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Search Result

Search Results for "leukotriene receptor"

Targets

Leukotriene Receptor

Compounds

Cat No. Product Name
T6736 Zafirlukast Vanticon,ICI 204219,Accolate,扎鲁司特 Leukotriene Receptor
Zafirlukast 是一种可口服的白三烯 D4受体拮抗剂，具有平喘、抗炎和抗菌作用。
T22946 LY255283 LY 255283 Leukotriene Receptor
LY 255283 是白三烯 B4 (LTB4) 受体的特异性拮抗剂，抑制人外周血多形核白细胞和由钙离子载体 A23187 激活的单核细胞中 LTB(4) 的产生。
T0694 Pranlukast 普鲁司特,普仑司特,ONO-1078 IL Receptor , Leukotriene Receptor , Others , TNF , NF-κB , LTR
Pranlukast 是一种半胱氨酰白三烯受体 1 拮抗剂，可拮抗或减少支气管痉挛，用于哮喘研究。
T1677 Montelukast 孟鲁司特,Singular LTR , Leukotriene Receptor , Lipoxygenase
Montelukast 是可口服的半胱氨酸白三烯受体1 选择性拮抗剂，可用于研究预防哮喘和肝损伤。它还可减少心脏损伤，在肠缺血-再灌注损伤中也具有抗氧化作用。
T1677L Montelukast sodium MK0476,孟鲁司特钠 Leukotriene Receptor , LTR
Montelukast sodium 是可口服的半胱氨酸白三烯受体1 选择性拮抗剂，可用于研究预防哮喘和肝损伤。它还可减少心脏损伤，在肠缺血-再灌注损伤中也具有抗氧化作用。
T22358 Etalocib LY293111,VML295 Apoptosis , Leukotriene Receptor , LTR
Etalocib 是一种具有口服活性的白三烯(LTB4)受体的拮抗剂，抑制 [3H]LTB4结合的 Ki 值为 25 nM。它还可诱导凋亡。它抑制 LTB4诱导的钙动员，lC50值为 20 nM。
T16280 Nedocromil FPL 59002,尼多克罗 Leukotriene Receptor , Prostaglandin Receptor , Histamine Receptor
Nedocromil 对多种介质的作用或形成有抑制作用，包括组胺，前列腺素 D2和白三烯 C4。
T26519 Ablukast 阿鲁司特,Ro 23-3544 Leukotriene Receptor
Ablukast 是白三烯受体的选择性拮抗剂，也是LTD4受体拮抗剂。可改善 LTC4 和抗原诱导的支气管狭窄。
T7786 Tryptanthrin DNA gyrase
Tryptanthrin 是一种口服具有活性的细胞内Leukotriene (LT) biosynthesis 抑制剂。 它能够降低大鼠胸膜炎模型中的 LTB4 水平，并抑制人全血中Leukotriene 的形成 (IC50= 10 µM)...
T6893 MK-886 MK886,L 663536 Apoptosis , Leukotriene Receptor , COX , PPAR , FLAP
MK-886是一种细胞可渗透的，具有口服活性的 FLAP (IC50为 30 nM) 和白三烯生物合成 (完整白细胞和人全血中的IC50分别为 3 nM 和 1.1μM) 的抑制剂。它也是一种非竞争性PPARα拮抗剂，可以诱导细胞凋亡。
T5714 5-O-Demethylnobiletin 去甲基川陈皮素,5-DEMETHYLNOBILETIN Lipoxygenase , Leukotriene Receptor
5-O-Demethylnobiletin 是从黄芪中分离出的多甲氧基黄酮，具有抗炎活性，可通过直接抑制 5-LOX 发挥作用，IC50为 0.1 μM。
T20615 Olsalazine Salicylic acid,Dipentium,奥沙拉嗪 Others
Olsalazine 是一种抗炎药，用于治疗炎症性肠病。它也是一种新型的 DNA 去甲基化剂。
T21504 γ-Linolenic Acid methyl ester γ-亚麻酸甲酯,Methyl gamma-linolenate LTR
γ-Linolenic Acid methyl ester 是一种弱白三烯 B4 (LTB4) 受体拮抗剂。
T68119 Ontazolast BIRM-270 LTR
Ontazolast 是一种小分子白三烯B4受体（LTB4R）拮抗剂，可用于治疗免疫系统疾病和呼吸系统疾病。Ontazolast 是治疗哮喘的候选化合物。
T28974 Ticolubant Calcium Channel , LTR
