的、可透过血脑屏障神经保护剂,可增强认知能力。它抑制单胺氧化酶 B 和多巴胺转运体,EC50分别为 1.88 μM 和 0.649 μM。它有研究阿尔茨海默氏症的潜力。
T0719 Tetrabenazine Xenazine,Ro 1-9569,丁苯那嗪 Dopamine Receptor , Others , Monoamine Transporter
Tetrabenazine 是 VMAT 抑制剂,用作抗精神病药和治疗各种运动障碍。
T13134 (+)-Tetrabenazine (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ Monoamine Transporter
(+)-Tetrabenazine 是一种可逆的囊泡单胺转运蛋白2 (VMAT-2)抑制剂,对 VMAT2转运的抑制作用是VMAT1的10倍。
T7651 Rose Bengal sodium Rose Bengal,酸性红 94 Monoamine Transporter , Influenza Virus
Rose Bengal 是一种合成的荧光素衍生物,主要成分是 4,5,6,7-tetrachloro-2,4,5,7-tetraiodo 荧光素,可以检测眼表干燥或受损的细胞,用作眼科诊断剂,具有抗病毒活性。它是一种 VGlut 和囊泡单胺...
T13133 Tetrabenazine Metabolite (-)-β-HTBZ,(-)-β-Dihydrotetrabenazine Monoamine Transporter
Tetrabenazine Metabolite 是一种囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,是 Tetrabenazine 的一种活性代谢物。Tetrabenazine Metabolite 对 VMAT2 具有高亲和力,其Ki ...
T3933 Jatrorrhizine 药根碱,neprotin,Yatrorizine AChE , Antibacterial , MAO , 5-HT Receptor
Jatrorrhizine 是一种从黄连中分离得到的生物碱,具有抗菌、抗氧化、抗疟原虫和神经保护活性。它通过抑制 uptake-2 transporter 的活性减少血清素和去甲肾上腺素的摄取。它是一种有口服活性的乙酰胆碱酯酶制剂。
T25750 Lobelane Hydrochloride
Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor.
T68488 Indatraline
Indatraline is a nonselective monoamine transporter inhibitor.
T31790 FFN200 dihydrochloride FFN-200,FFN200,FFN 200,FFN200 HCl
FFN200 is a vesicular monoamine transporter 2 (VMAT2) substrate that selectively traces monoamine exocytosis in both neu...
T31791 FFN246 HCl FFN 246,FFN-246,FFN246 hydrochloride,FFN246
FFN246 is a fluorescent substrate for both the serotonin transporter and the vesicular monoamine transporter 2 (VMAT2).
T70322 Valbenazine dihydrochloride
Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.
T24941 VMAT2-IN-I HCl VMAT2 IN I Hydrochloride,VMAT2INI Hydrochloride,VMAT2-IN-I Hydrochloride
VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A...
T23629 Adam I-123 Adam I 123,Adam I123
Adam I-123 is a radiopharmaceutical containing the serotonin transporter (SERT) ligand, with SERT-binding and radioisoto...
T36949 Niaprazine Adrenergic Receptor , Histamine Receptor , 5-HT Receptor
Niaprazine 是有效的组胺 H1 受体拮抗剂,具有抗组胺和抗血清素活性。Niaprazine 在睡眠障碍方面有研究的价值。
Valbenazine
T7147
synonym: NBI-98854
Target:
Decynium 22
T22714
synonym:
Target:
NBI-98782
T7563
synonym: (+)-α-二氢丁苯那嗪,[2R-(2a,3b,11bb)]-1,3,4,6,7,11b-六氢-9,10-二甲氧基-3-异丁基-2H-苯并[a]喹嗪-2-醇,(+)-α-DHTBZ,(+)-α-Dihydrotetrabenazine,(+)-DTBZ
Target:
Tetrabenazine Racemate
T3534
synonym: 丁苯那嗪外消旋体,丁苯那嗪,TETRABENAZINE,Nitoman,Ro 1-9569 Racemate,Rubigen
Target:
Reserpine
T0791
synonym: 利血平,Serpivite,Serpalan,Serpasil
Target:
Nisoxetine hydrochloride
T23070
synonym:
Target:
J-147
T1993
synonym: J147
Target:
Tetrabenazine
T0719
synonym: Xenazine,Ro 1-9569,丁苯那嗪
Target:
(+)-Tetrabenazine
T13134
synonym: (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ
Target:
Rose Bengal sodium
T7651
synonym: Rose Bengal,酸性红 94
Target:
Tetrabenazine Metabolite
T13133
synonym: (-)-β-HTBZ,(-)-β-Dihydrotetrabenazine
Target:
Jatrorrhizine
T3933
synonym: 药根碱,neprotin,Yatrorizine
Target:
Lobelane Hydrochloride
T25750
synonym:
Target:
Indatraline
T68488
synonym:
Target:
FFN200 dihydrochloride
T31790
synonym: FFN-200,FFN200,FFN 200,FFN200 HCl
Target:
FFN246 HCl
T31791
synonym: FFN 246,FFN-246,FFN246 hydrochloride,FFN246
Target:
Valbenazine dihydrochloride
T70322
synonym:
Target:
VMAT2-IN-I HCl
T24941
synonym: VMAT2 IN I Hydrochloride,VMAT2INI Hydrochloride,VMAT2-IN-I Hydrochloride
Target:
Adam I-123
T23629
synonym: Adam I 123,Adam I123
Target:
Niaprazine
T36949
synonym:
Target:
1 2