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Search Result

Search Results for "lysophospholipid receptor"

Compounds

Cat No. Product Name
T17183 TY-52156 S1P Receptor , LPL Receptor
TY-52156 是一种选择性S1P3受体拮抗剂，Ki 值为 110 nM。
T2000 AM095 LPL Receptor , LPA Receptor
AM095 是一种有效的 LPA1 受体拮抗剂，对重组人或小鼠 LPA1 的 IC50 值分别为 0.98 和 0.73 μM。
T7360 GSK2018682 S1P Receptor , LPL Receptor
GSK2018682 是 1-磷酸鞘氨醇受体S1P1和S1P5激动剂，pEC50值分别为 7.7 和 7.2，可用于多发性硬化的研究。
T9464 CYM50358 LPL Receptor
CYM50358 是选择性的S1PR4拮抗剂，IC50值为 25 nM，可用于流感研究。
T7393 ONO-7300243 LPL Receptor , LPA Receptor
ONO-7300243 是溶血磷脂酸受体 1 (LPA1)拮抗剂，IC50为 0.16 μM。
TQ0227 Etrasimod APD334 LPL Receptor , S1P Receptor
Etrasimod 是一种特异性和口服的S1P1受体拮抗剂，在CHO 细胞中的IC50值为1.88 nM。
T12821 S1PR1 modulator 1 LPL Receptor
S1PR1 modulator 1 是 S1PR1 的特异性抑制剂，pIC50 为 7.6。
T15629 JTE-013 Apoptosis , LPL Receptor , S1P Receptor
JTE-013 是一种选择性S1P2拮抗剂。它抑制放射性标记的 S1P 与人和大鼠 S1P2的特异性结合，IC50分别为 17 nM 和 22 nM。
T12086 Mocravimod hydrochloride KRP-203 LPL Receptor , Others
Mocravimod hydrochloride 是 1-磷酸鞘氨醇受体 1 型 (S1PR1) 的有效和口服活性激动剂。
T22703 CYM-5520 CYM 5520 LPL Receptor , S1P Receptor
CYM 5520 是一种选择性的变构鞘氨醇 1-磷酸受体 2 (S1PR2) 激动剂，EC50为 480 nM。它可以在 S1PR2 受体中与 S1P 结合，可用于骨质疏松症研究。
T28169 NIBR-0213 NIBR 0213 LPL Receptor
NIBR-0213 是S1P1选择性拮抗剂，有抗实验性自身免疫性脑脊髓炎的作用。在 GTPγ35S 试验中，它作用于人和大鼠S1P1的IC50分别为 2.0 nM 和 2.3 nM。
T22834 H2L 5765834 LPA Receptor , LPL Receptor
H2L 5765834 是溶血磷脂酸受体 LPA1、LPA3和 LPA5拮抗剂，IC50值分别为 94、752 和 463 nM。
T3258 Ponesimod ACT-128800 S1P Receptor , LPL Receptor
Ponesimod 是一种选择性 S1P1可口服激动剂，在放射性配体结合试验中的 IC50值为 6 nM。它可高效激活 S1P1介导的信号转导，EC50为5.7 nM。它可预防淋巴细胞介导的组织炎症，具有潜在的免疫调节活性。
T6347 Ki16198 LPA Receptor , LPL Receptor
Ki16198 是一种可口服的 LPA 受体拮抗剂，是 Ki16425 的甲酯衍生物。它抑制 LPA1 和 LPA3 诱导的肌醇磷酸的Ki 值分别为 0.34 和 0.93 μM，可用于胰腺癌发生和转移的研究。
T6108 Ki16425 Debio 0719 LPA Receptor , LPL Receptor
Ki16425 是一种竞争性、有效和可逆的 LPA1、LPA2 和 LPA3 拮抗剂，Ki 分别为 0.34、6.5 和 0.93 μM。它可抑制LPA 诱导的 HEK293A 细胞中 YAP/TAZ 的去磷酸化，降低LPA 诱导的 p42...
T22101 ML-031 S1P Receptor
ML-031 是鞘氨醇 1-磷酸受体 2 (S1PR2)的选择性激动剂，其IC50=1.0 μM，EC50=1.03 μM。它可用于癌症疾病的研究。
T10305 Amiselimod hydrochloride MT-1303 hydrochloride S1P Receptor , LPL Receptor
Amiselimod hydrochloride 是一种鞘氨醇 1-磷酸受体 1 (S1P1) 调节剂。
T15032 CYM50308 LPL Receptor , S1P Receptor
CYM50308 是选择性和高亲和力的鞘氨醇-1-磷酸受体 4 激动剂，EC50为 56 nM。它对 S1P4-R 的选择性比 S1P5-R 高 37 倍。
T4031 S1p receptor agonist 1 S1p-receptor-agonist-1 LPL Receptor , S1P Receptor
S1p receptor agonist 1 是有口服活性的S1P 受体激动剂，具有诱导 S1P1 内化的活性，EC50为9.83 nM。它有潜力用于关节炎和实验性自身免疫性脑炎)的相关研究，详细信息来自专利 WO2015039587A1 ...
T3961 CYM-5541 CID-17253208,CYM 5541,ML249 LPL Receptor , S1P Receptor
CYM 5541是一种选择性的S1P3受体变构激动剂，EC50值在72至132 nM 之间。
TY-52156
T17183
synonym:
Target:
AM095
T2000
synonym:
Target:
GSK2018682
T7360
synonym:
Target:
CYM50358
T9464
synonym:
Target:
ONO-7300243
T7393
synonym:
Target:
Etrasimod
TQ0227
synonym: APD334
Target:
S1PR1 modulator 1
T12821
synonym:
Target:
JTE-013
T15629
synonym:
Target:
Mocravimod hydrochloride
T12086
synonym: KRP-203
Target:
CYM-5520
T22703
synonym: CYM 5520
Target:
NIBR-0213
T28169
synonym: NIBR 0213
Target:
H2L 5765834
T22834
synonym:
Target:
Ponesimod
T3258
synonym: ACT-128800
Target:
Ki16198
T6347
synonym:
Target:
Ki16425
T6108
synonym: Debio 0719
Target:
ML-031
T22101
synonym:
Target:
Amiselimod hydrochloride
T10305
synonym: MT-1303 hydrochloride
Target:
CYM50308
T15032
synonym:
Target:
S1p receptor agonist 1
T4031
synonym: S1p-receptor-agonist-1
Target:
CYM-5541
T3961
synonym: CID-17253208,CYM 5541,ML249
Target:
1 2
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