a-estradiol — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T3378	Alpha-Estradiol	Alfatradiol,17α-Estradiol,Epiestrol,Epiestradiol	Estrogen/progestogen Receptor , Reductase , Endogenous Metabolite
	Alpha-Estradiol (Epiestradiol) is an estrogen that inhibits 5alpha-reductase and has potential in the study of androgenetic alopecia.
T7299	β-Estradiol 17-acetate	beta-estradiol 17-acetate,1,3,5(10)-Estratriene-3,17β-diol 17-acetate	Estrogen Receptor/ERR , Others
	β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) is a metabolite of estradiol.		Estrogen Receptor/ERR , Others
T2231	Estradiol dipropionate	17-Beta-Estradiol-3,17-Dipropionate	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Progesterone Receptor
	Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.
T0384	Estradiol benzoate	Benzoestrofol,Benzhormovarine,Benovocylin	Estrogen Receptor/ERR , Estrogen/progestogen Receptor
	Estradiol benzoate (Benzhormovarine) is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to the maintenance of fertility and secondary sexual characteristics in females.		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
T1048	Estradiol	E2,17β-Estradiol,17β-Oestradiol,β-Estradiol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	Estradiol (E2) is a naturally occurring steroidal sex hormone that is essential for female fertility and maintenance of secondary sexual characteristics. Estradiol upregulates IL-6 expression through estrogen receptor be...
T11235	Estradiol 3-sulfamate	ES-J 995,E2MATE,BLE 00084	Others
	.Estradiol 3-sulfamate inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor.		Others
T14577	Biotin-DADOO	EZ-Link Amine-PEO2-Biotin,Biotinyl-3,6-dioxaoctanediamine	Others
	Biotin-DADOO (Biotinyl-3,6-dioxaoctanediamine) is a biotinylation reagent that can be used to synthesize a biotin-estradiol conjugate(i.e., biotin-DADOO-estradiol) to develop a direct, broad-range enzyme immunoassay to m...		Others
T1424	Ethynyl estradiol	17α-Ethynylestradiol,Ethinyl Estradiol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is often used as the estrogenic component in ORAL CONTRACEPTIVES...
T13481	2-Methoxyestrone		Endogenous Metabolite
	2-Methoxyestrone is a methoxylated catechol estrogen and metabolite of estrone (pKa: 10.81).		Endogenous Metabolite
T11399	Giredestrant	GDC-9545	Estrogen Receptor/ERR , Estrogen/progestogen Receptor
	Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity. Giredestrant, a non-steroidal ER ligand,...		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
T10239	Acolbifene	EM-652,SCH 57068	Estrogen Receptor/ERR
	Acolbifene (SCH 57068) is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and ERβ. Acolbifene shows an anticarcinogenic property.		Estrogen Receptor/ERR
T16338	Norgestimate metabolite Norelgestromin	17-Deacetyl norgestimate,17-Deacylnorgestimate	Drug Metabolite
	Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate) is one of the active metabolites of norgestimate.It is a steroidal progestin used in contraceptive patches, where it is combined with the estrogen ethinyl es...		Drug Metabolite
T1571	Estriol	NSC-12169,Oestriol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , MRP , Endogenous Metabolite
	Estriol (Oestriol) is a hydroxylated metabolite of ESTRADIOL or ESTRONE that has a hydroxyl group at C3, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen. During PREGNANCY, a large amount of estriol is...
TJS0856	Dalbergin	6-Hydroxy-7-Methoxy-4-Phenylcoumarin	Others
	1. Dalbergin (6-Hydroxy-7-Methoxy-4-Phenylcoumarin) exhibits similar bone conserving effect against bone-loss as estradiol treatment, it as a therapeutic candidate against postmenopausal osteoporosis. 2. Dalbergin preven...		Others
T1009	Estrone	Oestrone,Fluoroethyl,Aquacrine	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	Estrone (Aquacrine) is an aromatized C18 steroid with a 3-hydroxyl group and a 17-ketone, a major mammalian estrogen. It is converted from ANDROSTENEDIONE directly, or from TESTOSTERONE via ESTRADIOL. In humans, it is pr...
T25048	Algestone acetophenide	Neolutin	Others
	Algestone acetophenide (Neolutin) is progesterone that used in estrus synchronization and has been evaluated as an injectable contraceptive in combination with estradiol enanthate. It is also used therapeutically as a to...		Others
T20681	Estramustine	NSC-89201,NSC 89201,LEO 275,LEO275,NSC89201,LEO-275	Microtubule Associated
	Estramustine (LEO-275) is a nitrogen mustard linked to estradiol, usually as phosphate. Estramustine has been used to treat prostatic neoplasms; also has radiation protective properties. Estramustine is selectively taken...		Microtubule Associated
T22794	G36	G-36	Estrogen Receptor/ERR
	G36 is a cell-permeable non-steroidal antagonist of GPER. G36 inhibits activation by either 17β-estradiol or the GPER-selective agonist G-1 (IC50 = 112 and 165 nM, respectively). G36 has no detectable binding activity to...		Estrogen Receptor/ERR
T40580	17β-Estradiol sulfate sodium	17β-Estradiol 3-sulfate sodium	Antibiotic
	17β-Estradiol sulfate sodium (17β-Estradiol 3-sulfate sodium) is a neuroactive estrogen with vasoprotective properties that inhibits the growth of Neisseria brasiliensis and disrupts aquatic ecosystems.		Antibiotic
T14344	Atrimustine	KM2210,Bestrabucil	Others
	Atrimustine is a conjugate of chlorambucil and β-estradiol benzoate. It has the antitumor activity.		Others