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Search Results for " kainate "

20

Compounds

Cat No. Product Name Synonyms Targets
T8458 CNQX disodium iGluR
CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.
T7178 CNQX FG9065 GluR , iGluR
CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)
T16963 SYM 2081 iGluR
SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude.
T21584 CP 465022 iGluR
CP 465022 hydrochloride is a potent, and selective noncompetitive antagonist of AMPA receptor with anticonvulsant activity. CP 465022 hydrochloride inhibits Kainate-induced response with an IC50 of 25 nM in rat cortical ...
T13456 (S)-Willardiine (-)-Willardiine,L-willardiine,Willardiine iGluR
(S)-Willardiine (L-willardiine) is present in the seeds of Acacia and Mimosa. (S)-Willardiine is an AMPA/kainate receptor agonist (EC50 = 44.8 μM).
T7304 DNQX FG 9041 GluR , iGluR
DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)
T20571 Cis-PDA cis PDA GluR , NMDAR , iGluR
cis-PDA (cis PDA) is a general ionotropic receptor antagonist. cis-PDA acts by blocking NMDA, AMPA, and kainate-mediated responses.
T31208 Dasolampanel NGX-426,NGX 426,NGX426 GluR , iGluR
Dasolampanel (NGX-426) is an orally available ionotropic glutamate receptor AMPA and Kainate receptor antagonist for the study of chronic pain disorders, including neuropathic pain and migraine.
T6134 IEM 1754 2HBr IEM 1754 dihydrobromide GluR
IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.
T27949 LY382884 LY-382884,LY 382884 GluR
LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade of mossy fibre LTP induction.
T0313 Evans blue Direct Blue 53,C.I. 23860 GluR
Evans blue (C.I. 23860) is an azo dye, inhibits L-glutamate uptake via the membrane-bound excitatory amino acid transporter (EAAT).
T8459 DNQX disodium salt DNQX Disodium NMDAR , iGluR
DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor
T0675 Topiramate RWJ 17021,McN 4853 Potassium Channel , Calcium Channel , GABA Receptor , Sodium Channel , GluR , Carbonic Anhydrase , iGluR
Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures. Topiramate has been rarely associated with hepatic injury and largely when used in combination ...
T23489 UBP301 UBP 301 Others
UBP301 is a kainate receptor antagonist.
T23295 (S)-(-)-5-Iodowillardiine Others
hGluR5 kainate receptor agonist
T23487 UBP-282 Others
AMPA and kainate receptor antagonist
T11522 GYKI 52466 dihydrochloride Others
GYKI 52466 dihydrochloride is orally active and non-competitive kainate- and AMPA-activated currents antagonist (IC50s: 7.5 μM and 11 μM). It is inactive against NMDA or γ-aminobutyric acid responses. It is a muscle rela...
T22546 UBP316 ACET Others
GluR5-containing kainate receptor antagonist
T23088 NS 3763 Others
NS 3763 is a kainate receptor antagonist.
T23488 UBP 296 Others
GluR5-subunit containing kainate receptor antagonist
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TargetMol