Shopping Cart

Remove All
Your shopping cart is currently empty

SYM 2081

Name: SYM 2081
Brand: TargetMol
SKU: T16963
Price: 87 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T16963Cas No. 31137-74-3

SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude.

SYM 2081

🥰Excellent

Purity: 99.59%

Catalog No. T16963Cas No. 31137-74-3

SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude.

Pack Size	Price	Availability
1 mg	$87	In Stock
5 mg	$213	In Stock
10 mg	$313	In Stock
25 mg	$533	In Stock
50 mg	$768	In Stock
100 mg	$1,080	In Stock
500 mg	$2,160	In Stock

Add to Cart

Add to Quotation

Bulk & Custom

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Purity:99.59%

Resource Download

COA HPLC HNMR

Product Introduction

Bioactivity

Description	SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude.
Targets&IC50	Kainate receptor:35 nM

Chemical Properties

Molecular Weight	161.16
Formula	C₆H₁₁NO₄
Cas No.	31137-74-3
Smiles	[C@@H](C[C@@H](C(O)=O)N)(C(O)=O)C
Relative Density.	1.3482 g/cm3 (Estimated)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: 45.0 mg/mL (279.2 mM), Sonication is recommended.

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
1 mM	6.2050 mL	31.0251 mL	62.0501 mL	310.2507 mL
5 mM	1.2410 mL	6.2050 mL	12.4100 mL	62.0501 mL
10 mM	0.6205 mL	3.1025 mL	6.2050 mL	31.0251 mL
20 mM	0.3103 mL	1.5513 mL	3.1025 mL	15.5125 mL
50 mM	0.1241 mL	0.6205 mL	1.2410 mL	6.2050 mL
100 mM	0.0621 mL	0.3103 mL	0.6205 mL	3.1025 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc