Cat. No. | Product name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
TP1323 | CGRP 8-37 (rat) | 129121-73-9 | 99.28% |
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CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation. | ||||
T78540 | α-CGRP (mouse, rat) TFA | 98% |
|
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α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions and f... | ||||
T6590 | MK-3207 Hydrochloride | 957116-20-0 | 98% |
|
MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, an... | ||||
T16107 | ML230 | 1776055-05-0 | 98% |
|
ML230 is a selective ATP-binding cassette (ABC) transporter ABCG2 inhibitor. It 36-fold selective for ABCG2 over ABCB1 (EC50s: 0.13 μM and 4.65 μM, respectively)... | ||||
T8682 | Vazegepant hydrochloride | 1414976-20-7 | 99.56% |
|
Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study. | ||||
TP1257L | Adrenomedullin (AM) (22-52), human acetate | 99.42% |
|
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Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an adrenomedul... | ||||
TP2167 | β-CGRP, human acetate | TP2167 | 99.35% |
|
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor ... | ||||
T4610 | Rimegepant | 1289023-67-1 | 99.33% |
|
Rimegepant (BMS 927711) is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM. | ||||
TP1040L | Calcitonin(salmon) Acetate(47931-85-1(free base)) | TP1040L | 99.29% |
|
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 yea... | ||||
TP1134L | HCGRP-(8-37) acetate | TP1134L | 99.29% |
|
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor. | ||||
T12293L | Olcegepant | 204697-65-4 | 96.08% |
|
Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4 pM... | ||||
T13453 | CGRP antagonist 1 | 1123757-49-2 | 100% |
|
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study... | ||||
T17194 | Ubrogepant | 1374248-77-7 |
|
|
Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies. | ||||
T76682 | Galcanezumab | 1578199-75-3 | 98% |
Galcanezumab
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Galcanezumab is a humanized IgG4 monoclonal antibody targeting the CGRP ligand, which binds to the ligand calcitonin gene-related peptide. Galcanezumab can be us... | ||||
T76874 | Erenumab | 1582205-90-0 | 98% |
Erenumab
|
Erenumab is a whole-human monoclonal antibody. Erenumab inhibits calcitonin gene-related peptide (CGRP) receptors. Erenumab can be used to prevent migraine attac... | ||||
TP1040 | Calcitonin (salmon) | 47931-85-1 | 98% |
|
Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause. |