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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T40712 | Diethyl fumarate | Others | |
Diethyl fumarate is a decomposition product of the pesticide Malathion. Diethyl fumarate causes nonimmune contact urticaria on the skin. | |||
T1532 | Pidotimod | Others , Antibacterial | |
Pidotimod is a synthetic dipeptide with immunomodulatory properties. | |||
T7893 | Bepotastine | Bepotastine free base | Others , Histamine Receptor |
Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis. | |||
T6242 | Rupatadine Fumarate | Rinialer,Rupafin,Alergoliber | PAFR , Autophagy , Histamine Receptor |
Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM. | |||
T6405 | Bepotastine Besilate | Talion,TAU 284,Bepreve,Bepotastine Beslilate | Histamine Receptor |
Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7). | |||
T2335 | Ebastine | Ebastel,LAS-W 090,Ebastin,Kestine,RP64305 | Histamine Receptor |
Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine. It does not penetrate the blood-brain barrier and thus allows an effective block of the H1 receptor in peripheral tiss... | |||
T20444 | Hexyl nicotinate | AI3 15769,AI3-15769,AI315769 | Others |
Hexyl nicotinate (AI3 15769) is a cutaneous vasodilator and can be used in research on non-immunologic contact urticaria on the scalp, face, and back. | |||
T1553 | Chlorpheniramine maleate | NCI-C55265,Chlorphenamine maleate | Histamine Receptor |
Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma. | |||
T1470 | Fexofenadine hydrochloride | Terfenidine carboxylate hydrochloride,MDL-16455 hydrochloride,Telfast,Fexofenadine HCl,Allegra,MDL 16455A | Histamine Receptor |
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis, angioedema and chronic urticaria. | |||
T1097 | Loratadine | SCH 29851,Loratidine | Influenza Virus , Histamine Receptor |
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical antihistamines (HISTAMINE H1 ANTAGONISTS) it lacks central ne... | |||
T0785 | Dexchlorpheniramine Maleate | S-(+)-Chlorpheniramine maleate salt | Dopamine Receptor , 5-HT Receptor , Norepinephrine , Histamine Receptor |
Dexchlorpheniramine Maleate (S-(+)-Chlorpheniramine maleate salt) is an antihistamine with anticholinergic properties used to treat allergic conditions such as hay fever or urticaria. It is the pharmacologically active d... | |||
T0053 | Hydroxyzine Pamoate | Hydroxyzine embonate,Bobsule,Equipose | Histamine Receptor |
Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIRIZINE, it does ca... | |||
T22354 | Levocetirizine Dihydrochloride | Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride | Histamine Receptor |
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydro... | |||
T16730 | Remibrutinib | BTK | |
Remibrutinib inhibits BTK activity with an IC50 value of 0.023 μM in blood. Remibrutinib is an effective and orally active Bruton tyrosine kinase inhibitor (IC50: 1 nM). Remibrutinib has the potential for Chronic urticar... | |||
T21390 | Fexofenadine | Carboxyterfenadine,Telfast,MDL 16.455,Allegra | Histamine Receptor |
Fexofenadine (Carboxyterfenadine), an antihistamine pharmaceutical drug, is used to treat allergy symptoms, such as nasal congestion, hay fever, and urticaria. Compared to first-generation antihistamines, Fexofenadine is... | |||
T1278 | Astemizole | Laridal,Histaminos,Paralergin | Potassium Channel , Histamine Receptor |
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re... | |||
T0089 | Cetirizine dihydrochloride | P071,UCB P071,Cetirizine DiHCl | Histamine Receptor |
Cetirizine dihydrochloride (UCB P071) is an effective second-generation histamine H1 antagonist that is potent in the therapy of allergic rhinitis, confirmed urticaria, and pollen-induced asthma. Unlike other conventiona... | |||
T2200 | Hydroxyzine dihydrochloride | Hydroxyzine 2HCl | Histamine Receptor |
Hydroxyzine dihydrochloride (Hydroxyzine 2HCl) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIR... | |||
T21247 | Carbinoxamine | Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine | |
Carbinoxamine, an anticholinergic and antihistamine agent, is used for hay fever, angioedema, vasomotor rhinitis, mild urticaria, dermatographism and allergic conjunctivitis. It is a histamine antagonist, specifically an... | |||
T21112 | Triprolidine hydrochloride | 295 C 51,Pro-Entra,Entra,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil | |
Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria. |