Cat. No. | Product name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T4170 | PKM2-IN-1 | 94164-88-2 | 98% |
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PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2. | ||||
T4223 | Mitapivat | 1260075-17-9 | 98% |
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Mitapivat, also known as PKM2 activator 1020 is a PKM2 activator (pyruvate kinase activator) for the treatment of pyruvate kinase deficiency. | ||||
T67900 | WAY-332616 | 904457-46-1 | 98% |
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WAY-332616 is a inhibitor of pyruvate kinase. | ||||
T12499 | PKR-IN-2 | 1628428-01-2 | 98% |
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PKR-IN-2 is a activator of pyruvate kinase (PKR). | ||||
T6816 | DASA-58 | 1203494-49-8 | 98% |
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DASA-58 is a specific and potent Pyruvate kinase M2 (PKM2) activator. | ||||
T7214 | TEPP-46 | 1221186-53-3 | 98% |
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ML265 is a potent PKM2 activator (AC50 : 92 nM) showing little or no effect on PKM1, PKL and PKR,induces tetramerization and reduces tumor formation and size in ... | ||||
T1125 | Shikonin | 517-89-5 | 98% |
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Shikonin is an TMEM16A chloride channel inhibitor (IC50: 6.5 μM). Shikonin is also a selective PKM2 inhibitor and can also suppress activation of the NF-κB pathw... | ||||
T8363 | DL-Serine | 302-84-1 | 98% |
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DL-Serine is a non-essential amino acid and a natural ligand and allosteric activator of pyruvate kinase M2. | ||||
T0745 | Disodium monofluorophosphate | 10163-15-2 | 98% |
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Sodium Monofluorophosphate is a competitive inhibitor of pyruvate kinase and alkaline phosphatase, which also irreversibly inhibits phosphorylase phosphatase. | ||||
T62758 | PKM2 activator 2 | 1186660-06-9 | 98% |
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PKM2 activator 2 is a pyruvate kinase M2 (PKM2) activator with an AC 50 value of 66 nM.PKM2 activator 2 has anti-tumor proliferative properties and attenuates th... |