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TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.

Foscarnet sodium (Phosphonoformate) is an antiviral agent used in the treatment of cytomegalovirus retinitis. Foscarnet also shows activity against human herpesviruses and HIV.

Ascaridole (NSC-406266) acts as an anthelmintic compound that repels parasitic helminths (worms) in humans and plants and has weak antimalarial activity.

Descarbamoyl cefuroxime is also an intermediate in the synthesis of cephalosporin antibiotics. Decarbamyl cefuroxime is a degradation product of cefuroxime.

Cascaroside A is a useful organic compound for research related to life sciences and the catalog number is T124690.

Foscarbidopa is a prodrug of carbidopa, which is metabolised by alkaline phosphatase into carbidopa upon entering the body, thereby increasing dopamine levels. It is often used in combination with levodopa to treat motor complications in advanced Parkinson's disease.

M1/M4 muscarinic agonist 1 (Compound 41) is a selective muscarinic M4/M1 agonist with EC50 values of 14 nM for M4 receptors and 55 nM for M1 receptors. This compound is utilized in research related to psychiatric disorders, including schizophrenia and delusional disorders.

Compound 43, known as M1/M2/M4 muscarinic agonist 2, functions as an mAChR M1/M2/M4 agonist with respective EC50 values of 30 nM, 200 nM, and 6.2 nM.

Descarbamylnovobiocin is a derivative of novobiocin.

Muscarinic M4 modulator-1 is a positive allosteric modulator of the Muscarinic M4 receptor. It activates the muscarinic M4 receptor with allosteric efficacy (EC50) values of 14 nM in CHO-K1 cells and 3 nM in HEK293 cells. Muscarinic M4 modulator-1 exhibits antipsychotic-like activity and shows potential for research in psychiatric and/or neurological disorders.

Muscarinic M3 receptor antagonist-1 (Example 4) is an antagonist of the muscarinic acetylcholine receptor M3. It can be used for research on inflammatory or obstructive respiratory diseases.

Muscarinic M3 receptor antagonist-2 (Compound 30) is an antagonist of the muscarinic M3 receptor.

Muscarinic acetylcholine receptor agonist

Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.

Muscarine chloride is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.

Scaritoxin is a potent toxic substance isolated from poisonous fish.

Liriope muscari baily saponins C has an anti-thrombotic activity due to down-regulation of the increased mRNA expression levels of TF and IL-6.

Saponin C from Liriope muscari can be extracted from Liriope muscari, family Liliaceae, has antithrombotic activity and induces autophagy.

(±)-Muscarine chloride is the racemate of Muscarine chloride, a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].

Muscarinic toxin 7 (MT7) is a peptide exhibiting selective, noncompetitive antagonistic activity at the muscarinic M1 receptor [1].

Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57 for α1B, 8.13 for α1D, 8.49 for α2A, <6.5 for α2B, and 7.29 for α2C receptors. MT3 notably demonstrates significant adrenoceptor activity [1].

Compound 40 is a selective M1/M4 muscarinic antagonist with an IC50 of 19 nM for M1 receptors and 42 nM for M4 receptors [1].

Muscarine ((+)-Muscarine) tosylate, a prototype mAChR agonist, serves as a parasympathetic nervous system stimulant and is recognized for its toxic properties [1] [2].

Descarbonyl-lacosamide is a potential impurity in commercial lacosamide preparations. It is a degradation product that forms under acidic conditions.