Ticolubant 是一种具有口服活性的白三烯 B4 拮抗剂，对人类中性粒细胞 LTB4 受体具有很高的亲和力（Ki = 0.78 nM），能阻断 LTB4 诱导的 Ca2+ 迁移，IC50 为 6.6±1.5 nM，并在小鼠皮肤炎症模型...
T68108L Moxilubant HCl Moxilubant hcl(146978-48-5 Free base) LTR
Moxilubant HCl 是一种小分子白三烯 B4 受体 1（LTB4R）拮抗剂，可用于治疗免疫系统疾病、皮肤和肌肉骨骼疾病，可用于研究银屑病和类风湿关节炎。
TN1182 11-​Keto-​beta-​boswellic acid 11-酮基-BETA-乳香酸,11-Keto-beta-boswellic acid NF-κB , Lipoxygenase , Leukotriene Receptor
11-Keto-beta-boswellic acid 是来自乳香的一种五环三萜酸，具有抗炎活性和剂量依赖性心脏保护作用，主要是由于抑制5-脂氧合酶、白三烯、NF-κB 的激活和肿瘤坏死因子 α 的产生。
T3148 MK-571 sodium Verlukast sodium,MK571,L-660711 sodium salt,MK-571 sodium salt,L-660711 (sodium salt),L-660711,Propanoic acid Leukotriene Receptor , LTR
MK-571 sodium 是一种可口服的选择性白三烯 D4受体拮抗剂，在豚鼠和人肺膜的 Ki 分别为0.22 和 2.1 nM。
T4973 Paraxanthine 1,7-DIMETHYLXANTHINE,1,7-二甲基黄嘌呤 Endogenous Metabolite
1,7-dimethylxanthine 是一种 caffeine 的代谢物，能够刺激Ryanodine 受体通道来抑制多巴胺能细胞的死亡。
T4657 WHI-P97 4-(3',5'-二溴-4-羟基苯基)氨基-6,7-二甲氧基喹唑啉 JAK
WHI-P97 是一种选择性 JAK-3抑制剂，可用于预防过敏性哮喘的研究。
Zafirlukast
T6736
synonym: Vanticon,ICI 204219,Accolate,扎鲁司特
Target:
LY255283
T22946
synonym: LY 255283
Target:
Pranlukast
T0694
synonym: 普鲁司特,普仑司特,ONO-1078
Target:
Montelukast
T1677
synonym: 孟鲁司特,Singular
Target:
Montelukast sodium
T1677L
synonym: MK0476,孟鲁司特钠
Target:
Etalocib
T22358
synonym: LY293111,VML295
Target:
Nedocromil
T16280
synonym: FPL 59002,尼多克罗
Target:
Ablukast
T26519
synonym: 阿鲁司特,Ro 23-3544
Target:
Tryptanthrin
T7786
synonym:
Target:
MK-886
T6893
synonym: MK886,L 663536
Target:
5-O-Demethylnobiletin
T5714
synonym: 去甲基川陈皮素,5-DEMETHYLNOBILETIN
Target:
Olsalazine
T20615
synonym: Salicylic acid,Dipentium,奥沙拉嗪
Target:
γ-Linolenic Acid methyl ester
T21504
synonym: γ-亚麻酸甲酯,Methyl gamma-linolenate
Target:
Ontazolast
T68119
synonym: BIRM-270
Target:
Ticolubant
T28974
synonym:
Target:
Moxilubant HCl
T68108L
synonym: Moxilubant hcl(146978-48-5 Free base)
Target:
11-​Keto-​beta-​boswellic acid
TN1182
synonym: 11-酮基-BETA-乳香酸,11-Keto-beta-boswellic acid
Target:
MK-571 sodium
T3148
synonym: Verlukast sodium,MK571,L-660711 sodium salt,MK-571 sodium salt,L-660711 (sodium salt),L-660711,Propanoic acid
Target:
Paraxanthine
T4973
synonym: 1,7-DIMETHYLXANTHINE,1,7-二甲基黄嘌呤
Target:
WHI-P97
T4657
synonym: 4-(3',5'-二溴-4-羟基苯基)氨基-6,7-二甲氧基喹唑啉
Target:
1 2 3 4
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