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Compounds

Cat No. Product Name
T27830 Lifarizine RS-87476 Calcium Channel
Lifarizine 是一种钙钠通道拮抗剂, 在简化的大鼠双血管闭塞存活模型中显示出神经保护活性。
T24873 TGX-115 TGX 115 PI3K
TGX-115是一种细胞渗透性和有效的PI 3-K 异构体p110β/p110δ抑制剂(对p110β IC50值为 0.13 μM, 对p110δ值为0.63 μM),是一种调节血小板粘附过程的酶,可抑制磷酸肌苷(PI)3-激酶,可用来治疗...
T4330 CaCCinh-A01 Chloride channel
CaCCinh-A01 是钙激活氯离子通道和TMEM16A 抑制剂,IC50值分别为 10 和 2.1 μM。
T11994 Melagatran Thrombin
Melagatran, a direct and orally active thrombin inhibitor, specifically inhibits thrombin without affecting other enzyme...
T28414 Piclozotan SUN-4057 5-HT Receptor
Piclozotan (anhydrous) 是一种 5-HT1A 受体激动剂,在短暂的大脑中动脉闭塞(t-MCAO)模型中表现出显着的神经保护活性,可以改善晚期帕金森病患者的运动并发症。
T1476 Pramipexole 普拉克索,SND 919 Dopamine Receptor
Pramipexole 是能够透过血脑屏障的 D2 型多巴胺受体的选择性激动剂,对 D2 型受体、D2、D3、D4亚型受体的Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1.3 nM。它可用于研究帕金森综合症和腿多动综合征。
T70540 Pinokalant LOE-908 SARS-CoV , TRP/TRPV Channel
Pinokalant 是一种新型非选性阳离子通道抑制剂。Pinokalant 在体内实验中可显著减少皮质梗死体积,可改善缺血半影区的代谢和电生理状态,可减少大鼠大脑中动脉闭塞后急性期磁共振图像上的病变大小。Pinokalant是一种潜在的S...
T23146 PHA 568487 free base PHA 568487 AChR
PHA 568487 free base 是一种选择性的 α7 烟碱乙酰胆碱受体激动剂,可用于减缓神经炎症。
T6951 Pramipexole dihydrochloride hydrate 普拉克索盐酸盐水合物,普拉克索,Mirapex,Pramipexole 2HCl Monohydrate Dopamine Receptor
Pramipexole 2HCl Monohydratee 是选择性的,具有血脑屏障 (BBB) 渗透性的 D2 型多巴胺受体激动剂,对 D2 型受体、D2、D3、D4亚型受体的 Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1....
T38063 N-Acetyl lysyltyrosylcysteine amide
N-Acetyl lysyltyrosylcysteine amide is a potent, reversible, specific, and non-toxic tripeptide inhibitor of myeloperoxi...
T2163 Dihydrocapsaicin 二氢辣椒素,CCRIS1589,8-Methyl-N-vanillylnonanamide,6,7-Dihydrocapsaicin Others , TRP/TRPV Channel
Dihydrocapsaicin 是一种天然来源的辣椒素,是TRPV1的选择性激动剂,同时可以增加 p-Akt 水平。它可以增强低温诱导的神经保护。
T35689 MTP 131 acetate Others
MTP 131 acetate 是一种小的线粒体靶向四肽。
T27897 LY 215490 LY215490,LY-215490
LY 215490 is a selective, competitive and systemically active antagonist of AMPA receptor. LY 215490 has neuroprotective...
T27351 Fostedil KB-944,KB 944,KB944,A 53986,BRN 3626546,A-53986
Fostedil is a calcium channel antagonist. KB-944 increased regional segment function in normal and ischemic regions and ...
T16902 SMND-309 Others
SMND-309 is a metabolite of salvianolic acid B. It also shows neuroprotective effects in cultured neurons and in permane...
T68814 GZN39838
GZN39838, also known as 6beta-Acetoxy-7alpha-hydroxyroyleanone is a natural blocker of Kv1.2 channels, not involving dir...
T41029 Streptokinase
Streptokinase is a bacterial protein that acts as a plasminogen activator, commonly employed in the investigation of blo...
T76987 Tarcocimab
Tarcocimab (OG1953) 是一种人源化抗VEGFA 单克隆抗体 (IgG1 型)。Tarcocimab 可用于视网膜静脉阻塞 (RVO) 和湿性老年性黄斑变性 (AMD) 的研究。
T35463 (±)14(15)-EET (±)14(15)-EET,(±)14,15-EpETrE,(±)14,15-EET
(±)14(15)-EET is a metabolite of arachidonic acid that is formed via epoxidation of arachidonic acid by cytochrome P450....
T36570 KUS121
KUS121 is a valosin-containing protein (VCP) modulator that inhibits VCP ATPase activity (IC50= 330 nM).1It inhibits cel...
Lifarizine
T27830
synonym: RS-87476
Target:
TGX-115
T24873
synonym: TGX 115
Target:
CaCCinh-A01
T4330
synonym:
Target:
Melagatran
T11994
synonym:
Target:
Piclozotan
T28414
synonym: SUN-4057
Target:
Pramipexole
T1476
synonym: 普拉克索,SND 919
Target:
Pinokalant
T70540
synonym: LOE-908
Target:
PHA 568487 free base
T23146
synonym: PHA 568487
Target:
Pramipexole dihydrochloride hydrate
T6951
synonym: 普拉克索盐酸盐水合物,普拉克索,Mirapex,Pramipexole 2HCl Monohydrate
Target:
N-Acetyl lysyltyrosylcysteine amide
T38063
synonym:
Target:
Dihydrocapsaicin
T2163
synonym: 二氢辣椒素,CCRIS1589,8-Methyl-N-vanillylnonanamide,6,7-Dihydrocapsaicin
Target:
MTP 131 acetate
T35689
synonym:
Target:
LY 215490
T27897
synonym: LY215490,LY-215490
Target:
Fostedil
T27351
synonym: KB-944,KB 944,KB944,A 53986,BRN 3626546,A-53986
Target:
SMND-309
T16902
synonym:
Target:
GZN39838
T68814
synonym:
Target:
Streptokinase
T41029
synonym:
Target:
Tarcocimab
T76987
synonym:
Target:
(±)14(15)-EET
T35463
synonym: (±)14(15)-EET,(±)14,15-EpETrE,(±)14,15-EET
Target:
KUS121
T36570
synonym:
Target:
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