T61969 |
AChE/BChE-IN-10
|
|
98%
|
|
AChE/BChE-IN-10 is a potent dual inhibitor of AChE and BChE with IC50 values of 0.176, and 0.47 μM, respectively. AChE/BChE-IN-10 exhibits good blood brain barri...
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T62360 |
AChE-IN-26
|
|
98%
|
|
AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).
|
T60739L |
Y13g dihydrochloride
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T60739L
|
98%
|
|
Y13g dihydrochloride is a potent inhibitor of interleukin 6 (IL-6) and acetylcholinesterase (AChE) (both targets of Alzheimer's disease (AD) progression are rela...
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T60891 |
AChE/BChE/MAO-B-IN-1
|
2416910-82-0
|
98%
|
|
AChE/BChE/MAO-B-IN-1 is a reversible, non-time-dependent inhibitor of AChE, BChE and MAO-B that crosses the blood-brain barrier and exhibits inhibitory effects o...
|
T77560 |
2-Amino-4-(4-chlorophenyl)thiazole
|
2103-99-3
|
98%
|
|
2-AMINO-4-(4-CHLOROPHENYL)THIAZOLE is a 2-aminothiazole derivative. 2-AMINO-4-(4-CHLOROPHENYL)THIAZOLE inhibited hCA I, hCA II, AChE and BChE with Ki values of 0...
|
T68084 |
Icopezil
|
145508-78-7
|
98%
|
|
Icopezil is a small molecule acetylcholinesterase in (AChE) inhibitor for the treatment of neurological disorders and can be used in the study of Alzheimer's dis...
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T32535 |
Ladostigil
|
209394-27-4
|
98%
|
|
Ladostigil is an orally active dual inhibitor of cholinesterase and brain-selective monoamine oxidase (MAO) with inhibitory effects on MAO-B and AChE, with IC50 ...
|
TN2217 |
Sophoflavescenol
|
216450-65-6
|
98%
|
|
Sophoflavescenol is a mixed inhibitor of PDE5 with a K(i) value of 0.005 microM. Sophoflavescenol has antioxidant, anti-inflammatory, and apoptotic effects , the...
|
T13446 |
(S)-Rivastigmine D6 tartrate
|
194930-00-2
|
98%
|
|
(R)-Rivastigmine D6 tartrate is the deuterium labeled (R)-Rivastigmine, and is an inhibitor of cholinesterase.
|
T15949 |
Mahanimbine
|
21104-28-9
|
98%
|
|
Mahanimbine is found in the roots, leaves and stems of Murraya koenigii and is an orally active alkaloid extracted from Murraya koenigii. Bifidobacterium bifidum...
|
T14194 |
β-NETA
|
31059-54-8
|
98%
|
|
α-NETA is a stable, noncompetitive, slowly reversible choline acetyltransferase (ChAT) inhibitor with an IC50 of 9 μM and is a potent chemokine-like receptor-1 (...
|
TN2131 |
Questin
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3774-64-9
|
98%
|
|
Questin is an antimicrobial agent derived from Aspergillus florescens with an antimicrobial activity profile that inhibits V. harveyi, V. anguillarum, V. cholera...
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T8306 |
Epiberberine chloride
|
889665-86-5
|
98%
|
|
Epiberberine chloride is an alkaloid isolated from Coptis chinensis, acts as a potent AChE and BChE inhibitor, and a non-competitive BACE1 inhibitor (IC50s: 1.07...
|
TN1858 |
Leptomerine
|
22048-97-1
|
98%
|
|
Leptomerine (IC50 = 2.5 mM) shows potent anticholinesterasic activity.
|
T2227 |
Hemicholinium 3
|
312-45-8
|
98%
|
|
Hemicholinium-3 is a potent and selective choline uptake blocker.
|
T3819 |
Ursolic acid acetate
|
7372-30-7
|
98%
|
|
Acetylursolic acid has cytotoxic activity, antimalarial activity, antitumor and anticancer activities. Acetylursolic acid has NO production inhibitory activities...
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TN1124 |
Neoeriocitrin
|
13241-32-2
|
98%
|
|
Neoeriocitrin is a natural product isolated from Drynaria Rhizome, shows activity on proliferation and osteogenic differentiation in MC3T3-E1. Neoeriocitrin is a...
|
T0998 |
Diazinon
|
333-41-5
|
98%
|
|
Diazinon is a thiophosphoric acid ester, functioning as a nonsystemic organophosphate insecticide that effectively targets and controls a variety of pests includ...
|
T6478 |
Donepezil Hydrochloride
|
120011-70-3
|
98%
|
|
Donepezil is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).
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T2191 |
Tacrine hydrochloride (hydrate)
|
206658-92-6
|
98%
|
|
Tacrine hydrochloride hydrate is a cholinesterase inhibitor that crosses the blood-brain barrier. Tacrine has been used to counter the effects of muscle relaxant...
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