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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T8458 | CNQX disodium | iGluR | |
CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures. | |||
T7178 | CNQX | FG9065 | GluR , iGluR |
CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively) | |||
T16963 | SYM 2081 | iGluR | |
SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude. | |||
T21584 | CP 465022 | iGluR | |
CP 465022 hydrochloride is a potent, and selective noncompetitive antagonist of AMPA receptor with anticonvulsant activity. CP 465022 hydrochloride inhibits Kainate-induced response with an IC50 of 25 nM in rat cortical ... | |||
T13456 | (S)-Willardiine | (-)-Willardiine,L-willardiine,Willardiine | iGluR |
(S)-Willardiine (L-willardiine) is present in the seeds of Acacia and Mimosa. (S)-Willardiine is an AMPA/kainate receptor agonist (EC50 = 44.8 μM). | |||
T7304 | DNQX | FG 9041 | GluR , iGluR |
DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively) | |||
T20571 | Cis-PDA | cis PDA | GluR , NMDAR , iGluR |
cis-PDA (cis PDA) is a general ionotropic receptor antagonist. cis-PDA acts by blocking NMDA, AMPA, and kainate-mediated responses. | |||
T31208 | Dasolampanel | NGX-426,NGX 426,NGX426 | GluR , iGluR |
Dasolampanel (NGX-426) is an orally available ionotropic glutamate receptor AMPA and Kainate receptor antagonist for the study of chronic pain disorders, including neuropathic pain and migraine. | |||
T6134 | IEM 1754 2HBr | IEM 1754 dihydrobromide | GluR |
IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM. | |||
T27949 | LY382884 | LY-382884,LY 382884 | GluR |
LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade of mossy fibre LTP induction. | |||
T0313 | Evans blue | Direct Blue 53,C.I. 23860 | GluR |
Evans blue (C.I. 23860) is an azo dye, inhibits L-glutamate uptake via the membrane-bound excitatory amino acid transporter (EAAT). | |||
T8459 | DNQX disodium salt | DNQX Disodium | NMDAR , iGluR |
DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor | |||
T0675 | Topiramate | RWJ 17021,McN 4853 | Potassium Channel , Calcium Channel , GABA Receptor , Sodium Channel , GluR , Carbonic Anhydrase , iGluR |
Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures. Topiramate has been rarely associated with hepatic injury and largely when used in combination ... | |||
T23489 | UBP301 | UBP 301 | Others |
UBP301 is a kainate receptor antagonist. | |||
T23295 | (S)-(-)-5-Iodowillardiine | Others | |
hGluR5 kainate receptor agonist | |||
T23487 | UBP-282 | Others | |
AMPA and kainate receptor antagonist | |||
T11522 | GYKI 52466 dihydrochloride | Others | |
GYKI 52466 dihydrochloride is orally active and non-competitive kainate- and AMPA-activated currents antagonist (IC50s: 7.5 μM and 11 μM). It is inactive against NMDA or γ-aminobutyric acid responses. It is a muscle rela... | |||
T22546 | UBP316 | ACET | Others |
GluR5-containing kainate receptor antagonist | |||
T23088 | NS 3763 | Others | |
NS 3763 is a kainate receptor antagonist. | |||
T23488 | UBP 296 | Others | |
GluR5-subunit containing kainate receptor antagonist |