TP1040 |
Calcitonin (salmon)
|
47931-85-1
|
98%
|
|
Calcitonin salmon, a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.
|
T6590 |
MK-3207 Hydrochloride
|
957116-20-0
|
98%
|
|
MK-3207 is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.
|
TP1257L |
Adrenomedullin (AM) (22-52), human acetate
|
|
98%
|
|
Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an adrenomedul...
|
T16107 |
ML230
|
1776055-05-0
|
98%
|
|
ML230 is a selective ATP-binding cassette (ABC) transporter ABCG2 inhibitor. It 36-fold selective for ABCG2 over ABCB1 (EC50s: 0.13 μM and 4.65 μM, respectively)...
|
T8682 |
Vazegepant hydrochloride
|
1414976-20-7
|
98%
|
|
Vazegepant is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.
|
TP2167 |
β-CGRP, human acetate
|
TP2167
|
98%
|
|
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor ...
|
TP1040L |
Calcitonin(salmon) Acetate(47931-85-1(free base))
|
TP1040L
|
98%
|
|
Calcitonin(salmon) Acetate, a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.
|
T12293L |
Olcegepant
|
204697-65-4
|
98%
|
|
Olcegepant is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4 pM for human C...
|
T13453 |
CGRP antagonist 1
|
1123757-49-2
|
98%
|
|
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study...
|
T17194 |
Ubrogepant
|
1374248-77-7
|
98%
|
|
Ubrogepant is a novel oral calcitonin gene-related peptide receptor antagonist in development for acute treatment of migraine.
|
TP1134L |
HCGRP-(8-37) acetate
|
TP1134L
|
98%
|
|
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.
|
T4610 |
Rimegepant
|
1289023-67-1
|
98%
|
|
BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.
|