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Search Results for "dna damage/dna repair"

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Compounds

Cat No. Product Name
T5399 GeA-69 PARP
GeA-69 是一种选择性变构 PARP14 大结构域 2 (MD2) 抑制剂,Kd 值为 2.1 µM。
T10406 Tuvusertib ATR inhibitor 1,M1774 Others , Chk , Apoptosis , ATM/ATR
Tuvusertib 是一种可口服的共济失调毛细血管扩张和 Rad3相关(ATR)激酶抑制剂(Ki< 1 µΜ),具有选择性和潜在的抗肿瘤活性。Tuvusertib 选择性抑制 ATR 活性,阻断丝氨酸/苏氨酸蛋白激酶检查点激酶1 (CHK...
T50098 TIQ-A PARP
TIQ-A 是一种 PARP1 抑制剂,通过碱基切除修复途径参与 DNA 单链断裂修复。 PARP1 由 DNA 损伤触发,其过度激活已被认为是许多病理状况的致病因素,包括缺血和再灌注损伤、哮喘相关炎症和动脉粥样硬化形成。
T7318 Elimusertib BAY-1895344 ATM/ATR
Elimusertib 是一种可口服的选择性ATR 抑制剂,IC50值为 7 nM。它具有抗肿瘤活性,可研究实体瘤和淋巴瘤。
T21320 Methoxyamine HCl TRC 102,TRC102,甲氧基胺盐酸盐,Methoxyamine,TRC-102 Others
Methoxyamine HCl 与脱嘌呤/脱嘧啶 (AP) DNA 损伤位点共价结合并抑制碱基切除修复 (BER),这可能导致 DNA 链断裂和细胞凋亡增加。 Methoxyamine 是一种具有潜在佐剂活性的口服生物可利用的小分子抑制剂...
T4971 5'-DEOXYADENOSINE 5-脱氧腺嘌呤核苷,5′-dAdo Endogenous Metabolite
5'-Deoxyadenosine 是正常受试者尿液中发现的氧化核苷,氧化核苷代表了用于确定遗传物质损伤程度的优秀生物标志物。
T25838 MS0017509 MS-0017509,MS 0017509
MS0017509 is a DNA damage repair inhibitor.
T25839 MS0019266 MS 0019266,MS-0019266
MS0019266 is a DNA damage repair inhibitor.
T10018 1-Methyladenine Others
1-Methyladenine is a DNA alkylation product that undergoes damage reversal through oxidative demethylation for repair pu...
T14282 Amuvatinib hydrochloride HPK 56 hydrochloride,MP470 hydrochloride Others
Amuvatinib hydrochloride (MP470 hydrochloride) is an orally bioavailable multi-targeted tyrosine kinase inhibitor with p...
T70873 M3541
M3541 is a potent, selective, orally active ATM inhibitor with potential chemo-/radio-sensitizing and antineoplastic act...
T69931 MFH290
MFH290 is a novel cysteine (Cys)-directed covalent inhibitor of CDK12/13. MFH290 forms a covalent bond with Cys-1039 of ...
T40345 AV-153
AV-153 is a 1,4-dihydropyridine derivative with antimutagenic properties. It intercalates into DNA at single strand brea...
T36701 Phosphoramide mustard (cyclohexanamine)
Phosphoramide mustard cyclohexanamine is the major metabolite for Cyclophosphamide , with anticancer activitiy. Phosphor...
T26981 Ceralasertib formate Ceralasertib,AZD-6738,AZD6738,AZD 6738
Ceralasertib is an orally available inhibitor of ataxia telangiectasia and rad3 related (ATR) kinase. Ceralasertib selec...
T63923 ATR-IN-5
ATR-IN-5 是 ATR 的有效抑制剂。其中 ATR 是 PIKK 家族的成员,是一类参与基因组稳定性和 DNA 损伤修复的蛋白激酶。ATR-IN-5 对 ATR 激酶介导的疾病如增殖性疾病和癌症表现出研究潜力,信息来源于专利 CN11...
T75335 Ethylenediaminetetraacetic acid dipotassium dihydrate
Ethylenediaminetetraacetic acid (EDTA) dipotassium dihydrate 是抗凝血剂,可螯合重金属,解除毒性。Ethylenediaminetetraacetic acid dipotassi...
T75021 SZUH280
SZUH280 是一种有效的、选择性的 PROTACHDAC8降解剂,在 A549 细胞中的 DC50为 0.58 μM。SZUH280 诱导癌细胞凋亡 (apoptosis)。SZUH280 在癌细胞中阻碍 DNA 损伤修复,促进细胞放射...
T32189 Iproplatin Code name: JM9,JM 9,JM-9,CHIP
Iproplatin is a synthetic second-generation platinum-containing compound related to cisplatin. Iproplatin binds to and f...
T37729 IMP-1700
IMP-1700 is an inhibitor of bacterial DNA repair.1It potentiates the activity of the quinolone antibiotic ciprofloxacin ...
GeA-69
T5399
synonym:
Target:
Tuvusertib
T10406
synonym: ATR inhibitor 1,M1774
Target:
TIQ-A
T50098
synonym:
Target:
Elimusertib
T7318
synonym: BAY-1895344
Target:
Methoxyamine HCl
T21320
synonym: TRC 102,TRC102,甲氧基胺盐酸盐,Methoxyamine,TRC-102
Target:
5'-DEOXYADENOSINE
T4971
synonym: 5-脱氧腺嘌呤核苷,5′-dAdo
Target:
MS0017509
T25838
synonym: MS-0017509,MS 0017509
Target:
MS0019266
T25839
synonym: MS 0019266,MS-0019266
Target:
1-Methyladenine
T10018
synonym:
Target:
Amuvatinib hydrochloride
T14282
synonym: HPK 56 hydrochloride,MP470 hydrochloride
Target:
M3541
T70873
synonym:
Target:
MFH290
T69931
synonym:
Target:
AV-153
T40345
synonym:
Target:
Phosphoramide mustard (cyclohexanamine)
T36701
synonym:
Target:
Ceralasertib formate
T26981
synonym: Ceralasertib,AZD-6738,AZD6738,AZD 6738
Target:
ATR-IN-5
T63923
synonym:
Target:
Ethylenediaminetetraacetic acid dipotassium dihydrate
T75335
synonym:
Target:
SZUH280
T75021
synonym:
Target:
Iproplatin
T32189
synonym: Code name: JM9,JM 9,JM-9,CHIP
Target:
IMP-1700
T37729
synonym:
Target:
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