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Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling
MAPK Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination Others
Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library

Search Result

Search Results for "gpcr/g protein"

Libraries

GPCR Compound Library GPCR Compound Library Plus Serotonin Receptor-Targeted Compound Library Neuronal Signaling Compound Library Chemokine Inhibitor Library
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Compounds

Cat No. Product Name
T21874 CID 2745687 GPR
CID 2745687 是可逆的、特异性 GPR35竞争性拮抗剂（Ki:12.8 nM）。
T8329 AR 231453 GPR
AR 231453 是一种口服具有活性的、特异性的 GPR119激动剂。它能够刺激细胞增殖，改善胰岛 β 细胞的功能。
T3433 TUG-891 TUG891,TUG 891 GPR
TUG891 是一种选择性的长链游离脂肪酸受体 4 (FFA4/GPR120) 的激动剂。
T10843 CMF019 Apelin receptor
CMF019 是一种有效的小分子 Apelin receptor (APJ) 激动剂，具有 G protein 偏向性。 CMF019 在人，大鼠和小鼠中与 APJ 结合的 pKi 值分别为 8.58、8.49 和 8.71。CMF-019...
T9146 Ms48107 Benzenemethanol, 2-[4-amino-6-[[(4-phenoxyphenyl)methyl]amino]-1,3,5-triazin-2-yl]-3-fluoro- Others
MS48107 是 G 蛋白偶联受体 68 (GPR68) 的选择性正变构调节剂，对GPR68的选择性高于密切相关的神经递质转运蛋白，质子 GPCR 和 hERG 离子通道。它可以穿越过小鼠的血脑屏障。
T50088 N-phenylthiophene-2-carboximidamide Others
N-phenylthiophene-2-carboximidamide 是一种噻吩衍生物类的有机化合物，已被用于合成各种有机化合物，包括药物和农用化学品。它还可以作为蛋白酪氨酸激酶（PTKs）的抑制剂和G 蛋白偶联受体（GPCR）的配体发挥...
T27428 GP-1681 GP 1681,GP1681
GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection.
T26962 CBP-307 CBP307
CBP-307 is a selective second generation S1P1 (a G-protein coupled receptor -GPCR) modulator.
T10363 Arazine N-Acetyl-S-farnesyl-L-cysteine Others
Arazine 可以成为异戊二烯基半胱氨酸甲基转移酶的底物通过与异戊二烯化 G 蛋白或其受体位点竞争。 Arazine 是 G 蛋白和 GPCR 信号传导的细胞渗透性调节剂。
T11044 Dihydromunduletone DHM GPR
Dihydromunduletone (DHM) is a carotenoid derivative and selective strong adhesion G protein-coupled receptor (aGPCR) (GP...
TN5580 Rediocide A
Rediocide A, an insecticide, can inhibit calcium mobilization in Drosophila G-protein- coupled receptors (GPCR)s other t...
T73005 PF-07054894
PF-07054894 是一种有效的 CCR6拮抗剂。 PF-07054894 靶向 G 蛋白偶联受体 (GPCR)。 PF-07054894 可用于炎症性肠病的研究。
T63340 CCG-273220
CCG-273220 是 G 蛋白偶联受体 (GPCR) 激酶 5 (GRK5) 共价抑制剂 (IC50: 220 nM)。CCG-273220 可以共价结合GRK5亚家族特异性残基 Cys474 ，而对GRK5的选择性比 GRK2 高。
TMPY-04562 GRK2 Protein, Human, Recombinant (His & GST Tag)
G-protein coupled receptor kinase 2 (GRK2), also referred as Adrenergic, beta, receptor kinase 1 (ADRBK1), is a ubiquito...
T70468 MK-8666
MK-8666 is a partial GPCR (G-protein-coupled receptor) agonist that is coordinated with the action of GPR40. GPR40, also...
T69953 MK-8666 Tris
MK-8666 is a partial GPCR (G-protein-coupled receptor) agonist that is coordinated with the action of GPR40. GPR40, also...
TMPY-02837 GPR114 Protein, Human, Recombinant (hFc Tag)
GPR114 belongs to the G-protein coupled receptor 2 family. Members of this family share a common molecular architecture ...
T36578 Boc-Lys(Ac)-AMC
Commendamide (N-acyl-3-hydroxypalmitoyl-glycine) is a newly discovered GPCR G2A/GPR132 agonist (EC50=11.8 μM) that isola...
T36550 CAY10535
TPα and TPβ are two isoforms of the human TP receptor, the G protein-coupled receptor (GPCR) that mediates the actions o...
T36013 Lysophosphatidylcholines ​Lyso-Lecithins (egg)
Lysophosphatidylcholines are produced by hydrolysis of the fatty acid of phosphatidylcholine at either the sn-1 or sn-2 ...
CID 2745687
T21874
synonym:
Target:
AR 231453
T8329
synonym:
Target:
TUG-891
T3433
synonym: TUG891,TUG 891
Target:
CMF019
T10843
synonym:
Target:
ms48107
T9146
synonym: Benzenemethanol, 2-[4-amino-6-[[(4-phenoxyphenyl)methyl]amino]-1,3,5-triazin-2-yl]-3-fluoro-
Target:
N-phenylthiophene-2-carboximidamide
T50088
synonym:
Target:
GP-1681
T27428
synonym: GP 1681,GP1681
Target:
CBP-307
T26962
synonym: CBP307
Target:
Arazine
T10363
synonym: N-Acetyl-S-farnesyl-L-cysteine
Target:
Dihydromunduletone
T11044
synonym: DHM
Target:
Rediocide A
TN5580
synonym:
Target:
PF-07054894
T73005
synonym:
Target:
CCG-273220
T63340
synonym:
Target:
GRK2 Protein, Human, Recombinant (His & GST Tag)
TMPY-04562
synonym:
Target:
MK-8666
T70468
synonym:
Target:
MK-8666 Tris
T69953
synonym:
Target:
GPR114 Protein, Human, Recombinant (hFc Tag)
TMPY-02837
synonym:
Target:
Boc-Lys(Ac)-AMC
T36578
synonym:
Target:
CAY10535
T36550
synonym:
Target:
Lysophosphatidylcholines
T36013
synonym: ​Lyso-Lecithins (egg)
Target:
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