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TSH Receptor

The thyrotropin receptor (or TSH receptor) is a receptor (and associated protein) that responds to thyroid-stimulating hormone (also known as "thyrotropin") and stimulates the production of thyroxine (T4) and triiodothyronine (T3). The TSH receptor is a member of the G protein-coupled receptor superfamily of integral membrane proteins and is coupled to the Gs protein.
Cat. No. Product name CAS No. Purity Chemical Structure
T5383 D3-βArr 662164-09-2 99.43%
D3-βArr is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct TSHR activation.
T12192 NCGC00229600 1338824-20-6 99.27%
NCGC00229600 is an allosteric inverse thyrotropin receptor (TSHR) agonist. NCGC00229600 inhibits both TSH and stimulating antibody activation of TSHRs endogenous...
T13216 TSHR antagonist S37 1217616-61-9 98.35%
TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).
T12073 ML-109 1186649-91-1 98.14%
ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)
T29087 VA-K-14 hydrochloride 1171341-19-7 98.01%
VA-K-14 hydrochloride(VAK14 HCl) is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits TSHR stimulation by serum and monoclonal TSH...
D3-βArr
T5383
D3-βArr is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct TSHR activation.
NCGC00229600
T12192
NCGC00229600 is an allosteric inverse thyrotropin receptor (TSHR) agonist. NCGC00229600 inhibits both TSH and stimulating antibody activation of TSHRs endogenous...
TSHR antagonist S37
T13216
TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).
ML-109
T12073
ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)
VA-K-14 hydrochloride
T29087
VA-K-14 hydrochloride(VAK14 HCl) is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits TSHR stimulation by serum and monoclonal TSH...